GLPBio

Estrogen/progestogen Receptor

The estrogen/progestogen receptors are activated by the hormone estrogen/progesterone and regulate the gene transcription.

Products Related to Estrogen/progestogen Receptor(156)

  • GC10245 structure
    GC10245Bazedoxifene HCl
    CAS: 198480-56-7
    Purity: >98%

    Bazedoxifene HCl (TSE-424 hydrochloride) is an oral active, BBB-penetrant nonsteroidal selective estrogen receptor modulator (SERM), with IC50s of 23 nM and 99 nM for ERα and ERβ, respectively. Bazedoxifene HCl can be used for the research of osteoporosis. Bazedoxifene HCl acts as an inhibitor of IL-6/GP130 protein-protein interactions. Bazedoxifene HCl can be used for the research of pancreatic cancer.

  • GC11282 structure
    GC11282β-Estradiol
    CAS: 50-28-2
    Purity: >99.50%

    Sex hormone

  • GC11436 structure
    GC11436Ethisterone
    CAS: 434-03-7
    Purity: >98%

    Progestogen hormone

  • GC11677 structure
    GC11677Ulipristal acetate
    CAS: 126784-99-4
    Purity: >99.50%

    Novel selective progesterone receptor modulator (SPRM)

  • GC11688 structure
    GC11688Megestrol Acetate
    CAS: 595-33-5
    Purity: >99.50%

    Anti-estrogen agent

  • GC11781 structure
    GC11781Medroxyprogesterone
    CAS: 520-85-4
    Purity: >99.00%

    potent progesterone receptor agonist

  • GC11822 structure
    GC11822Erteberel (LY500307)
    CAS: 533884-09-2
    Purity: >98.00%

    Erteberel (LY500307) (LY500307) is a potent and selective estrogen receptor beta (ERβ) agonist with Ki and EC50 of 1.54 nM and 3.61 nM, respectively.

  • GC12000 structure
    GC12000Ethynodiol diacetate
    CAS: 297-76-7
    Purity: >99.00%

    Progestogen receptor agonist

  • GC12148 structure
    GC12148Ethinyl Estradiol
    CAS: 57-63-6
    Purity: >99.50%

    Ethinyl Estradiol (17α-Ethynylestradiol;Ethynylestradiol) is an orally bio-active estrogen used in almost all modern formulations of combined oral contraceptive pills.

  • GC12182 structure
    GC12182Estriol
    CAS: 50-27-1
    Purity: >99.00%

    Estriol is an agonist of estrogen receptors (ERα and ERβ) and G protein-coupled receptor 30 (GPR30) antagonist.

  • GC12379 structure
    GC12379Drospirenone
    CAS: 67392-87-4
    Purity: >98.00%

    Synthetic progestin

  • GC12408 structure
    GC12408Progesterone
    CAS: 57-83-0
    Purity: >98.00%

    Progesterone

  • GC12974 structure
    GC12974Medroxyprogesterone acetate
    CAS: 71-58-9
    Purity: >99.50%

    Medroxyprogesterone acetate (MPA) is a synthetic progestin.

  • GC13297 structure
    GC13297Altrenogest
    CAS: 850-52-2
    Purity: >99.50%

    Progestogen receptor agonist

  • GC13350 structure
    GC13350Raloxifene HCl
    CAS: 82640-04-8
    Purity: >99.50%

    Raloxifene HCl (Keoxifene hydrochloride) is a second generationselective and orally active estrogen receptor modulator.

  • GC13835 structure
    GC13835Toremifene Citrate
    CAS: 89778-27-8
    Purity: >99.50%

    Oral selective estrogen receptor modulator (SERM)

  • GC14385 structure
    GC14385Estrone
    CAS: 53-16-7
    Purity: >98.00%

    Estrone is one of the three major endogenous estrogens, the others being estradiol and estriol.

  • GC14704 structure
    GC14704Levonorgestrel
    CAS: 797-63-7
    Purity: >98.00%

    Levonorgestrel is an effective oral progesterone inhibitor.

  • GC15324 structure
    GC15324Hexestrol
    CAS: 84-16-2
    Purity: >98.00%

    Estrogen receptor agonist

  • GC15366 structure
    GC15366Clomiphene citrate
    CAS: 50-41-9
    Purity: >98.00%

    Selective estrogen receptor modulator

  • GC15578 structure
    GC15578Dienogest
    CAS: 65928-58-7
    Purity: >98.00%

    Orally active synthetic progesterone

  • GC16292 structure
    GC16292Equol
    CAS: 94105-90-5
    Purity: >98.00%

    non-steroidal estrogen

  • GC18000 structure
    GC18000Fulvestrant (ICI 182,780)
    CAS: 129453-61-8
    Purity: >98.00%

    Fulvestrant is a selective estrogen receptor (ER) antagonist. It binds, blocks and degrades estrogen receptor, then inhibits estrogen receptor(ER)-mediated transcriptional activity with an IC 50 of 9.4 nM .

  • GC10002 structure
    GC10002Coumestrol
    CAS: 479-13-0
    Purity: >98.00%

    Coumestrol is a natural, orally active coumestan phytoestrogen. Coumestrol competitively binds estrogen receptor ERα (IC 50 =11nM) and ERβ (IC 50 =2nM) to regulate estrogen-responsive genes.