GLPBio

Opioid Receptor

Opioid receptor is a group of G protein-coupled receptors with opioids as ligands.

Products Related to Opioid Receptor(151)

  • GC17939 structure
    GC17939JDTic
    CAS: 361444-66-8
    Purity: >98%
  • GC18432 structure
    GC184326α-Naloxol
    CAS: 20410-95-1

    An Analytical Reference Material

  • GC18679 structure
    GC18679Salvinorin B
    CAS: 92545-30-7
    Purity: >95.00%

    Salvinorin B is an analytical reference standard categorized as a diterpene.

  • GC19229 structure
    GC19229CERC-501 (Aticaprant)
    CAS: 1174130-61-0
    Purity: >99.50%

    CERC-501 (Aticaprant) is a potent and centrally-penetrant kappa opioid(KOR) receptor antagonist with a Ki of 0.807nM.

  • GC19500 structure
    GC19500LY2795050
    CAS: 1346133-08-1
    Purity: >98.00%

    LY2795050 is a novel selective κ-opioid Receptor (KOR) antagonist

  • GC30328 structure
    GC30328Gluten Exorphin C
    CAS: 142479-62-7
    Purity: >98.50%

    Gluten exorphin C is an opioid peptide derived from wheat gluten.

  • GC30639 structure
    GC30639Bevenopran (CB-5945)
    CAS: 676500-67-7
    Purity: >98%

    Bevenopran (CB-5945) is a peripheral μ-opioid receptor antagonist.

  • GC30771 structure
    GC30771PZM21
    CAS: 1997387-43-5
    Purity: >98.00%

    A µ-opioid receptor agonist

  • GC30816 structure
    GC30816Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin)
    CAS: 58569-55-4
    Purity: >98.00%

    Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin) is an endogenous opioid that acts as the δ opioid receptor with an EC 50 value of 1.03nM.

  • GC30881 structure
    GC30881Naloxegol oxalate (NKTR-118 oxalate)
    CAS: 1354744-91-4
    Purity: >98%

    A peripherally acting antagonist of the µ-opioid receptor

  • GC30932 structure
    GC30932Naloxegol (NKTR-118)
    CAS: 854601-70-0
    Purity: >98%
  • GC30994 structure
    GC30994Vanilpyruvic acid (Vanylpyruvic acid)
    CAS: 1081-71-6
    Purity: >98.00%

    Vanilpyruvic acid (Vanylpyruvic acid) is a catecholamine metabolite and precursor to vanillactic acid.

  • GC31006 structure
    GC31006ZT 52656A hydrochloride
    CAS: 115730-24-0
    Purity: >99.50%

    ZT 52656A is a selective kappa opioid agonist, used for the prevention or alleviation of pain in the eye.

  • GC31117 structure
    GC31117β-Endorphin, human
    CAS: 61214-51-5
    Purity: >98%

    β-Endorphin, human, a prominent endogenous peptide, existing in the hypophysis cerebri and hypothalamus, is an agonist of opioid receptor, with preferred affinity for μ-opioid receptor and δ-opioid receptor; β-Endorphin, human exhibits antinociception activity.

  • GC31126 structure
    GC31126Valorphin
    CAS: 144313-54-2
    Purity: >98%

    Valorphin is an endogenous hemoglobin β-chain (33-39) fragment with opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM; Valorphin also shows anti-tumor activity.

  • GC31127 structure
    GC31127ORL1 antagonist 1
    CAS: 1174985-59-1
    Purity: >98%

    ORL1 antagonist 1 is an opioid receptor-like 1 (ORL1) antagonist with an IC50 of 61 nM.

  • GC31138 structure
    GC31138[Met5]-Enkephalin, amide (5-Methionine-enkephalin amide)
    CAS: 60117-17-1
    Purity: >98%

    [Met5]-Enkephalin, amide (5-Methionine-enkephalin amide) is an agonist for δ opioid receptors as well as putative ζ (zeta) opioid receptors.

  • GC31151 structure
    GC31151Kelatorphan
    CAS: 92175-57-0
    Purity: >98%

    Kelatorphan is a full inhibitor of enkephalin degrading enzymes.

  • GC31168 structure
    GC31168Dermorphin
    CAS: 77614-16-5
    Purity: >99.50%

    Dermorphin is a natural heptapeptide μ-opioid receptor (MOR) agonist found in amphibian skin.

  • GC31250 structure
    GC31250Opioid receptor modulator 1
    CAS: 77514-44-4
    Purity: >98%

    Opioid receptor modulator 1 is a opioid receptor modulator extracted from patent WO2014072809A2, Compound RA11 in EXAMPLE 7.

  • GC31762 structure
    GC31762Asimadoline (EMD-61753)
    CAS: 153205-46-0
    Purity: >98%

    Asimadoline (EMD-61753) (EMD-61753) is an orally active, selective and peripherally active κ-opioid agonist with IC50s of 5.6 nM (guinea pig) and 1.2 nM (human recombinant).

  • GC32489 structure
    GC32489Hemorphin-7
    CAS: 152685-85-3
    Purity: >99.50%

    Hemorphin-7 is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.

  • GC33081 structure
    GC33081[D-Ala2]leucine-enkephalin
    CAS: 64963-01-5
    Purity: >99.50%

    [D-Ala2]leucine-enkephalin, a delta opioid agonist, is a degradation resistant long-acting Leu-enkephalin.

  • GC33736 structure
    GC33736β-Casomorphin, bovine (β-Casomorphin-7 (bovine))
    CAS: 72122-62-4
    Purity: >99.50%

    β-Casomorphin, bovine (β-Casomorphin-7 (bovine)) (β-Casomorphin-7 (bovine) ) is a opioid peptide with an IC50 of 14 μM in an Opioid receptors binding assay.