GLPBio

Drug Metabolite

Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.

Products Related to Drug Metabolite(546)

  • GC70731 structure
    GC70731Anhydrosimvastatin
    CAS: 210980-68-0

    Anhydrosimvastatin (Impurity C) is an impurity of Simvastatin.

  • GC70763 structure
    GC707632-NP-AMOZ
    CAS: 183193-59-1

    2-NP-AMOZ is a 2-nitrophenyl derivative of AMOZ (a metabolite of antibiotic Furaltadone), can be used to detect protein bound AMOZ.

  • GC70767 structure
    GC70767T-705RMP ammonium
    CAS: 2096342-42-4

    T-705RMP (ammonium) is the ammonium form of T-705RMP.

  • GC70795 structure
    GC70795Voriconazole N-oxide hydrochloride
    Purity: >99.00%

    Voriconazole N-oxide (Voriconazole oxynitride) (hydrochloride) is the main metabolite of Voriconazole , a widely used triazole antibiotic (fungal).

  • GC71042 structure
    GC7104218β-Glycyrrhetyl-3-O-sulfate
    CAS: 10251-38-4
    Purity: >98.00%

    18β-Glycyrrhetyl-3-O-sulfate (Glycyrrhetic acid 3-O-(hydrogen sulfate)) is a potent type 2 11β-hydroxysteroid dehydrogenase (11β-HSD2) inhibitor with an IC50 of 0.10 µM using rat kidney microsome.

  • GC71908 structure
    GC71908Deoxynivalenol-3-β-D-glucoside
    CAS: 131180-21-7

    Deoxynivalenol-3-β-D-glucoside (DON-3-β-D-glucoside) is a plant metabolite of the Fusarium mycotoxin Deoxynivalenol .

  • GC72920 structure
    GC72920Ketanserinol
    CAS: 76330-73-9
    Purity: >98.00%

    Ketanserinol (R 46742) is a metabolite of Ketanserin.

  • GC78906 structure
    GC78906Ternidazole
    CAS: 1077-93-6
    Purity: >99.00%

    Ternidazole is a nitroimidazole Antibiotic with anti-pathogenic microbial activity.

  • GC79576 structure
    GC795761-(3-Carboxypropyl)-3,7-dimethylxanthine
    CAS: 6493-07-8
    Purity: >98.00%

    1-(3-Carboxypropyl)-3,7-dimethylxanthine is the major circulating oxidative carboxylation metabolite of Pentoxifylline.

  • GC79584 structure
    GC79584UDP-Glucosamine
    CAS: 17479-04-8
    Purity: >98%

    UDP-Glucosamine is a sugar nucleotide analog, glycosyl donor, and metabolite of D-galactosamine.

  • GC79588 structure
    GC795884'-Hydroxywarfarin
    CAS: 24579-14-4
    Purity: >99.50%

    4′-Hydroxywarfarin is a regioisomeric phenolic derivative of Warfarin.

  • GC79594 structure
    GC795941-(4-Methoxyphenyl)-1-propanol
    CAS: 5349-60-0
    Purity: >99.00%

    1-(4-Methoxyphenyl)-1-propanol (Compound 2) is an orally active derivative of anethole.

  • GC79595 structure
    GC79595N-Nitrosoglyphosate
    CAS: 56516-72-4
    Purity: >98%

    N-Nitrosoglyphosate is the nitrosamine degradation product of glyphosate herbicidee.

  • GC79596 structure
    GC79596(S)-4-Hydroxymephenytoin
    CAS: 82695-93-0
    Purity: >98%

    (S) -4-Hydroxy mephenytoin is a metabolite derived from the stereoselective metabolism of mephenytoin.

  • GC79597 structure
    GC79597N-Acetyl-S-(N-methylcarbamoyl)cysteine
    CAS: 103974-29-4
    Purity: >98.00%

    N-Acetyl-S-(N-methylcarbamoyl) cysteine is a metabolite of solvent N,N-dimethylformamide and could be used for monitoring industrial exposure.

  • GC79598 structure
    GC79598Tyramine O-sulfate sodium
    CAS: 2083619-07-0
    Purity: >99.00%

    Tyramine O-sulfate (Tyramine sulfate) sodium is a metabolite of Tyramine formed via sulfation, which serves as a biomarker for depression.

  • GC79599 structure
    GC79599Melatonin-OH
    CAS: 67199-08-0
    Purity: >98.50%

    Melatonin -OH is an oxidative Melatonin metabolite with free radical-scavenging activity.

  • GC79600 structure
    GC796003-Hydroxybenzo[a]pyrene
    CAS: 13345-21-6
    Purity: >98%

    3-Hydroxybenzo[a]pyrene (3-OHBaP) is a preferable biomarker to assess exposure to benzo[a]pyrene (BaP), a carcinogenic agent.

  • GC79601 structure
    GC79601Diazoxon
    CAS: 962-58-3
    Purity: >98%

    Diazoxon is a metabolite of Diazinon.

  • GC79602 structure
    GC796025Oxo-MEHTP
    CAS: 1684398-40-0
    Purity: >98%

    5Oxo-MEHTP is an urinary metabolite of di(2-ethylhexyl) terephthalate (DEHTP).

  • GC79603 structure
    GC796033-(3-Sulfooxyphenyl)propanoic acid disodium
    Purity: >98.00%

    3-(3-Sulfooxyphenyl) propanoic acid disodium is a metabolite of Echinacoside.

  • GC79604 structure
    GC79604Fenthion sulfoxide
    CAS: 3761-41-9
    Purity: >98.00%

    Fenthion sulfoxide is a metabolite of the organophosphate insecticide Fenthion.

  • GC79605 structure
    GC796051-(7-Hydroxy-4-methyloctyl) 1,2-cyclohexanedicarboxylate
    CAS: 1637562-52-7
    Purity: >98%

    1-(7-Hydroxy-4-methyloctyl) 1,2-cyclohexanedicarboxylate is a metabolite of di (isononyl) cyclohexane-1,2-dicarboxylate (DINCH), an alternative for phthalate plasticizers.

  • GC79606 structure
    GC7960620α-Dihydrodydrogesterone
    CAS: 4243-74-7
    Purity: >98%

    20α-dihydrodydrogesterone is the major active metabolite of Dydrogesterone produced in the human body after oral administration.