GLPBio

Histamine Receptor

Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.

Products Related to Histamine Receptor(243)

  • GC37959 structure
    GC37959Zaltidine
    CAS: 85604-00-8
    Purity: >99.00%

    Zaltidine(CP-57361) is a H2-receptor antagonist, which has the antisecretory action.

  • GC38450 structure
    GC38450LML134
    CAS: 1542135-76-1
    Purity: >99.50%

    LML134 (compound 18b) is an orally active and high selective Histamine 3 receptor (H3R) inverse agonist with Kis of 0.3 nM and 12 nM for hH3R cAMP and hH3R bdg.

  • GC38558 structure
    GC38558PF-03654746 Tosylate
    CAS: 1039399-17-1
    Purity: >99.50%

    PF-03654746 Tosylate is a potent and selective histamine H3 receptor antagonist with high brain penetration.

  • GC39108 structure
    GC39108Panaxydol
    CAS: 72800-72-7
    Purity: >70.00%

    Panaxydol, a C17-polyacetylene from Panax ginseng roots, exhibits cytotoxic and antimicrobial activities.

  • GC39378 structure
    GC39378Emedastine
    CAS: 87233-61-2
    Purity: >98.00%

    Emedastine is an orally active, selective and high affinity histamine H1 receptor antagonist with a Ki value of 1.3 nM.

  • GC39479 structure
    GC39479Bepotastine
    CAS: 125602-71-3
    Purity: >98.00%

    Bepotastine is a non-sedating, orally active second-generation histamine H1 receptor antagonist with higher selectivity than H3 receptors, α1, α2 and β adrenergic receptors, dopamine D2 receptors, serotonin 5-HT2 receptors, vagus nerve acetylcholine receptors, and benzodiazepine receptors.

  • GC39735 structure
    GC39735Triprolidine hydrochloride monohydrate
    CAS: 6138-79-0
    Purity: >99.50%

    Triprolidine hydrochloride monohydrate, a first-generation antihistamine, is an oral active histamine H1 antagonist.

  • GC41715 structure
    GC41715(R)-Cetirizine (hydrochloride)
    CAS: 130018-87-0
    Purity: >99.50%

    (R)-Cetirizine (hydrochloride) is a selective, potent, oral histamine H1 receptor antagonist.

  • GC43353 structure
    GC43353Cyproheptadine (hydrochloride hydrate)
    CAS: 41354-29-4
    Purity: >99.00%

    Cyproheptadine (hydrochloride hydrate) is an antihistamine and is an antagonist of serotonin and histamine2.

  • GC43427 structure
    GC43427Dexchlorpheniramine (maleate)
    CAS: 2438-32-6
    Purity: >98.00%

    Dexchlorpheniramine is a histamine H1 receptor antagonist with a pA2 value of 9.36 in guinea pig ileal tissue in vitro.

  • GC43598 structure
    GC43598Emedastine (fumarate)
    CAS: 87233-62-3
    Purity: >98.00%

    Emedastine (fumarate) is an orally active, selective and high affinity histamine H1 receptor antagonist with a Ki value of 1.3 nM.

  • GC44360 structure
    GC44360Nedocromil (sodium salt)
    CAS: 69049-74-7
    Purity: >98.00%

    Nedocromil (sodium salt) suppresses the action or formation of multiple mediators, including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).

  • GC46185 structure
    GC46185Nimbin
    CAS: 5945-86-8
    Purity: >98.00%

    A limonoid with diverse biological activities

  • GC48835 structure
    GC48835Diphenylpyraline
    CAS: 147-20-6
    Purity: >95.00%

    A histamine H 1 receptor antagonist

  • GC48892 structure
    GC48892NSC 19005
    CAS: 5452-87-9
    Purity: >95.00%

    NSC 19005 (NSC19005) is an impurity of Betahistine.

  • GC50405 structure
    GC50405JNJ 39758979 dihydrochloride
    Purity: >98%

    High affinity and selective histamine H4 antagonist; orally bioavailable

  • GC60072 structure
    GC60072Betahistine
    CAS: 5638-76-6
    Purity: >98.00%

    Betahistine is an orally active histamine H1 receptor agonist and a H3 receptor antagonist.

  • GC60563 structure
    GC60563Acrivastine D7
    CAS: 172165-56-9
    Purity: >98%

    Acrivastine D7 (BW825C D7) is a deuterium labeled Acrivastine.

  • GC60641 structure
    GC60641Betahistine mesylate
    CAS: 54856-23-4
    Purity: >98.00%

    Betahistine mesylate is an orally active histamine H1 receptor agonist and a H3 receptor antagonist.

  • GC60691 structure
    GC60691Cetirizine Impurity C
    CAS: 83881-59-8
    Purity: >98%

    Cetirizine Impurity C is an impurity of Cetirizine.

  • GC60709 structure
    GC60709Cinnarizine D8
    CAS: 1185242-27-6
    Purity: >98%

    An internal standard for the quantification of cinnarizine

  • GC60791 structure
    GC60791Doxepin D3 Hydrochloride
    CAS: 347840-07-7
    Purity: >98%

    Doxepin D3 Hydrochloride is a deuterium labeled Doxepin Hydrochloride.

  • GC60924 structure
    GC60924Hydroxyzine D8
    CAS: 1189480-47-4
    Purity: >98%

    Hydroxyzine D8 is deuterium labeled Hydroxyzine.

  • GC61256 structure
    GC61256Rupatadine D4 fumarate
    CAS: 1795153-63-7
    Purity: >98%

    Rupatadine D4 fumarate (UR-12592 D4 fumarate) is a deuterium labeled Rupatadine fumarate.