Opioid Receptor
Opioid receptor is a group of G protein-coupled receptors with opioids as ligands.
Products for Opioid Receptor
- Cat.No. Product Name Information
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GC13688
Naltrindole hydrochloride
δ opioid antagonist
- GC15408 Neuropeptide AF (human) Endogenous antiopioid peptide implicated in pain modulation and endocrine functions
- GC17325 Nociceptin Endogenous ligand for the NOP opioid receptor
- GC63115 Nociceptin (1-13), amide TFA Nociceptin (1-13), amide TFA is a potent ORL1 receptor (opioid receptor-like 1 receptor, OP4) agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain membranes.
- GC13645 nor-Binaltorphimine dihydrochloride κ-opioid receptor antagonist
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GC31250
Opioid receptor modulator 1
Opioid receptor modulator 1 is a opioid receptor modulator extracted from patent WO2014072809A2, Compound RA11 in EXAMPLE 7.
- GC31127 ORL1 antagonist 1 ORL1 antagonist 1 is an opioid receptor-like 1 (ORL1) antagonist with an IC50 of 61 nM.
- GC10807 PL 017 Selective μ opioid receptor agonist
- GC36947 Porcine dynorphin A(1-13) Porcine dynorphin A (1-13) is a potent, endogenous κ opioid receptor agonist and is antinociceptive at physiological concentrations.
- GC30771 PZM21 A µ-opioid receptor agonist
- GC38842 Ro 64-6198 Ro 64-6198 is a potent, selective, nonpeptide, high-affinity, high cellular permeability and brain penetration N/OFQ receptor (NOP) agonist with an EC50 value of 25.6 nM.
- GC13910 Salvinorin A Non-nitrogenous κ-opioid selective agonist
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GC18679
Salvinorin B
Salvinorin B is an analytical reference standard categorized as a diterpene.
- GC13581 SB 205607 dihydrobromide non-peptide δ1 opioid receptor agonist
- GC39619 SB-612111 SB-612111 is a novel and potent opiate receptor-like orphan receptor (ORL-1) antagonist with a high affinity for hORL-1 (Ki=0.33 nM).
- GC10011 SDM25N hydrochloride δ receptor antagonist
- GN10135 Sec-O-Glucosylhamaudol
- GN10213 Sinomenine Hydrochloride
- GC12041 SNC 162 δ-opioid receptor agonist
- GC11355 SNC 80 A δ-opioid agonist
- GC63200 Spiradoline
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GC50558
TAN 452
Potent and selective peripherally acting δ opioid antagonist; antianalgesic.
- GC10702 Trimebutine Antimuscarinic
- GC37829 Trimebutine maleate Trimebutine maleate is a drug with antimuscarinic and weak mu opioid agonist effects.
- GC30816 Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin) Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin) regulates human immune function and inhibits tumor growth via binding to the opioid receptor.
- GC15512 U-54494A hydrochloride κ-opioid agonist and NMDA antagonist
- GC61586 UFP-101 TFA UFP-101 TFA is a potent, selective, and competitive antagonist of the N/OFQ peptide (NOP) receptor, with a pKi of 10.24.
- GC31126 Valorphin Valorphin is an endogenous hemoglobin β-chain (33-39) fragment with opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM; Valorphin also shows anti-tumor activity.
- GC30994 Vanilpyruvic acid (Vanylpyruvic acid) Vanilpyruvic acid (Vanylpyruvic acid) is a catecholamine metabolite and precursor to vanillactic acid.
- GC31006 ZT 52656A hydrochloride ZT 52656A is a selective kappa opioid agonist, used for the prevention or alleviation of pain in the eye.
- GC11848 [D-Ala2]-Deltorphin II [D-Ala2]-Deltorphin II is a selective peptide agonist for the δ opioid receptor.
- GC33081 [D-Ala2]leucine-enkephalin [D-Ala2]leucine-enkephalin, a delta opioid agonist, is a degradation resistant long-acting Leu-enkephalin.
- GC11236 [Leu5]-Enkephalin Endogenous opioid agonist peptide
- GC35017 [Leu5]-Enkephalin, amide [Leu5]-Enkephalin, amide is a δ opioid receptor agonist.
- GC31138 [Met5]-Enkephalin, amide (5-Methionine-enkephalin amide) [Met5]-Enkephalin, amide (5-Methionine-enkephalin amide) is an agonist for δ opioid receptors as well as putative ζ (zeta) opioid receptors.
- GC35018 [Met5]-Enkephalin, amide TFA [Met5]-Enkephalin, amide TFA is an agonist for δ opioid receptors as well as putative ζ (zeta) opioid receptors.