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Home >> Signaling Pathways >> Proteases >> Drug Metabolite

Drug Metabolite

Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.

Targets for  Drug Metabolite

Products for  Drug Metabolite

  1. Cat.No. Product Name Information
  2. GC45208 α-hydroxy Metoprolol α-hydroxy Metoprolol is an active metabolite of the β1-adrenergic receptor blocker metoprolol. α-hydroxy Metoprolol Chemical Structure
  3. GC40480 α-Phenyl-α-(2-pyridyl)acetonitrile α-Phenyl-α-(2-pyridyl)thioacetamide, also known as antigastrin and SC-15396, is an inhibitor of gastric acid secretion. α-Phenyl-α-(2-pyridyl)acetonitrile Chemical Structure
  4. GC41661 (±)-4-hydroxy Propranolol β-D-Glucuronide (±)-4-hydroxy Propranolol β-D-glucuronide is a metabolite of (±)-4-hydroxy propranolol, which is a metabolite of propranolol. (±)-4-hydroxy Propranolol β-D-Glucuronide Chemical Structure
  5. GC46284 (±)-Cotinine-d3 An internal standard for the quantification of cotinine (±)-Cotinine-d3 Chemical Structure
  6. GC41671 (±)-Equol 4'-sulfate (sodium salt)

    (±)-Equol 4'-sulfate is a gut-mediated phase II metabolite of the isoflavonoid phytoestrogen (±)-equol.

     (±)-Equol 4'-sulfate (sodium salt) Chemical Structure
  7. GC41315 (±)-Ketoprofen Glucuronide (±)-Ketoprofen glucuronide is a phase II metabolite of the non-steroidal anti-inflammatory drug (NSAID) ketoprofen. (±)-Ketoprofen Glucuronide Chemical Structure
  8. GC49875 (±)-N-desmethyl Venlafaxine (hydrochloride) A minor active metabolite of venlafaxine (±)-N-desmethyl Venlafaxine (hydrochloride) Chemical Structure
  9. GC45252 (-)-Sitagliptin Carbamoyl Glucuronide (-)-Sitagliptin carbamoyl glucuronide is a minor phase II metabolite of the dipeptidyl peptidase 4 (DPP-4) inhibitor (-)-sitagliptin. (-)-Sitagliptin Carbamoyl Glucuronide Chemical Structure
  10. GC18622 (2'S)-Nicotine-1-oxide (2'S)-Nicotine-1-oxide is a metabolite of nicotine . (2'S)-Nicotine-1-oxide Chemical Structure
  11. GC68509 (25R)-12α-Hydroxyspirost-4-en-3-one

    (25R)-12α-Hydroxyspirost-4-en-3-one is a secondary metabolite produced by Nocardia globerula from Hecogenin.

     (25R)-12α-Hydroxyspirost-4-en-3-one Chemical Structure
  12. GC41694 (3S)-hydroxy Quinidine (3S)-hydroxy Quinidine is an active quinidine metabolite. (3S)-hydroxy Quinidine Chemical Structure
  13. GC60399 (E)-10-Hydroxynortriptyline (E)-10-Hydroxynortriptyline (E-10-OH-NT) is a metabolite of Nortriptyline. (E)-10-Hydroxynortriptyline Chemical Structure
  14. GC40286 (E,Z)-2-propyl-2-Pentenoic Acid (E,Z)-2-propyl-2-Pentenoic acid is a bioactive metabolite of valproic acid that exhibits the same profile and potency of anticonvulsant activity in animal models as its parent compound without any observed teratogenicity and hepatotoxicity. (E,Z)-2-propyl-2-Pentenoic Acid Chemical Structure
  15. GC49189 (E/Z)-4-hydroxy Tamoxifen-d5 An internal standard for the quantification of (E/Z)-4-hydroxy tamoxifen (E/Z)-4-hydroxy Tamoxifen-d5 Chemical Structure
  16. GC62737 (R)-(-)-O-Desmethyl Venlafaxine D6 (R)-(-)-O-Desmethyl Venlafaxine D6 Chemical Structure
  17. GC41722 (R,S)-Carvedilol Glucuronide (R,S)-Carvedilol glucuronide is a racemic mixture of the carvedilol metabolites (R)-carvedilol glucuronide and (S)-carvedilol glucuronide. (R,S)-Carvedilol Glucuronide Chemical Structure
  18. GC60410 (Rac)-3′-Hydroxy simvastatin (Rac)-3′-Hydroxy simvastatin is a metabolite of Simvastatin. (Rac)-3′-Hydroxy simvastatin Chemical Structure
  19. GC40145 (S)-Laudanosine (S)-Laudanosine is the (S) enantiomer of laudanosine, a metabolite of the neuromuscular blocking agents atracurium and cisatracurium. (S)-Laudanosine Chemical Structure
  20. GC49179 (S)-O-Desmethyl Naproxen A metabolite of (S)-naproxen (S)-O-Desmethyl Naproxen Chemical Structure
  21. GC60419 (S)-O-Desmethyl Venlafaxine N-Oxide (S)-O-Desmethyl Venlafaxine N-Oxide is a N-oxyde of (S)-O-Desmethyl Venlafaxine. (S)-O-Desmethyl Venlafaxine N-Oxide Chemical Structure
  22. GC60427 (Z)-10-Hydroxynortriptyline (Z)-10-Hydroxynortriptyline is a metabolite of Nortriptyline. (Z)-10-Hydroxynortriptyline Chemical Structure
  23. GC67761 (Z)-10-Hydroxynortriptyline-d3 (Z)-10-Hydroxynortriptyline-d3 Chemical Structure
  24. GC18596 (±)-2-propyl-4-Pentenoic Acid

