Androgen Receptor
AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.
Products Related to Androgen Receptor(159)
- GC81354Androgen receptor ligand 4CAS: 92071-89-1Purity: >96.50%
Androgen receptor ligand 4 (Compound MDG486) is an androgen receptor ligand with an IC 50 of >100 µM.
- GC81356Bisphenol F bis(2-chloro-1-propanol) etherCAS: 374772-79-9Purity: >98%
Bisphenol F bis(2-chloro-1-propanol) ether (BFDGE·2HCl) is an androgen receptor antagonist with a human IC 50 of 18 μM.
- GC81682Sialorphin TFAPurity: >97.00%
Sialorphin TFA is a neutral endopeptidase ( NEP ) and aminopeptidase N ( APN ) inhibitor that responds to androgen signals.
- GC92094KISS1-305 (trifluoroacetate salt)Purity: >98.00%
KISS1-305 (trifluoroacetate salt) es un agonista peptídico del receptor de kisspeptin.
- GC11796Estradiol valerateCAS: 979-32-8Purity: >99.00%
El valerato de estradiol (β-estradiol 17-valerato) es un estrÓgeno sintético ampliamente utilizado en combinaciÓn con otras hormonas esteroides en medicamentos de terapia de reemplazo hormonal.
- GC12516SpironolactoneCAS: 52-01-7Purity: >97.00%
Spironolactone es un antagonista dual activo oralmente del receptor mineralocorticoide (MR; IC₅₀=24nM) y receptor de andrógenos (AR; IC₅₀=77nM).
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC81354 | Androgen receptor ligand 4 | 92071-89-1 | >96.50% | |
Androgen receptor ligand 4 (Compound MDG486) is an androgen receptor ligand with an IC 50 of >100 µM. | ||||
| GC81355 | JZY3221 | - | >98.00% | |
JZY3221 is an androgen receptor ( AR ) inhibitor. | ||||
| GC81356 | Bisphenol F bis(2-chloro-1-propanol) ether | 374772-79-9 | >98% | |
Bisphenol F bis(2-chloro-1-propanol) ether (BFDGE·2HCl) is an androgen receptor antagonist with a human IC 50 of 18 μM. | ||||
| GC81357 | JZY3032 | - | >98.00% | |
JYZ3032 is an orally active super inhibitor of androgen receptor ( AR ) and p300/CBP. | ||||
| GC81360 | RU 56279 | 143782-20-1 | >98.00% | |
RU 56279 is an androgen receptor ( AR ) antagonist with strong and systemic anti-androgenic activity. | ||||
| GC81682 | Sialorphin TFA | - | >97.00% | |
Sialorphin TFA is a neutral endopeptidase ( NEP ) and aminopeptidase N ( APN ) inhibitor that responds to androgen signals. | ||||
| GC90891 | Furosine (hydrochloride) | 157974-36-2 | >95.00% | |
Un derivado de L-lisina | ||||
| GC91430 | RAD150 | 1208070-53-4 | >95.00% | |
RAD150 es un modulador del receptor de andrógenos no esteroideo (IC50 = 130 nM) y un derivado de éster benzoato del modulador selectivo del receptor de andrógenos (SARM) RAD140. | ||||
| GC92094 | KISS1-305 (trifluoroacetate salt) | - | >98.00% | |
KISS1-305 (trifluoroacetate salt) es un agonista peptídico del receptor de kisspeptin. | ||||
| GN10142 | Lupeol | 545-47-1 | >98.00% | |
| GN10268 | Triptophenolide | 74285-86-2 | >98.00% | |
| GC11796 | Estradiol valerate | 979-32-8 | >99.00% | |
El valerato de estradiol (β-estradiol 17-valerato) es un estrÓgeno sintético ampliamente utilizado en combinaciÓn con otras hormonas esteroides en medicamentos de terapia de reemplazo hormonal. | ||||
| GC12126 | Flutamide | 13311-84-7 | >99.50% | |
La flutamida es un fÁrmaco antiandrÓgeno, con su metabolito activo que se une al receptor de andrÓgenos con valores de Ki de 55 nM, y se usa principalmente para tratar el cÁncer de prÓstata. | ||||
| GC12516 | Spironolactone | 52-01-7 | >97.00% | |
Spironolactone es un antagonista dual activo oralmente del receptor mineralocorticoide (MR; IC₅₀=24nM) y receptor de andrógenos (AR; IC₅₀=77nM). | ||||
| GC13072 | Epiandrosterone | 481-29-8 | >98.00% | |
steroid hormone with weak androgenic activity | ||||