mGluR

The mGluR (metabotropic glutamate receptor) is a group C GPCR and is active through an indirect metabotropic process.

Products Related to mGluR (123)

GC79304 VU6066098
CAS: 3055537-47-5
Purity: >98%
VU6066098 is a blood-brain barrier penetrant, orally active inhibitor of metabotropic glutamate receptor subtype 2 ( mGlu2 ), with IC 50 values of 77 nM and 111 nM against human and rat targets, respectively.
GC79305 MPPG TFA
Purity: >99.50%
MPPG TFA, phenylglycine analogue, is a potent and selective metabotropic glutamate receptor ( mGluR ) antagonist with a k D value of 9.2 μM.
GC79306 VU6053371
Purity: >98%
VU6053371 (BI03738809) is a first-in-class (FIC), selective, orally active, and brain-penetrant metabotropic glutamate receptor subtype 3 ( mGlu3 ) positive allosteric modulator (PAM) with EC 50 s of 103 nM and 112 nM for human and rat mGlu3.

Category Product List
Catalog No.	Product Name	CAS No.	Purity
GC79304	VU6066098	3055537-47-5	>98%
GC79304	VU6066098 is a blood-brain barrier penetrant, orally active inhibitor of metabotropic glutamate receptor subtype 2 ( mGlu2 ), with IC 50 values of 77 nM and 111 nM against human and rat targets, respectively.
GC79305	MPPG TFA	-	>99.50%
GC79305	MPPG TFA, phenylglycine analogue, is a potent and selective metabotropic glutamate receptor ( mGluR ) antagonist with a k D value of 9.2 μM.
GC79306	VU6053371	-	>98%
GC79306	VU6053371 (BI03738809) is a first-in-class (FIC), selective, orally active, and brain-penetrant metabotropic glutamate receptor subtype 3 ( mGlu3 ) positive allosteric modulator (PAM) with EC 50 s of 103 nM and 112 nM for human and rat mGlu3.