    (±)-2-propyl-4-Pentenoic acid (4-ene VPA) is a major metabolite of valproic acid .

     (±)-2-propyl-4-Pentenoic Acid Chemical Structure
  25. GC41995 1'-hydroxy Midazolam Major metabolite of the anesthetic, midazolam 1'-hydroxy Midazolam Chemical Structure
  26. GC41837 1,3,7-Trimethyluric Acid

    1,3,7-Trimethyluric acid is a methyl derivative of uric acid and a product of C-8 oxidation of caffeine by cytochrome P450 enzymes.

     1,3,7-Trimethyluric Acid Chemical Structure
  27. GC46387 1,3,7-Trimethyluric Acid-d9 An internal standard for the quantification of 1,3,7-trimethyluric acid 1,3,7-Trimethyluric Acid-d9 Chemical Structure
  28. GC49294 1-(4-Chlorobenzhydryl)piperazine An inactive metabolite of meclizine and chlorcyclizine 1-(4-Chlorobenzhydryl)piperazine Chemical Structure
  29. GC49366 1-Salicylate Glucuronide A metabolite of salicylic acid and aspirin 1-Salicylate Glucuronide Chemical Structure
  30. GC49820 10,11-dihydro-10,11-dihydroxy Carbamazepine A metabolite of carbamazepine and oxcarbazepine 10,11-dihydro-10,11-dihydroxy Carbamazepine Chemical Structure
  31. GC66057 10,11-Dihydrocarbamazepine 10,11-Dihydrocarbamazepine is the active metabolite of Oxcarbazepine. 10,11-Dihydrocarbamazepine also is an intermediate. Oxcarbazepine is rapidly and almost completely converted to 10,11-Dihydrocarbamazepine with probable Anticonvulsant efficacy. 10,11-Dihydrocarbamazepine Chemical Structure
  32. GC49118 10-hydroxy Warfarin A metabolite of (R)-warfarin 10-hydroxy Warfarin Chemical Structure
  33. GC49759 13C17-Mycophenolic Acid An internal standard for the quantification of mycophenolic acid 13C17-Mycophenolic Acid Chemical Structure
  34. GC19442 15-Acetyldeoxy Nivalenol 15-Acetyldeoxy nivalenol is a trichothecene mycotoxin produced by certain species of the fungus Fusarium, particularly those found on cereal crops. 15-Acetyldeoxy Nivalenol Chemical Structure
  35. GC41937 15-keto-17-phenyl trinor Prostaglandin F2α ethyl amide Bimatoprost is the Allergan trade name for 17-phenyl trinor prostaglandin F2α ethyl amide (17-phenyl trinor PGF2α ethyl amide), an F-series PG analog which has been approved for use as an ocular hypotensive drug. 15-keto-17-phenyl trinor Prostaglandin F2α ethyl amide Chemical Structure
  36. GC41309 16α-hydroxy Prednisolone 16α-hydroxy Prednisolone is a stereoselective metabolite of the 22(R) epimer of the glucocorticoid budesonide. 16α-hydroxy Prednisolone Chemical Structure
  37. GC41300 17β-hydroxy Exemestane 17β-hydroxy Exemestane is the primary active metabolite of exemestane. 17β-hydroxy Exemestane Chemical Structure
  38. GC49823 2′-C-β-Methylguanosine An active nucleoside metabolite of BMS-986094 2′-C-β-Methylguanosine Chemical Structure
  39. GC46508 2',2'-Difluoro-2'-deoxyuridine An active metabolite of gemcitabine 2',2'-Difluoro-2'-deoxyuridine Chemical Structure
