GLPBio

Histamine Receptor

Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.

Products Related to Histamine Receptor(243)

  • GC31897 structure
    GC31897Pirolate (CP-32387)
    CAS: 55149-05-8
    Purity: >98%

    Pirolate (CP-32387) is a histamine H1 receptor antagonist.

  • GC31994 structure
    GC31994CI-949
    CAS: 104961-19-5
    Purity: >98%

    CI-949 is an allergic mediator release inhibitor, which inhibits histamine, leukotriene C4/D4 (LTC4/LTD4), and thromboxane B2 (TXB2) release with IC50s of 11.4 μM, 0.5 μM and 0.1 μM, respectively.

  • GC32001 structure
    GC32001KP136 (AL136)
    CAS: 76239-32-2
    Purity: >98%

    KP136 (AL136) (AL136) is an orally effective antiallergic agent.

  • GC32050 structure
    GC32050FRG8701
    CAS: 108498-50-6
    Purity: >98%

    FRG-8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.

  • GC32979 structure
    GC32979Chloropyramine hydrochloride
    CAS: 6170-42-9
    Purity: >99.50%

    Chloropyramine hydrochloride is a histamine receptor H1 antagonist which can also inhibit the biochemical function of VEGFR-3 and FAK.

  • GC33499 structure
    GC33499Fexofenadine D6 (MDL-16455 D6)
    CAS: 548783-71-7
    Purity: >99.00%

    Fexofenadine D6 (MDL-16455 D6) is deuterium labeled is Fexofenadine, which is an antihistamine pharmaceutical agent.

  • GC33544 structure
    GC33544(±)-Methotrimeprazine (D6) (dl-Methotrimeprazine D6)
    CAS: 1189805-51-3
    Purity: >98.00%

    (±)-Levomepromazine D6 ((±)-Methotrimeprazine D6) is the deuterium labeled Methotrimeprazine, which is a D3 dopamine and Histamine H1 receptor antagonist.

  • GC33879 structure
    GC33879Azelastine
    CAS: 58581-89-8
    Purity: >98.00%

    Azelastine, an antihistamine, is a potent and selective histamine 1 (H1) antagonist.

  • GC34338 structure
    GC34338H3R-IN-1 Hydrochloride
    Purity: >98%
  • GC35222 structure
    GC35222ABT-239
    CAS: 460746-46-7
    Purity: >99.00%

    ABT-239 is a novel, highly efficacious, non-imidazole?class of H3R antagonist and a transient receptor potential vanilloid type 1 (TRPV1) antagonist.

  • GC35284 structure
    GC35284Alimemazine D6
    CAS: 1346603-88-0
    Purity: >98%

    Alimemazine D6 is deuterium labeled Alimemazine, which is an antihistamine.

  • GC35471 structure
    GC35471Bavisant
    CAS: 929622-08-2
    Purity: >98%

    Bavisant (JNJ-31001074) is an orally active, potent, brain-penetrating and highly selective antagonist of the histamine H3 receptor.

  • GC35472 structure
    GC35472Bavisant dihydrochloride
    CAS: 929622-09-3
    Purity: >98%

    Bavisant (JNJ-31001074) dihydrochloride is an orally active, potent, brain-penetrating and highly selective antagonist of the histamine H3 receptor.

  • GC35473 structure
    GC35473Bavisant dihydrochloride hydrate
    CAS: 1103522-80-0
    Purity: >99.50%

    Bavisant dihydrochloride hydrate (JNJ31001074AAC) is an orally active, potent, brain-penetrating and highly selective antagonist of the histamine H3 receptor.

  • GC35655 structure
    GC35655Cetirizine D4 dihydrochloride
    Purity: >98%

    Cetirizine D4 dihydrochloride is a deuterium labeled Cetirizine.

  • GC35656 structure
    GC35656Cetirizine D8 dihydrochloride
    CAS: 2070015-04-0
    Purity: >98%

    Cetirizine D8 dihydrochloride is a deuterium labeled Cetirizine.

  • GC35826 structure
    GC35826Decloxizine dihydrochloride
    CAS: 13073-96-6
    Purity: >98.50%

    Decloxizine dihydrochloride(UCB-1402; NSC289116) is a histamine 1 receptor antagonist.

  • GC36278 structure
    GC36278Hydroxyzine D4 dihydrochloride
    Purity: >98%

    Hydroxyzine D4 dihydrochloride is deuterium labeled Hydroxyzine.

  • GC36279 structure
    GC36279Hydroxyzine pamoate
    CAS: 10246-75-0
    Purity: >99.50%

    Hydroxyzine pamoate is a histamine H1-receptor antagonist.

  • GC36476 structure
    GC36476Lodoxamide tromethamine
    CAS: 63610-09-3
    Purity: >99.00%

    Lodoxamide tromethamine (U-42585E) is a medication for the treatment of prophylaxis of mast cell-mediated allergic disease.

  • GC36875 structure
    GC36875Perphenazine D8 Dihydrochloride
    Purity: >98%

    Perphenazine D8 Dihydrochloride is the deuterium labeled Perphenazine, which is a typical antipsychotic drug(5-HT, Dopamine receptor ligand).

  • GC36878 structure
    GC36878PF-03654746
    CAS: 935840-31-6
    Purity: >98%

    PF-03654746 is a potent and selective histamine H3 receptor antagonist with high brain penetration.

  • GC36931 structure
    GC36931Pitolisant
    CAS: 362665-56-3
    Purity: >98%

    A histamine H 3 receptor antagonist and inverse agonist

  • GC36932 structure
    GC36932Pitolisant oxalate
    CAS: 362665-57-4
    Purity: >98%

    Pitolisant oxalate is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM).