Estrogen/progestogen Receptor
The estrogen/progestogen receptors are activated by the hormone estrogen/progesterone and regulate the gene transcription.
Products Related to Estrogen/progestogen Receptor(156)
- GC14370Propyl pyrazole triol (PPT)CAS: 263717-53-9Purity: >98.00%
Propyl pyrazole triol (PPT) is a selective estrogen receptor α (ERα) agonist that can shield neurons from oxidative stress and inflammatory damage through ERα activation in the nervous system.
- GC15373(E)-2-Decenoic acidCAS: 334-49-6Purity: >98.00%
An unsaturated fatty acid found in royal jelly
- GC15975α-EstradiolCAS: 57-91-0Purity: >98.00%
α-Estradiol, a natural form of the hormone lacking estrogenic effects, inhibits the activity of 5-alpha reductase enzymes.
- GC16372(Z)-4-HydroxytamoxifenCAS: 68047-06-3Purity: >99.50%
(Z)-4-Hydroxytamoxifen is a selective estrogen receptor modulator (SERM) that influences the binding of [3H]oestradiol to the estrogen receptor with an IC50 value of 3.3 nM.
- GC17161Methylpiperidino pyrazoleCAS: 289726-02-9Purity: >98.00%
Methylpiperidino pyrazole is a highly selective estrogen receptor α (Erα) antagonist with an IC 50 value of 20.01nM.
- GC17258β-Estradiol-d3CAS: 79037-37-9Purity: >97.50%
β-Estradiol-d3 is a deuterated labeling compound of the endogenous estrogen 17β-Estradiol.
- GC1747517-HydroxyprogesteroneCAS: 68-96-2Purity: >99.50%
An endogenous progestogen and chemical intermediate
- GC17688Diarylpropionitrile(DPN)CAS: 1428-67-7Purity: >99.50%
Diarylpropionitrile(DPN) (Diarylpropionitrile) is a non-steroidal estrogen receptor β (ERβ) selective ligand, with an EC50 of 0.85 nM.
- GC178034-HydroxytamoxifenCAS: 68392-35-8Purity: >98.00%
4-hydroxytamoxifen is a major metabolite of tamoxifen and selective estrogen receptor antagonist.
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC14370 | Propyl pyrazole triol (PPT) | 263717-53-9 | >98.00% | |
Propyl pyrazole triol (PPT) is a selective estrogen receptor α (ERα) agonist that can shield neurons from oxidative stress and inflammatory damage through ERα activation in the nervous system. | ||||
| GC14405 | AZD9496 | 1639042-08-2 | >99.00% | |
estrogen receptor inhibitor, orally active | ||||
| GC14883 | Bazedoxifene | 198481-32-2 | >98% | |
| GC14902 | G-36 | 1392487-51-2 | >98.00% | |
G-36 is a cell-permeable G protein-coupled estrogen receptor (GPER/GPR30) antagonist that inhibits estrogen-mediated calcium mobilization (IC 50 =112nM). | ||||
| GC15373 | (E)-2-Decenoic acid | 334-49-6 | >98.00% | |
An unsaturated fatty acid found in royal jelly | ||||
| GC15599 | Hydroxyprogesterone caproate | 630-56-8 | >98.00% | |
synthetic progestational agent | ||||
| GC15975 | α-Estradiol | 57-91-0 | >98.00% | |
α-Estradiol, a natural form of the hormone lacking estrogenic effects, inhibits the activity of 5-alpha reductase enzymes. | ||||
| GC16372 | (Z)-4-Hydroxytamoxifen | 68047-06-3 | >99.50% | |
(Z)-4-Hydroxytamoxifen is a selective estrogen receptor modulator (SERM) that influences the binding of [3H]oestradiol to the estrogen receptor with an IC50 value of 3.3 nM. | ||||
| GC16618 | G-15 | 1161002-05-6 | >99.00% | |
G-15 is a high-affinity, selective antagonist of G protein-coupled estrogen receptor (GPER/ GPR30) (K i = 20nM). | ||||
| GC16719 | Ormeloxifene | 31477-60-8 | >98% | |
estrogen receptor modulator | ||||
| GC16742 | ZK 164015 | 177583-70-9 | >98% | |
estrogen receptor silent antagonist | ||||
| GC16847 | Tanaproget | 304853-42-7 | >99.50% | |
| GC16852 | Estropipate | 7280-37-7 | >98.00% | |
Estrogen receptor agonist | ||||
| GC17119 | 8-Prenylnaringenin | 53846-50-7 | >99.00% | |
estrogen receptor inhibitor | ||||
| GC17161 | Methylpiperidino pyrazole | 289726-02-9 | >98.00% | |
Methylpiperidino pyrazole is a highly selective estrogen receptor α (Erα) antagonist with an IC 50 value of 20.01nM. | ||||
| GC17200 | Nestoron | 7759-35-5 | >99.50% | |
A synthetic progestin | ||||
| GC17258 | β-Estradiol-d3 | 79037-37-9 | >97.50% | |
β-Estradiol-d3 is a deuterated labeling compound of the endogenous estrogen 17β-Estradiol. | ||||
| GC17475 | 17-Hydroxyprogesterone | 68-96-2 | >99.50% | |
An endogenous progestogen and chemical intermediate | ||||
| GC17588 | Bavachin | 19879-32-4 | >98.00% | |
estrogen receptors ERα and ERβ activator | ||||
| GC17688 | Diarylpropionitrile(DPN) | 1428-67-7 | >99.50% | |
Diarylpropionitrile(DPN) (Diarylpropionitrile) is a non-steroidal estrogen receptor β (ERβ) selective ligand, with an EC50 of 0.85 nM. | ||||
| GC17803 | 4-Hydroxytamoxifen | 68392-35-8 | >98.00% | |
4-hydroxytamoxifen is a major metabolite of tamoxifen and selective estrogen receptor antagonist. | ||||
| GC17856 | RU 58668 | 151555-47-4 | >98% | |
Pure antiestrogen that downregulates estrogen receptor expression | ||||
| GC18003 | (R,R)-THC | 138090-06-9 | >98% | |
ERα receptor agonist | ||||
| GC18333 | Equilenin | 517-09-9 | >98% | |
Equilenin is an equine estrogen found in the urine of pregnant mares. | ||||
