Drug Metabolite
Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.
Products Related to Drug Metabolite(546)
- GC79607Tiopronin disulfideCAS: 21269-37-4Purity: >98%
Tiopronin disulfide, a Tiopronin dimer, is an oxidative product of Tiopronin.
- GC796081,2-Cyclohexanedicarboxylic acid mono 4-methyl-7-carboxy-heptyl esterCAS: 1637562-51-6Purity: >98%
1,2-Cyclohexanedicarboxylic Acid Mono 4-Methyl-7-carboxy-heptyl Ester is a secondary oxidized metabolite of di(isononyl) cyclohexane-1,2-dicarboxylate (DINCH), an alternative for phthalate plasticizer.
- GC796092-Hydroxymethyl olanzapineCAS: 174756-45-7Purity: >98.00%
2-Hydroxymethyl olanzapine is a metabolite and a degradation product of Olanzapine [1] [2] .
- GC796107-Hydroxycoumarin glucuronideCAS: 66695-14-5Purity: >98.00%
7-Hydroxycoumarin glucuronide is a transport substrate and main human coumarin metabolite.
- GC79611Bupivacaine N-oxide hydrochlorideCAS: 1796927-05-3Purity: >98.00%
Bupivacaine N-oxide hydrochloride is a metabolite of Bupivacaine.
- GC796131',4-Dihydroxy midazolamCAS: 64740-68-7Purity: >98.00%
1',4-Dihydroxymidazolam is a hydroxylated metabolite produced by cytochrome P450 -mediated metabolism of midazolam in the liver [1] .
- GC796145α-DihydrocortisolCAS: 516-41-6Purity: >98.00%
5α-Dihydrocortisol (5α-DHF), a metabolite of Hydrocortisone (Cortisol), is a steroid hormone.
- GC7961520α-DihydrocortisolCAS: 1719-79-5Purity: >96.50%
20α-Dihydrocortisol (20α-DHF) is a metabolite of Hydrocortisone (Cortisol) [1] .
- GC79616Acetaminophen glucuronide potassiumPurity: >99.50%
Acetaminophen glucuronide potassium (APAP-glu potassium) is the inactive glucuronide metabolite of Acetaminophen.
- GC79617Clethodim sulfoxideCAS: 111031-14-2Purity: >98%
Clethodim sulfoxide is the aerobic metabolite of clethodim, a cyclohexanedione oxime herbicide [1] .
- GC79618Prucalopride N-oxideCAS: 1900715-98-1Purity: >98.00%
Prucalopride N-oxide is a metabolite of Prucalopride with motility-enhancing effects [1] .
- GC79619Fipronil sulfideCAS: 120067-83-6Purity: >98.00%
Fipronil sulfide is a toxic, persistent metabolite of Fipronil.
- GC79620Dapagliflozin keto impurityCAS: 2169998-23-4Purity: >98.00%
Dapagliflozin keto impurity (Oxo-dapagliflozin) is an oxo metabolite and related impurity of Dapagliflozin.
- GC796215α,6α-EpoxysitosterolCAS: 53034-66-5Purity: >99.50%
5α,6α-Epoxysitosterol is a minor β-sitosterol oxidation product and 5,6-epoxy thermo-oxidation product of sitosterol [1] [2] .
- GC79622Ginsenoside C-YCAS: 83480-65-3Purity: >98%
Ginsenoside C-Y (Ginsenoside Y) is a metabolite of Ginsenoside Rb2.
- GC7962441-O-DemethylrapamycinCAS: 142382-16-9Purity: >98%
41-O-Demethylrapamycin is a metabolite of Rapamycin produced by Bacillus megaterium [1] .
- GC79625Febuxostat 67M-1CAS: 887945-96-2Purity: >95.00%
Febuxostat 67M-1 is an active metabolite of Febuxostat.
- GC79713D-Ribonic acid ammoniumCAS: 90801-23-3Purity: >98.00%
D-Ribonic acid ammonium is a metabolite of D-Ribose.
- GC804914-Methylamino antipyrine-d 3 -1CAS: 1246820-06-3Purity: >98%
4-Methylamino antipyrine-d 3 -1 is the deuterium labeled 4-Methylamino antipyrine-1.
- GC816012-HydroxymelatoninCAS: 229018-17-1Purity: >98.00%
2-Hydroxymelatonin is a major hydroxylated metabolite of Melatonin.
- GC81606DX-8951 Hydroxy-acid sodiumPurity: >98.50%
DX-8951 Hydroxy-acid sodium is a prodrug of phosphoramide.