  40. GC49159 2-(1-Piperazinyl)pyrimidine An α2-AR antagonist and active metabolite of azapirones 2-(1-Piperazinyl)pyrimidine Chemical Structure
  41. GC49330 2-(2-Aminoethyl)-3-(4-chlorophenyl)-3-hydroxyisoindol-1-one (hydrochloride) A metabolite of mazindol 2-(2-Aminoethyl)-3-(4-chlorophenyl)-3-hydroxyisoindol-1-one (hydrochloride) Chemical Structure
  42. GC52029 2-Aminoflubendazole 2-Aminoflubendazole Chemical Structure
  43. GC46539 2-Chloroadenine A heterocyclic building block 2-Chloroadenine Chemical Structure
  44. GC40675 2-deoxy-Artemisinin 2-deoxy-Artemisinin is an inactive metabolite of the antimalarial agent artemisinin. 2-deoxy-Artemisinin Chemical Structure
  45. GC35090 2-Hydroxy atorvastatin calcium salt An active metabolite of atorvastatin 2-Hydroxy atorvastatin calcium salt Chemical Structure
  46. GC60474 2-Hydroxy atorvastatin lactone 2-Hydroxy atorvastatin lactone is a metabolite of Atorvastatin. 2-Hydroxy atorvastatin lactone Chemical Structure
  47. GC64336 2-Hydroxyemodin 2-Hydroxyemodin is an active metabolite of emodin in the hepatic microsomes. 2-Hydroxyemodin Chemical Structure
  48. GC42189 2-oxo Clopidogrel 2-oxo Clopidogrel is an intermediary metabolite of clopidogrel. 2-oxo Clopidogrel Chemical Structure
  49. GC40968 21-hydroxy Eplerenone 21-hydroxy Eplerenone is a major metabolite of the mineralocorticoid receptor antagonist eplerenone. 21-hydroxy Eplerenone Chemical Structure
  50. GC35079 24, 25-Dihydroxy VD2 24, 25-Dihydroxy VD2 is a hydroxylated metabolite of Vitamin D2; a synthetic analog of Vitamin D. 24, 25-Dihydroxy VD2 Chemical Structure
  51. GC49365 25-Desacetyl Rifampicin A major active metabolite of rifampicin 25-Desacetyl Rifampicin Chemical Structure
  52. GC41480 3'-hydroxy Lidocaine 3'-hydroxy Lidocaine is an active metabolite of lidocaine formed by the cytochrome P450 (CYP) isoforms CYP1A2 and CYP3A4. 3'-hydroxy Lidocaine Chemical Structure
  53. GC39611 3'-Hydroxy Repaglinide 3'-Hydroxy Repaglinide is a main CYP2C8 metabolite of Repaglinide. 3'-Hydroxy Repaglinide Chemical Structure
  54. GC60500 3'-Hydroxy Repaglinide D5 3'-Hydroxy Repaglinide D5 is the deuterium labeled 3'-Hydroxy Repaglinide. 3'-Hydroxy Repaglinide D5 Chemical Structure
  55. GC68082 3,4,5-Trimethoxyphenylacetic acid 3,4,5-Trimethoxyphenylacetic acid Chemical Structure
  56. GC39841 3,4-Dehydro Cilostazol 3,4-Dehydro Cilostazol (OPC-13015) is an active metabolite of Cilostazol. 3,4-Dehydro Cilostazol Chemical Structure
  57. GC52324 3-(3-Hydroxyphenyl)propionic Acid sulfate A metabolite of certain phenols and glycosides 3-(3-Hydroxyphenyl)propionic Acid sulfate Chemical Structure
  58. GC42198 3-(4-Chlorophenyl)-4-hydroxybutyric Acid (sodium salt) An inactive metabolite of baclofen 3-(4-Chlorophenyl)-4-hydroxybutyric Acid (sodium salt) Chemical Structure
  59. GC46583 3-Amino-2,6-Piperidinedione An active metabolite of (±)-thalidomide 3-Amino-2,6-Piperidinedione Chemical Structure
