GLPBio

Opioid Receptor

Opioid receptor is a group of G protein-coupled receptors with opioids as ligands.

Products Related to Opioid Receptor(151)

  • GC33784 structure
    GC33784β-Casomorphin, human (Human β-casomorphin 7)
    CAS: 102029-74-3
    Purity: >98%

    is an opioid peptide, acts as an agonist of opioid receptor.

  • GC34223 structure
    GC34223Dermorphin Analog
    CAS: 115814-08-9
    Purity: >98%

    Dermorphin Analog is an analog of Dermorphin.

  • GC35017 structure
    GC35017[Leu5]-Enkephalin, amide
    CAS: 60117-24-0
    Purity: >99.00%

    [Leu5]-Enkephalin, amide is a δ opioid receptor agonist.

  • GC35018 structure
    GC35018[Met5]-Enkephalin, amide TFA
    CAS: 2918768-28-0
    Purity: >99.50%

    [Met5]-Enkephalin, amide TFA is an agonist for δ opioid receptors as well as putative ζ (zeta) opioid receptors.

  • GC35311 structure
    GC35311Alvimopan monohydrate
    CAS: 1383577-62-5
    Purity: >98%

    Alvimopan monohydrate (ADL 8-2698 monohydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM.

  • GC35638 structure
    GC35638Cebranopadol ((1α,4α)stereoisomer)
    CAS: 863513-93-3
    Purity: >98%

    Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol.

  • GC35805 structure
    GC35805DAMGO (TFA)
    CAS: 950492-85-0
    Purity: >98.00%

    DAMGO (TFA) is a μ-opioid receptor (μ-OPR ) selective agonist with a Kd of 3.46 nM for native μ-OPR.

  • GC35917 structure
    GC35917Dynorphin A (1-10) TFA
    Purity: >99.00%
  • GC35918 structure
    GC35918Dynorphin A 1-10
    CAS: 79994-24-4
    Purity: >98%

    Dynorphin A 1-10 an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.

  • GC35919 structure
    GC35919Dynorphin B (1-13) (TFA)
    Purity: >99.50%

    Dynorphin B (1-13) TFA acts as an agonist on opioid κ-receptor.

  • GC35986 structure
    GC35986Endomorphin 2 TFA
    CAS: 1276124-00-5
    Purity: >99.50%

    Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.

  • GC36479 structure
    GC36479Loperamide hydrochloride
    CAS: 34552-83-5
    Purity: >99.50%

    Loperamide (hydrochloride) (R-18553 (hydrochloride)) is an opioid receptor agonist.

  • GC36508 structure
    GC36508LY-2940094
    CAS: 1307245-86-8
    Purity: >99.50%

    LY-2940094 (BTRX-246040) is a potent, selective and orally available nociceptin receptor (NOP receptor) antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM).

  • GC36562 structure
    GC36562MCOPPB triHydrochloride
    CAS: 1108147-88-1
    Purity: >99.50%

    MCOPPB 3Hcl is a nociceptin receptor agonist with pKi of 10.07; weaker activity at other opioid receptors.

  • GC36778 structure
    GC36778N-terminally acetylated Leu-enkephalin
    CAS: 2703746-32-9
    Purity: >98%

    N-terminally acetylated Leu-enkephalin is the N-terminally acetylated form of Leu-enkephalin.

  • GC36947 structure
    GC36947Porcine dynorphin A(1-13)
    CAS: 72957-38-1
    Purity: >98.50%

    Porcine dynorphin A (1-13) is a potent, endogenous κ opioid receptor agonist and is antinociceptive at physiological concentrations.

  • GC37829 structure
    GC37829Trimebutine maleate
    CAS: 34140-59-5
    Purity: >98.00%

    Trimebutine maleate is a drug with antimuscarinic and weak mu opioid agonist effects.

  • GC38005 structure
    GC38005β-Endorphin, equine
    CAS: 79495-86-6
    Purity: >98%

    β-Endorphin, equine is an endogenous opioid peptide, which binds at high affinity to both μ/δ opioid receptors.

  • GC38030 structure
    GC38030β-Endorphin, equine (TFA)
    Purity: >98%
  • GC38741 structure
    GC38741BPR1M97
    CAS: 2059904-66-2
    Purity: >98.50%

    BPR1M97 is a novel, dual-activity agonist of the mu-opioid receptor (MOP) and the nociceptin/orphanin FQ peptide (NOP) receptor.

  • GC38842 structure
    GC38842Ro 64-6198
    CAS: 280783-56-4
    Purity: >98.00%

    Ro 64-6198 is a potent, selective, nonpeptide, high-affinity, high cellular permeability and brain penetration N/OFQ receptor (NOP) agonist with an EC50 value of 25.6 nM.

  • GC39193 structure
    GC39193LY2444296
    CAS: 1346133-11-6
    Purity: >99.50%

    LY2444296 is an orally bioavailable, high-affinity and selective short-acting kappa opioid receptor (KOPR) antagonist, with a Ki value of ?1 nM.

  • GC39619 structure
    GC39619SB-612111
    CAS: 371980-98-2
    Purity: >98%

    SB-612111 is a novel and potent opiate receptor-like orphan receptor (ORL-1) antagonist with a high affinity for hORL-1 (Ki=0.33 nM).

  • GC43808 structure
    GC43808Hecogenin Acetate
    CAS: 915-35-5
    Purity: >98.00%

    Hecogenin acetate is a steroid sapogenin and an acetylated form of hecogenin that has anthelmintic and antinociceptive properties.