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC79607 | Tiopronin disulfide | 21269-37-4 | >98% | |
Tiopronin disulfide, a Tiopronin dimer, is an oxidative product of Tiopronin. | ||||
| GC79608 | 1,2-Cyclohexanedicarboxylic acid mono 4-methyl-7-carboxy-heptyl ester | 1637562-51-6 | >98% | |
1,2-Cyclohexanedicarboxylic Acid Mono 4-Methyl-7-carboxy-heptyl Ester is a secondary oxidized metabolite of di(isononyl) cyclohexane-1,2-dicarboxylate (DINCH), an alternative for phthalate plasticizer. | ||||
| GC79609 | 2-Hydroxymethyl olanzapine | 174756-45-7 | >98.00% | |
2-Hydroxymethyl olanzapine is a metabolite and a degradation product of Olanzapine [1] [2] . | ||||
| GC79610 | 7-Hydroxycoumarin glucuronide | 66695-14-5 | >98.00% | |
7-Hydroxycoumarin glucuronide is a transport substrate and main human coumarin metabolite. | ||||
| GC79611 | Bupivacaine N-oxide hydrochloride | 1796927-05-3 | >98.00% | |
Bupivacaine N-oxide hydrochloride is a metabolite of Bupivacaine. | ||||
| GC79612 | BTS44596 | 139542-32-8 | >98% | |
BTS44596 (Prochloraz-desimidazole-formylamino) is a metabolite of the antifungal agent Prochloraz. | ||||
| GC79613 | 1',4-Dihydroxy midazolam | 64740-68-7 | >98.00% | |
1',4-Dihydroxymidazolam is a hydroxylated metabolite produced by cytochrome P450 -mediated metabolism of midazolam in the liver [1] . | ||||
| GC79614 | 5α-Dihydrocortisol | 516-41-6 | >98.00% | |
5α-Dihydrocortisol (5α-DHF), a metabolite of Hydrocortisone (Cortisol), is a steroid hormone. | ||||
| GC79615 | 20α-Dihydrocortisol | 1719-79-5 | >96.50% | |
20α-Dihydrocortisol (20α-DHF) is a metabolite of Hydrocortisone (Cortisol) [1] . | ||||
| GC79616 | Acetaminophen glucuronide potassium | - | >99.50% | |
Acetaminophen glucuronide potassium (APAP-glu potassium) is the inactive glucuronide metabolite of Acetaminophen. | ||||
| GC79617 | Clethodim sulfoxide | 111031-14-2 | >98% | |
Clethodim sulfoxide is the aerobic metabolite of clethodim, a cyclohexanedione oxime herbicide [1] . | ||||
| GC79618 | Prucalopride N-oxide | 1900715-98-1 | >98.00% | |
Prucalopride N-oxide is a metabolite of Prucalopride with motility-enhancing effects [1] . | ||||
| GC79619 | Fipronil sulfide | 120067-83-6 | >98.00% | |
Fipronil sulfide is a toxic, persistent metabolite of Fipronil. | ||||
| GC79620 | Dapagliflozin keto impurity | 2169998-23-4 | >98.00% | |
Dapagliflozin keto impurity (Oxo-dapagliflozin) is an oxo metabolite and related impurity of Dapagliflozin. | ||||
| GC79621 | 5α,6α-Epoxysitosterol | 53034-66-5 | >99.50% | |
5α,6α-Epoxysitosterol is a minor β-sitosterol oxidation product and 5,6-epoxy thermo-oxidation product of sitosterol [1] [2] . | ||||
| GC79622 | Ginsenoside C-Y | 83480-65-3 | >98% | |
Ginsenoside C-Y (Ginsenoside Y) is a metabolite of Ginsenoside Rb2. | ||||
| GC79623 | Ichangin | 10171-61-6 | >98% | |
Ichangin is a metabolite of ponderosa lemon Citrus pyriformis. | ||||
| GC79624 | 41-O-Demethylrapamycin | 142382-16-9 | >98% | |
41-O-Demethylrapamycin is a metabolite of Rapamycin produced by Bacillus megaterium [1] . | ||||
| GC79625 | Febuxostat 67M-1 | 887945-96-2 | >95.00% | |
Febuxostat 67M-1 is an active metabolite of Febuxostat. | ||||
| GC79713 | D-Ribonic acid ammonium | 90801-23-3 | >98.00% | |
D-Ribonic acid ammonium is a metabolite of D-Ribose. | ||||
| GC80491 | 4-Methylamino antipyrine-d 3 -1 | 1246820-06-3 | >98% | |
4-Methylamino antipyrine-d 3 -1 is the deuterium labeled 4-Methylamino antipyrine-1. | ||||
| GC81360 | RU 56279 | 143782-20-1 | >98.00% | |
RU 56279 is an androgen receptor ( AR ) antagonist with strong and systemic anti-androgenic activity. | ||||
| GC81601 | 2-Hydroxymelatonin | 229018-17-1 | >98.00% | |
2-Hydroxymelatonin is a major hydroxylated metabolite of Melatonin. | ||||
| GC81606 | DX-8951 Hydroxy-acid sodium | - | >98.50% | |
DX-8951 Hydroxy-acid sodium is a prodrug of phosphoramide. | ||||