  60. GC67902 3-Amino-2-oxazolidinone-d4 3-Amino-2-oxazolidinone-d4 Chemical Structure
  61. GC42274 3-hydroxy Darifenacin 3-hydroxy Darifenacin is a metabolite of darifenacin. 3-hydroxy Darifenacin Chemical Structure
  62. GC42275 3-hydroxy Desloratidine 3-hydroxy Desloratidine is a major metabolite of desloratadine , a tricyclic antagonist of the histamine H1 receptor. 3-hydroxy Desloratidine Chemical Structure
  63. GC41565 3-hydroxy Medetomidine 3-hydroxy Medetomidine is a metabolite of the α2-adrenergic receptor agonist medetomidine. 3-hydroxy Medetomidine Chemical Structure
  64. GC48457 3-keto Fusidic Acid An active metabolite of fusidic acid 3-keto Fusidic Acid Chemical Structure
  65. GC33738 3-Methoxytyramine hydrochloride (3-O-methyl Dopamine hydrochloride) 3-Methoxytyramine hydrochloride (3-O-methyl Dopamine hydrochloride) is an inactive metabolite of dopamine which can activate trace amine associated receptor 1 (TAAR1). 3-Methoxytyramine hydrochloride (3-O-methyl Dopamine hydrochloride) Chemical Structure
  66. GC68324 3-Methoxytyramine-d4 hydrochloride 3-Methoxytyramine-d4 hydrochloride Chemical Structure
  67. GC49869 3-Methoxytyrosine An active metabolite of L-DOPA 3-Methoxytyrosine Chemical Structure
  68. GC42307 3-O-methyl-L-DOPA (hydrate) 3-O-methyl-L-DOPA is a metabolite of L-DOPA, produced by the activity of catechol O-methyltransferase. 3-O-methyl-L-DOPA (hydrate) Chemical Structure
  69. GC49367 4’-hydroxy Atomoxetine Glucuronide (hydrate) A metabolite of atomoxetine 4’-hydroxy Atomoxetine Glucuronide (hydrate) Chemical Structure
  70. GC49252 4’-hydroxy Trazodone A metabolite of trazodone 4’-hydroxy Trazodone Chemical Structure
  71. GC18527 4'-hydroxy Flurbiprofen A major active metabolite of flurbiprofen 4'-hydroxy Flurbiprofen Chemical Structure
  72. GC49752 4,5-Desisopropylidene Topiramate An inactive metabolite of topiramate 4,5-Desisopropylidene Topiramate Chemical Structure
  73. GC49337 4-Acetamidobenzenesulfonamide A metabolite of asulam and sulfanilamide 4-Acetamidobenzenesulfonamide Chemical Structure
  74. GC42370 4-desmethoxy Omeprazole 4-desmethoxy Omeprazole is a potential impurity found in commercial omeprazole and esomeprazole magnesium preparations. 4-desmethoxy Omeprazole Chemical Structure
  75. GC18194 4-Epidoxycycline 4-Epidoxycycline is the 4-epimer hepatic metabolite of the antibiotic doxycycline . 4-Epidoxycycline Chemical Structure
  76. GC42401 4-hydroperoxy Cyclophosphamide An activated analog of cyclophosphamide 4-hydroperoxy Cyclophosphamide Chemical Structure
  77. GC42405 4-hydroxy Atorvastatin (calcium salt) 4-hydroxy Atorvastatin is a metabolite of atorvastatin, an HMG-CoA reductase inhibitor present in formulations that have been used to treat hypercholesterolemia and certain dyslipidemias. 4-hydroxy Atorvastatin (calcium salt) Chemical Structure
  78. GC18425 4-hydroxy Atorvastatin lactone

