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Glucocorticoid Receptor

Glucocorticoid receptor is a neuroendocrine integration that functions as a major component of endocrine influence - specifically the stress response - upon the brain.

Products for  Glucocorticoid Receptor

  1. Cat.No. Product Name Information
  2. GC34965 (20S)-Protopanaxatriol An active ginsenoside metabolite (20S)-Protopanaxatriol  Chemical Structure
  3. GC35002 (S)-Mapracorat (S)-Mapracorat is a selective and less active glucocorticoid receptor agonist. (S)-Mapracorat  Chemical Structure
  4. GC60467 21-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione 21-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione is an intermediate of delta 9,11 steroids synthesis, for example, Vamorolone? 21-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione  Chemical Structure
  5. GC63737 21-Desacetyldeflazacort-D5 21-Desacetyldeflazacort-D5  Chemical Structure
  6. GC42587 6α-Methylprednisolone 21-hemisuccinate 6α-Methylprednisolone 21-hemisuccinate is a synthetic glucocorticoid and widely used as an anti-inflammatory agent. 6α-Methylprednisolone 21-hemisuccinate  Chemical Structure
  7. GC32405 AL 082D06 (D06) AL 082D06 (D06) is a selective, nonsteroidal glucocorticoid receptor (GR) antagonist with Ki of 210 nM. AL 082D06 (D06)  Chemical Structure
  8. GC42782 Amcinonide Amcinonide is a synthetic corticosteroid. Amcinonide  Chemical Structure
  9. GC31929 Amebucort Amebucort is a synthetic glucocorticoid corticosteroid, may used for the research of inflammatory disorders. Amebucort  Chemical Structure
  10. GC32585 AZD2906 AZD2906 is a selective glucocorticoid receptor (GR) agonist, increases micronucleated immature erythrocytes in the bone marrow of rats. AZD2906  Chemical Structure
  11. GC64949 AZD5423 AZD5423 is an inhaled, potent, selective, and non-steroidal glucocorticoid receptor (GR) modulator (SGRM). AZD5423  Chemical Structure
  12. GC19051 AZD7594 AZD7594 is a potent selective nonsteroidal glucocorticoid receptor modulator, with an IC50 of 0.9 nM. AZD7594  Chemical Structure
  13. GC31894 AZD9567 AZD9567 (compound 15) is a potent, oral active, non-steroidal and selective glucocorticoid receptor modulator (SGRM), with an IC50 of 3.8 nM. AZD9567  Chemical Structure
  14. GC33856 Beclometasone (Beclomethasone) Beclometasone (Beclomethasone) (Beclomethasone) is a prototype glucocorticoid receptor agonist. Beclometasone (Beclomethasone)  Chemical Structure
  15. GC35485 Beclometasone dipropionate Beclometasone dipropionate  Chemical Structure
  16. GC61536 Beclomethasone 17-propionate Beclomethasone 17-propionate (Beclomethasone-17-monopropionate), an active metabolite of Beclomethasone dipropionate, is a glucocorticoid receptor (GR) agonist. Beclomethasone 17-propionate  Chemical Structure
  17. GC17465 Beclomethasone dipropionate Corticosteroid used for asthma and rhinitis Beclomethasone dipropionate  Chemical Structure
  18. GC10936 Betamethasone Glucocorticoid receptor agonist Betamethasone  Chemical Structure
  19. GC35502 Betamethasone acibutate Betamethasone acibutate, derives from Betamethasone, is an acetate ester. Betamethasone acibutate  Chemical Structure
  20. GC12122 Betamethasone Dipropionate Glucocorticoid receptor agonist Betamethasone Dipropionate  Chemical Structure
  21. GC35503 Betamethasone hydrochloride Betamethasone hydrochloride is a synthetic glucocorticoid with anti-inflammatory and immunosuppressive activities. Betamethasone hydrochloride  Chemical Structure
  22. GC13638 Betamethasone Valerate anti-inflammatory corticosteroid Betamethasone Valerate  Chemical Structure
  23. GC65345 BI 653048 BI 653048 is a selective and orally active nonsteroidal?glucocorticoid (GC)?agonist with an IC50 value of 55 nM. BI 653048  Chemical Structure
  24. GC11897 Budesonide Anti-inflammatory corticosteroid Budesonide  Chemical Structure
  25. GC17571 Ciclesonide glucocorticoid Ciclesonide  Chemical Structure
  26. GC11976 Clobetasol propionate Glucocorticoid receptor agonist Clobetasol propionate  Chemical Structure
  27. GC39362 Clobetasone butyrate Clobetasone butyrate is a synthetic glucocorticoid and has topical anti-inflammatory activity especially in skin. Clobetasone butyrate  Chemical Structure
  28. GC12327 Corticosterone

    Corticosterone (17 deoxycortisol) is a glucocorticoid with oral activity and produced by adrenal cortex, which plays an important role in regulating the neuronal function of limbic system (including hippocampus, prefrontal cortex and amygdala).

