GLPBio

Somatostatin Receptor

Somatostatin receptor is a G protein-coupled receptor that includes five known somatostatin receptors.

Products Related to Somatostatin Receptor(43)

  • GC10181 structure
    GC10181L-803,087 trifluoroacetate
    CAS: 217480-26-7
    Purity: >96.00%

    L-803,087 trifluoroacetate is a potent and selective somatostatin sst4 receptor agonist with a Ki of 0.7 nM.

  • GC10328 structure
    GC10328TT 232
    CAS: 147159-51-1
    Purity: >98%

    sst1/sst4 somatostatin receptors agonist

  • GC10899 structure
    GC10899Octreotide acetate
    CAS: 83150-76-9
    Purity: >99.50%

    A somatostatin receptor agonist

  • GC12448 structure
    GC12448NNC 26-9100
    CAS: 199522-35-5
    Purity: >98%

    Somatostatin sst4 receptor agonist

  • GC12835 structure
    GC12835Cortistatin 14
    CAS: 193829-96-8
    Purity: >99.50%

    Cortistatin 14 (CST-14, human, rat), a neuropeptide with neuronal depressant and sleep modulating properties, can bind to all five cloned somatostatin receptors (SSTRs) and ghrelin receptor to exert its biological activities and co-exists with GABA within the cortex and hippocampus.

  • GC13686 structure
    GC13686CH 275
    CAS: 174688-78-9
    Purity: >98%

    Potent somatostatin receptor 1 (sst1) agonist

  • GC13758 structure
    GC13758Seglitide
    CAS: 81377-02-8
    Purity: >98%

    sst2 and sst5 somatostatin receptors agonist

  • GC14119 structure
    GC14119BIM 23052
    CAS: 133073-82-2
    Purity: >98%

    sst5 receptor agonist

  • GC14747 structure
    GC14747CYN 154806
    CAS: 183658-72-2
    Purity: >98%

    CYN 154806 is a cyclic octapeptide and a potent, selective somatostatin sst2 receptor antagonist (pIC₅₀=8.58). CYN 154806 also inhibits sst1, sst3, sst4, and sst5 receptors.

  • GC15495 structure
    GC15495Cyclosomatostatin
    CAS: 84211-54-1
    Purity: >98%

    somatostatin receptor antagonist

  • GC16400 structure
    GC16400BIM 23056
    CAS: 150155-61-6
    Purity: >99.50%

    Somatostatin receptor ligand

  • GC16422 structure
    GC16422Somatostatin 1-28
    CAS: 74315-46-1
    Purity: >98%

    Somatostatin receptor agonist

  • GC16919 structure
    GC16919(1R,1'S,3'R/1R,1'R,3'S)-L-054,264
    CAS: 208706-12-1
    Purity: >98%

    somatostatin sst2 receptor agonist

  • GC17668 structure
    GC17668L-817,818
    CAS: 217480-27-8
    Purity: >98%

    somatostatin sst5 receptor agonist

  • GC31349 structure
    GC31349MK-4256
    CAS: 1104599-69-0
    Purity: >99.00%

    MK-4256 is a potent and selective SSTR3 antagonist with IC50s of 0.66 nM and 0.36 nM in human and mouse receptor binding assays, respectively.

  • GC34130 structure
    GC34130Vapreotide acetate (RC-160 acetate)
    CAS: 849479-74-9
    Purity: >99.50%

    Vapreotide acetate (RC-160 acetate) (RC-160 acetate; BMY-41606 acetate) is a neurokinin-1 (NK1) receptor antagonist, with an IC50 of 330 nM.

  • GC35730 structure
    GC35730Cortistatin-14 TFA
    CAS: 186901-48-4
    Purity: >98.00%

    Cortistatin-14 TFA, a neuropeptide, is present primarily in the cortex and hippocampus, which inhibits neuronal firing of hippocampal CA1 neurons.

  • GC35787 structure
    GC35787CYN 154806 TFA
    CAS: 2828432-46-6
    Purity: >98%

    CYN 154806 TFA, a cyclic octapeptide, is a potent and selective somatostatin sst2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively.

  • GC36358 structure
    GC36358J-2156
    CAS: 848647-56-3
    Purity: >98%

    J-2156 is a high potent, selective somatostatin receptor type 4 (SST4 receptor) agonist with IC50s of 0.05 nM and 0.07 nM for human and rat SST4 receptors, respectively.

  • GC36857 structure
    GC36857Pasireotide ditrifluoroacetate
    Purity: >99.00%

    Pasireotide (SOM230) ditrifluoroacetate, a long-acting cyclohexapeptide somatostatin analogue, can improve agonist activity at somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/<7.0/9.9, respectively).

  • GC36858 structure
    GC36858Pasireotide L-aspartate salt
    CAS: 396091-77-3
    Purity: >99.00%

    Pasireotide (SOM230) L-aspartate salt, a long-acting cyclohexapeptide somatostatin analogue, can improve agonist activity at somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/<7.0/9.9, respectively).

  • GC50094 structure
    GC50094TC-G 1003
    CAS: 1021912-42-4
    Purity: >98%

    TC-G 1003 is a potent somatostatin receptor subtype 2 (sst2) agonist with a Ki value of 0.025 nM and a cAMP IC50 value of 4.8 nM.

  • GC61413 structure
    GC61413J-2156 TFA
    CAS: 2387505-73-7
    Purity: >99.50%

    J-2156 TFA is a high potent, selective somatostatin receptor type 4 (SST4 receptor) agonist with IC50s of 0.05 nM and 0.07 nM for human and rat SST4 receptors, respectively.

  • GC62194 structure
    GC62194Pasireotide acetate
    CAS: 396091-76-2
    Purity: >99.50%

    Pasireotide (SOM230) acetate, a long-acting cyclohexapeptide somatostatin analogue, can improve agonist activity at somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/<7.0/9.9, respectively).