    4-hydroxy Atorvastatin lactone is a metabolite of atorvastatin , an HMG-CoA reductase inhibitor present in formulations that have been used to treat hypercholesterolemia and certain dyslipidemias.

     4-hydroxy Atorvastatin lactone Chemical Structure
  79. GC42407 4-hydroxy Diclofenac

    4-hydroxy Diclofenac is a CYP2C9 metabolite of the NSAID diclofenac.

     4-hydroxy Diclofenac Chemical Structure
  80. GC49575 4-hydroxy Omeprazole sulfide A metabolite of omeprazole 4-hydroxy Omeprazole sulfide Chemical Structure
  81. GC40879 4-hydroxy Solifenacin N-oxide 4-hydroxy Solifenacin N-oxide is an N-oxide form of 4-hydroxy solifenacin, the major metabolite of solifenacin . 4-hydroxy Solifenacin N-oxide Chemical Structure
  82. GC42415 4-hydroxy Valsartan 4-hydroxy Valsartan is a major metabolite of the angiotensin II type 1 (AT1) receptor antagonist valsartan. 4-hydroxy Valsartan Chemical Structure
  83. GC18417 4-hydroxy Xylazine 4-hydroxy Xylazine is a metabolite of xylazine . 4-hydroxy Xylazine Chemical Structure
  84. GC39307 4-Methylamino antipyrine 4-Methylamino antipyrine is an active metabolite of Metamizole. 4-Methylamino antipyrine Chemical Structure
  85. GC60523 4-Methylamino antipyrine hydrochloride An active metabolite of metamizole 4-Methylamino antipyrine hydrochloride Chemical Structure
  86. GC49127 4-oxo Cyclophosphamide An inactive metabolite of cyclophosphamide 4-oxo Cyclophosphamide Chemical Structure
  87. GC41399 5α-dihydro Levonorgestrel 5α-dihydro Levonorgestrel is a metabolite of the synthetic progestin levonorgestrel. 5α-dihydro Levonorgestrel Chemical Structure
  88. GC18582 5'-hydroxy Meloxicam A metabolite of meloxicam 5'-hydroxy Meloxicam Chemical Structure
  89. GC18542 5,6-dihydro-5-Fluorouracil

    5,6-dihydro-5-Fluorouracil (5-FUH2) is formed by the hydrogenation of 5-fluorouracil via the enzyme dihydropyrimidine dehydrogenase (DPD).

     5,6-dihydro-5-Fluorouracil Chemical Structure
  90. GC18466 5,6-epoxy-13-cis Retinoic Acid 5,6-epoxy-13-cis Retinoic acid is a metabolite of 13-cis retinoic acid. 5,6-epoxy-13-cis Retinoic Acid Chemical Structure
  91. GC52227 5-(3',4'-Dihydroxyphenyl)-γ-Valerolactone An active metabolite of various polyphenols 5-(3',4'-Dihydroxyphenyl)-γ-Valerolactone Chemical Structure
  92. GC49655 5-hydroxy Buspirone A metabolite of buspirone 5-hydroxy Buspirone Chemical Structure
  93. GC42546 5-hydroxy Diclofenac 5-hydroxy Diclofenac is a metabolite of the NSAID diclofenac formed by the cytochrome P450 (CYP) isoform CYP3A4. 5-hydroxy Diclofenac Chemical Structure
  94. GC49119 5-hydroxy Flunixin A metabolite of flunixin 5-hydroxy Flunixin Chemical Structure
  95. GC49315 5-hydroxy Indomethacin A metabolite of indomethacin 5-hydroxy Indomethacin Chemical Structure
  96. GC41312 5-hydroxy Omeprazole

    5-hydroxy Omeprazole is a major metabolite of omeprazole, an inhibitor of the gastric H+/K+-ATPase pump.

     5-hydroxy Omeprazole Chemical Structure
  97. GC42549 5-hydroxy Thiabendazole 5-hydroxy Thiabendazole (5-OH TBZ) is a major metabolite of the anthelmintic thiabendazole. 5-hydroxy Thiabendazole Chemical Structure
  98. GC42550 5-hydroxy-6-methoxy (S)-Duloxetine 5-hydroxy-6-methoxy (S)-Duloxetine is a metabolite of (S)-duloxetine. 5-hydroxy-6-methoxy (S)-Duloxetine Chemical Structure
  99. GC42551 5-hydroxymethyl Tolterodine (formate) 5-hydroxymethyl Tolterodine is an active metabolite of the muscarinic acetylcholine receptor antagonists tolterodine and fesoterodine. 5-hydroxymethyl Tolterodine (formate) Chemical Structure
  100. GC42586 6α-hydroxy Paclitaxel 6α-hydroxy Paclitaxel is a primary metabolite of the anticancer compound paclitaxel, produced by the action of the cytochrome P450 isoform CYP2C8. 6α-hydroxy Paclitaxel Chemical Structure
  101. GC49676 6β-hydroxy Budesonide A metabolite of budesonide 6β-hydroxy Budesonide Chemical Structure

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