    Corticosterone  Chemical Structure
  29. GC33839 Cortisone (17-Hydroxy-11-dehydrocorticosterone) Cortisone (17-Hydroxy-11-dehydrocorticosterone)  Chemical Structure
  30. GC16772 Cortisone acetate Glucocorticoid receptor agonist Cortisone acetate  Chemical Structure
  31. GC39363 Cortodoxone Cortodoxone is a glucocorticoid steroid hormone that can be oxygenated to cortisol (Hydrocortisone). Cortodoxone  Chemical Structure
  32. GC31844 Dagrocorat (PF-00251802) Dagrocorat (PF-00251802) (PF-00251802) is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor. Dagrocorat (PF-00251802)  Chemical Structure
  33. GC63872 Dagrocorat hydrochloride Dagrocorat (PF-00251802) hydrochloride is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor. Dagrocorat hydrochloride  Chemical Structure
  34. GC64330 Dazucorilant Dazucorilant (CORT113176) is a selective and high affinity non-steroidal glucocorticoid receptor (GR) modulator with a Ki value <1 nM in vitro. Dazucorilant  Chemical Structure
  35. GC12931 Deflazacort anti-inflammatory and immunosuppressant Deflazacort  Chemical Structure
  36. GC63739 Deflazacort-D5 Deflazacort-D5  Chemical Structure
  37. GC63738 Deflazacort-D7 Deflazacort-D7  Chemical Structure
  38. GC35843 Desisobutyryl-ciclesonide Desisobutyryl-ciclesonide is the active metabolite of Ciclesonide. Desisobutyryl-ciclesonide  Chemical Structure
  39. GC15690 Desonide nonfluorinated corticosteroid anti-inflammatory agent Desonide  Chemical Structure
  40. GC40775 Dexamethasone

    Dexamethasone, as one member of the glucocorticoid family, can protect against arthritis-related changes in cartilage structure and function, including matrix loss, inflammation and cartilage viability.

    Dexamethasone  Chemical Structure
  41. GC11237 Dexamethasone acetate

    IL Receptor modulator

    Dexamethasone acetate  Chemical Structure
  42. GC38573 Dexamethasone palmitate

    Dexamethasone palmitate (DXP), a lipophilic prodrug of Dexamethasone (DXM), is a glucocorticoid receptor agonist with a 47-fold lower affinity for the glucocorticoid receptor than DXM.

    Dexamethasone palmitate  Chemical Structure
  43. GC31658 Dexamethasone phosphate disodium (Dexamethasone 21-phosphate disodium salt) Dexamethasone phosphate disodium (Dexamethasone 21-phosphate disodium salt) is a glucocorticoid receptor agonist. Dexamethasone phosphate disodium (Dexamethasone 21-phosphate disodium salt)  Chemical Structure
  44. GC64466 Dexamethasone-d5 Dexamethasone-d5  Chemical Structure
  45. GC31747 Flunisolide A fluorinated corticosteroid receptor agonist Flunisolide  Chemical Structure
  46. GC11257 Fluocinolone Acetonide Glucocorticoid receptor agonist Fluocinolone Acetonide  Chemical Structure
  47. GC10714 Fluocinonide Glucocorticoid receptor agonist Fluocinonide  Chemical Structure
  48. GC40771 Fluorometholone Fluorometholone is a synthetic glucocorticoid that binds to glucocorticoid receptors (IC50 = 1.5 nM; Kd = 2.8 nM in a radioligand binding assay). Fluorometholone  Chemical Structure
  49. GC39222 Fluticasone furoate A synthetic glucocorticoid Fluticasone furoate  Chemical Structure
  50. GC13371 Fluticasone propionate

    High affinity, selective glucocorticoid receptor agonist

    Fluticasone propionate  Chemical Structure
  51. GC31885 Fosdagrocorat (PF-04171327) Fosdagrocorat (PF-04171327) (PF-04171327) is a dissociated glucocorticoid receptor agonist. Fosdagrocorat (PF-04171327)  Chemical Structure
  52. GC11399 Glucocorticoid receptor agonist Glucocorticoid receptor agonist  Chemical Structure
  53. GC62663 Glucocorticoid receptor agonist-1 Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM extracted from patent WO2017210471A1, compound 41. Glucocorticoid receptor agonist-1  Chemical Structure
  54. GC13900 GSK 9027 glucocorticoid receptor agonist GSK 9027  Chemical Structure
  55. GC31936 GW-870086 GW-870086 is a potent anti-inflammatory agent, acting as a glucocorticoid receptor agonist, with a pIC50 of 10.1 in A549 cells expressing NF-κB. GW-870086  Chemical Structure
  56. GC11551 Hydrocortisone

