Opioid Receptor
Opioid receptor is a group of G protein-coupled receptors with opioids as ligands.
Products Related to Opioid Receptor(151)
- GC46860AP-238 (hydrochloride)CAS: 2749171-05-7Purity: >98.00%
A neuropeptide with diverse biological activities
- GC47913para-methyl AP-237 (hydrochloride)CAS: 2749048-12-0Purity: >98.00%
A neuropeptide with diverse biological activities
- GC60857Frakefamide TFAPurity: >99.00%
Frakefamide TFA is a potent analgesic that acts as a peripheral active μ-selective receptor agonist.
- GC61003Loperamide D6 hydrochlorideCAS: 1189469-46-2Purity: >98%
Loperamide D6 hydrochloride (R-18553 D6 hydrochloride) is a deuterium labeled Loperamide hydrochloride.
- GC61397Asimadoline hydrochlorideCAS: 185951-07-9Purity: >99.50%
Asimadoline (EMD-61753) hydrochloride is an orally active, selective and peripherally active κ-opioid agonist with IC50s of 5.6 nM (guinea pig) and 1.2 nM (human recombinant).
- GC61586UFP-101 TFAPurity: >99.00%
UFP-101 TFA is a potent, selective, and competitive antagonist of the N/OFQ peptide (NOP) receptor, with a pKi of 10.24.
- GC61954Deltorphin 2 TFAPurity: >98.00%
Deltorphin 2 TFA is a selective peptide agonist for the δ opioid receptor.
- GC63115Nociceptin (1-13), amide TFAPurity: >99.50%
Nociceptin (1-13), amide TFA is a potent ORL1 receptor (opioid receptor-like 1 receptor, OP4) agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain membranes.
- GC64147Acetyl tetrapeptide-15CAS: 928007-64-1Purity: >98%
Acetyl tetrapeptide-15 is a synthetic peptide used in the cosmetics for sensitive skin.
- GC666792,6-Dimethyl-L-tyrosineCAS: 123715-02-6Purity: >98%
2,6-Dimethyl-L-tyrosine (Dmt) is a tyrosine derivative that enhances receptor affinity, functional bioactivity and in vivo analgesia of opioid peptides.
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC46182 | Naldemedine | 916072-89-4 | >95.00% | |
A peripherally acting opioid receptor antagonist | ||||
| GC46860 | AP-238 (hydrochloride) | 2749171-05-7 | >98.00% | |
A neuropeptide with diverse biological activities | ||||
| GC47913 | para-methyl AP-237 (hydrochloride) | 2749048-12-0 | >98.00% | |
A neuropeptide with diverse biological activities | ||||
| GC50558 | TAN 452 | 892039-23-5 | >98% | |
Potent and selective peripherally acting δ opioid antagonist; antianalgesic. | ||||
| GC60391 | β-Casomorphin, bovine TFA | - | >98% | |
| GC60730 | CTAP TFA | - | >99.00% | |
CTAP TFA is a potent, highly selective, and BBB penetrant μ opioid receptor antagonist, with an IC50 of 3.5 nM. | ||||
| GC60731 | CTOP TFA | - | >99.50% | |
CTOP TFA is a potent and highly selective μ-opioid receptor antagonist. | ||||
| GC60857 | Frakefamide TFA | - | >99.00% | |
Frakefamide TFA is a potent analgesic that acts as a peripheral active μ-selective receptor agonist. | ||||
| GC61003 | Loperamide D6 hydrochloride | 1189469-46-2 | >98% | |
Loperamide D6 hydrochloride (R-18553 D6 hydrochloride) is a deuterium labeled Loperamide hydrochloride. | ||||
| GC61397 | Asimadoline hydrochloride | 185951-07-9 | >99.50% | |
Asimadoline (EMD-61753) hydrochloride is an orally active, selective and peripherally active κ-opioid agonist with IC50s of 5.6 nM (guinea pig) and 1.2 nM (human recombinant). | ||||
| GC61484 | β-Casomorphin, human TFA | - | >99.50% | |
| GC61586 | UFP-101 TFA | - | >99.00% | |
UFP-101 TFA is a potent, selective, and competitive antagonist of the N/OFQ peptide (NOP) receptor, with a pKi of 10.24. | ||||
| GC61954 | Deltorphin 2 TFA | - | >98.00% | |
Deltorphin 2 TFA is a selective peptide agonist for the δ opioid receptor. | ||||
| GC63072 | Methyl-6-alpha-Naltrexol | 116388-85-3 | >98% | |
| GC63115 | Nociceptin (1-13), amide TFA | - | >99.50% | |
Nociceptin (1-13), amide TFA is a potent ORL1 receptor (opioid receptor-like 1 receptor, OP4) agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain membranes. | ||||
| GC63200 | Spiradoline | 87151-85-7 | >98% | |
| GC63431 | DPDPE TFA | 172888-59-4 | >99.50% | |
DPDPE TFA, an opioid peptide, is a selective δ-opioid receptor?(DOR) agonist?with anticonvulsant effects. | ||||
| GC63686 | Naloxone methiodide | 93302-47-7 | >99.00% | |
| GC64007 | (±)-U-50488 hydrate hydrochloride | - | >99.00% | |
| GC64147 | Acetyl tetrapeptide-15 | 928007-64-1 | >98% | |
Acetyl tetrapeptide-15 is a synthetic peptide used in the cosmetics for sensitive skin. | ||||
| GC66679 | 2,6-Dimethyl-L-tyrosine | 123715-02-6 | >98% | |
2,6-Dimethyl-L-tyrosine (Dmt) is a tyrosine derivative that enhances receptor affinity, functional bioactivity and in vivo analgesia of opioid peptides. | ||||
| GC67907 | CCG258747 | 2615910-00-2 | >98% | |
| GC67956 | Endomorphin 1 acetate | 1276123-71-7 | >99.50% | |
| GC68427 | GSK1521498 free base | 1007573-18-3 | >98.00% | |