GLPBio

Estrogen/progestogen Receptor

The estrogen/progestogen receptors are activated by the hormone estrogen/progesterone and regulate the gene transcription.

Products Related to Estrogen/progestogen Receptor(156)

  • GC10012 structure
    GC10012Chlorotrianisene
    CAS: 569-57-3
    Purity: >99.00%

    Estrogen agonist

  • GC10180 structure
    GC10180Cyclofenil
    CAS: 2624-43-3
    Purity: >98%

    Non-steroidal selective estrogen receptor modulator (SERM)

  • GC10346 structure
    GC10346Y 134
    CAS: 849662-80-2
    Purity: >98.00%

    estrogen receptor modulator

  • GC10389 structure
    GC10389ERB 041
    CAS: 524684-52-4
    Purity: >98.00%

    ERB 041 (ERB-041) is a potent and selective estrogen receptor (ER) β agonist with IC50s of 5.4, 3.1 and 3.7 nM for human, rat and mouse ERβ, respectively. ERB 041 displays >200-fold selectivity for ERβ over ERα. ERB 041 is a potent skin cancer chemopreventive agent that acts by dampening the WNT/β-catenin signaling pathway. ERB 041 induces ovarian cancer apoptosis.

  • GC10558 structure
    GC10558GSK 4716
    CAS: 101574-65-6
    Purity: >98.00%

    estrogen-related receptors ERRβ and ERRγ agonist

  • GC10663 structure
    GC10663Dihydrodaidzein
    CAS: 17238-05-0
    Purity: >98.00%

    estrogen receptor agonist

  • GC10684 structure
    GC10684Zearalanone
    CAS: 5975-78-0
    Purity: >98.00%

    estrogen receptor agonist

  • GC10852 structure
    GC10852Bazedoxifene acetate
    CAS: 198481-33-3
    Purity: >99.50%

    A selective estrogen receptor modulator

  • GC11144 structure
    GC11144Chlormadinone acetate
    CAS: 302-22-7
    Purity: >98.00%

    steroidal progestin with additional antiandrogen and antigonadotropic effects

  • GC11425 structure
    GC11425Lasofoxifene (tartrate)
    CAS: 190791-29-8
    Purity: >99.50%

    third-generation, non-steroidal selective estrogen receptor modulator (SERM)

  • GC11544 structure
    GC11544Toremifene
    CAS: 89778-26-7
    Purity: >98%
  • GC11606 structure
    GC116064-Methylbenzylidene camphor
    CAS: 36861-47-9
    Purity: >99.50%

    ultraviolet light blocker used in cosmetics and sunscreen preparations that also has estrogenic activities.

  • GC11734 structure
    GC11734α-Zearalenol
    CAS: 36455-72-8
    Purity: >98.00%

    estrogen receptor agonist

  • GC11863 structure
    GC11863PHTPP
    CAS: 805239-56-9
    Purity: >98.00%

    PHTPP is a selective ERβ full antagonist with 36-fold selectivity for ERβ over ERα. PHTPP can selectively antagonize the ligand binding and transcriptional functions of ERβ, blocking its inhibitory effect on tumor cells, thereby promoting cell proliferation. PHTPP was used to verify ERβ function.

  • GC11881 structure
    GC11881MPP dihydrochloride
    CAS: 911295-24-4
    Purity: >98.00%

    MPP dihydrochloride is a selective estrogen receptor α (ERα) antagonist.

  • GC11996 structure
    GC11996Ospemifene
    CAS: 128607-22-7
    Purity: >99.50%

    non-hormonal selective estrogen receptor modulator (SERM)

  • GC12140 structure
    GC12140Endoxifen
    CAS: 112093-28-4
    Purity: >98%

    Endoxifen Z-isomer is the most important Tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERα).

  • GC12644 structure
    GC12644Quinestrol
    CAS: 152-43-2
    Purity: >98.00%

    synthetic estrogen that is effective in hormone replacement therapy

  • GC12766 structure
    GC12766G-1
    CAS: 881639-98-1
    Purity: >99.50%

    G-1 is a selective and potent agonist of GPR30 with EC50 value about 2 nM.

  • GC12767 structure
    GC12767Zearalenone
    CAS: 17924-92-4
    Purity: >98.00%

    Zearalenone is an estrogenic fusariotoxin that binds to estrogen receptors, including the 17β-estradiol-specific subtype.

  • GC13309 structure
    GC13309WAY 200070
    CAS: 440122-66-7
    Purity: >99.00%

    ERβ receptor agonist

  • GC13373 structure
    GC13373(R)-DPN
    CAS: 524047-78-7
    Purity: >98%

    estrogen receptor (ER) β agonist

  • GC13917 structure
    GC139174’-hydroxy Tamoxifen
    CAS: 82413-23-8
    Purity: ≥98% (may contain up to 10% of the (E) isomer)

    metabolite of tamoxifen, an estrogen receptor modulator

  • GC14131 structure
    GC14131FERb 033
    CAS: 1111084-78-6
    Purity: >98%

    ERβ receptor agonist