AMPAR

AMPA receptor antagonist

positive allosteric modulator of AMPA receptors

Ca2+-permeable AMPA receptor antagonist

NBQX disodium salt is a potent, highly selective, and competitive antagonist of AMPA receptors, with IC 50 values of 0.7±0.1μM and 0.7±0.03μM for AMPA and kainic acid receptors, respectively.

AMPA agonist

positive allosteric modulator of AMPA receptors

AMPA receptor antagonist

AMPA receptors blocker

NBQX is a highly selective and competitive AMPA receptor antagonist.

inhibitor of the interaction between AMPA receptor and N-ethylmaleimide-sensitive fusion protein (NSF)

CNQX disodium salt (FG9065 disodium) is a potent and competitive AMPA/kainate receptor antagonist with IC50s of 0.3 μM and 1.5 μM, respectively.

positive allosteric modulator of AMPA receptors

CX 546 is a potent activator of 3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor, with an EC 50 value of 93.2μM.

AMPA receptor agonist

AMPA and kainate receptor antagonist

desensitising AMPA receptor agonist

L-Quisqualic acid (L-L-Quisqualic acid), a natural analog of glutamate, is a potent and pan two subsets (iGluR and mGluR) of excitatory amino acid (EAA) agonist with an EC50 of 45 nM and a Ki of 10 nM for mGluR1R.

Inactive control peptide analog of pep2-SVKI

ZK 200775 (ZK200775) is a highly selective AMPA/kainate antagonist with little activity against NMDA; have Ki values of 3.2 nM, 100 nM, and 8.5 μM against quisqualate, kainate, and NMDA, respectively.

YM 90K hydrochloride is a potent and selective AMPA receptor antagonist with a Ki of 84 nM.

Peptide inhibitor of the interaction between the C-terminus of the GluR2 subunit and N-ethylmaleimide-sensitive fusion protein

Peptide containing the 'TGL' motif that corresponds to the C-terminus of GluR1 subunit

(S)-AMPA is the active S-enantiomer of AMPA. (S)-AMPA is a potent and highly selective AMPA-type ionotropic glutamate receptor agonist.

AMPA agonist,subtype-selective,weakly desensitizing