    Hydrocortisone, a natural glucocorticoid secreted by adrenal and extra-adrenal tissues

    Hydrocortisone  Chemical Structure
  57. GC45994 Hydrocortisone Acetate A synthetic corticosteroid Hydrocortisone Acetate  Chemical Structure
  58. GC36268 Hydrocortisone cypionate Hydrocortisone cypionate is a synthetic glucocorticoid corticosteroid and a corticosteroid ester. Hydrocortisone cypionate  Chemical Structure
  59. GC60914 Hydrocortisone hemisuccinate Hydrocortisone hemisuccinate (Hydrocortisone 21-hemisuccinate), a physiological glucocorticoid, is an orally active steroidal anti-in?ammatory drug (SAID). Hydrocortisone hemisuccinate  Chemical Structure
  60. GC36269 Hydrocortisone phosphate Hydrocortisone phosphate (Hydrocortisone 21-phosphate), a physiological glucocorticoid, and is an orally active steroidal anti-in?ammatory drug (SAID). Hydrocortisone phosphate  Chemical Structure
  61. GC14975 Loteprednol etabonate potent glucocorticoid receptor agonist Loteprednol etabonate  Chemical Structure
  62. GC68316 Loteprednol Etabonate-d5 Loteprednol Etabonate-d5  Chemical Structure
  63. GC19239 Mapracorat Mapracorat is a novel non-steroidal selective glucocorticoid receptor agonist. Mapracorat  Chemical Structure
  64. GC12974 Medroxyprogesterone acetate

    Steroidal progestin

    Medroxyprogesterone acetate  Chemical Structure
  65. GC61850 Medroxyprogesterone acetate D3 Medroxyprogesterone acetate D3  Chemical Structure
  66. GC15668 Meprednisone Glucocorticoid receptor (GR) agonist Meprednisone  Chemical Structure
  67. GC15505 Methylprednisolone A synthetic glucocorticoid Methylprednisolone  Chemical Structure
  68. GC11637 Mifepristone Progesterone receptor antagonist Mifepristone  Chemical Structure
  69. GC15746 Mometasone furoate glucocorticoid receptor agonist Mometasone furoate  Chemical Structure
  70. GC36809 OP-3633 OP-3633 is a potent and selective steroidal glucocorticoid receptor (GR) antagonist with an IC50 of 29 nM, with inhibition of GR transcriptional activity. OP-3633  Chemical Structure
  71. GC65370 ORIC-101 ORIC-101 is a highly potent and selective glucocorticoid receptor antagonist, with an EC50 of 5.6 nM. ORIC-101  Chemical Structure
  72. GC15331 Prednisolone synthetic glucocorticoid Prednisolone  Chemical Structure
  73. GC44678 Prednisolone Phosphate (sodium salt) Prednisolone Phosphate (sodium salt) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. Prednisolone Phosphate (sodium salt)  Chemical Structure
  74. GC36961 Prednisolone Tebutate Prednisolone tebutate is a synthetic glucocorticoid used as an antiinflammatory and immunosuppressant. Prednisolone Tebutate  Chemical Structure
  75. GC16450 Prednisone Glucocorticoid receptor agonist Prednisone  Chemical Structure
  76. GC36962 Prednisone acetate Prednisone acetate (Prednisone 21-acetate), the acetate salt form of prednisolone, is a glucocorticoid receptor agonist with anti-inflammatory and immunomodulating properties. Prednisone acetate  Chemical Structure
  77. GC10434 Triamcinolone synthetic glucocorticoid agonist Triamcinolone  Chemical Structure
  78. GC12611 Triamcinolone Acetonide Antiinflammatory steroid Triamcinolone Acetonide  Chemical Structure
  79. GC33868 Triamcinolone Benetonide Triamcinolone benetonide is a synthetic glucocorticoid corticosteroid with anti-inflammatory activity. Triamcinolone Benetonide  Chemical Structure
  80. GC39564 Vamorolone Vamorolone (VBP15) is a first-in-class, orally active dissociative steroidal anti-inflammatory drug and membrane-stabilizer. Vamorolone  Chemical Structure

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