Glucocorticoid Receptor
Glucocorticoid receptor is a neuroendocrine integration that functions as a major component of endocrine influence - specifically the stress response - upon the brain.
Products Related to Glucocorticoid Receptor(94)
- GC15505MethylprednisoloneCAS: 83-43-2Purity: >98.00%
Methylprednisolone is a corticosteroid that interacts with the glucocorticoid receptor and inhibits cortisol secretion with an IC50 of 1.7ng/ml.
- GC19239MapracoratCAS: 887375-26-0Purity: >99.00%
Mapracorat is a novel non-steroidal selective glucocorticoid receptor agonist.
- GC31658Dexamethasone phosphate disodium (Dexamethasone 21-phosphate disodium salt)CAS: 2392-39-4Purity: >99.50%
Dexamethasone phosphate disodium (Dexamethasone 21-phosphate disodium salt) is a glucocorticoid receptor agonist.
- GC31844Dagrocorat (PF-00251802)CAS: 1044535-52-5Purity: >98%
Dagrocorat (PF-00251802) (PF-00251802) is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor.
- GC31885Fosdagrocorat (PF-04171327)CAS: 1044535-58-1Purity: >99.00%
Fosdagrocorat (PF-04171327) (PF-04171327) is a dissociated glucocorticoid receptor agonist.
- GC32405AL 082D06 (D06)CAS: 256925-03-8Purity: >99.00%
AL 082D06 (D06) is a selective, nonsteroidal glucocorticoid receptor (GR) antagonist with Ki of 210 nM.
- GC33839Cortisone (17-Hydroxy-11-dehydrocorticosterone)CAS: 53-06-5Purity: >97.00%
Cortisone (17-Hydroxy-11-dehydrocorticosterone) is an oxidized metabolite of Cortisol with anti-inflammatory properties.
- GC33856Beclometasone (Beclomethasone)CAS: 4419-39-0Purity: >98%
Beclometasone (Beclomethasone) (Beclomethasone) is a prototype glucocorticoid receptor agonist.
- GC33868Triamcinolone BenetonideCAS: 31002-79-6Purity: >98%
Triamcinolone benetonide is a synthetic glucocorticoid corticosteroid with anti-inflammatory activity.
- GC34965(20S)-ProtopanaxatriolCAS: 34080-08-5Purity: >98.00%
(20S)-Protopanaxatriol is a metabolite derived from ginsenosides, possessing diverse biological activities and pharmacological effects.
- GC35002(S)-MapracoratCAS: 887375-15-7Purity: >99.00%
(S)-Mapracorat is a selective and less active glucocorticoid receptor agonist.
- GC35502Betamethasone acibutateCAS: 5534-05-4Purity: >98%
Betamethasone acibutate, derives from Betamethasone, is an acetate ester.
- GC35503Betamethasone hydrochlorideCAS: 956901-32-9Purity: >98%
Betamethasone hydrochloride is a synthetic glucocorticoid with anti-inflammatory and immunosuppressive activities.
- GC35843Desisobutyryl-ciclesonideCAS: 161115-59-9Purity: >95.00%
Desisobutyryl-ciclesonide is the active metabolite of Ciclesonide.
- GC36268Hydrocortisone cypionateCAS: 508-99-6Purity: >99.00%
Hydrocortisone cypionate is a synthetic glucocorticoid corticosteroid and a corticosteroid ester.
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC15505 | Methylprednisolone | 83-43-2 | >98.00% | |
Methylprednisolone is a corticosteroid that interacts with the glucocorticoid receptor and inhibits cortisol secretion with an IC50 of 1.7ng/ml. | ||||
| GC15746 | Mometasone furoate | 83919-23-7 | >99.50% | |
glucocorticoid receptor agonist | ||||
| GC16450 | Prednisone | 53-03-2 | >99.00% | |
Glucocorticoid receptor agonist | ||||
| GC19051 | AZD7594 | 1196509-60-0 | >99.00% | |
AZD7594 is a potent selective nonsteroidal glucocorticoid receptor modulator, with an IC50 of 0.9 nM. | ||||
| GC19239 | Mapracorat | 887375-26-0 | >99.00% | |
Mapracorat is a novel non-steroidal selective glucocorticoid receptor agonist. | ||||
| GC31658 | Dexamethasone phosphate disodium (Dexamethasone 21-phosphate disodium salt) | 2392-39-4 | >99.50% | |
Dexamethasone phosphate disodium (Dexamethasone 21-phosphate disodium salt) is a glucocorticoid receptor agonist. | ||||
| GC31747 | Flunisolide | 3385-03-3 | >99.50% | |
A fluorinated corticosteroid receptor agonist | ||||
| GC31844 | Dagrocorat (PF-00251802) | 1044535-52-5 | >98% | |
Dagrocorat (PF-00251802) (PF-00251802) is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor. | ||||
| GC31885 | Fosdagrocorat (PF-04171327) | 1044535-58-1 | >99.00% | |
Fosdagrocorat (PF-04171327) (PF-04171327) is a dissociated glucocorticoid receptor agonist. | ||||
| GC31894 | AZD9567 | 1893415-00-3 | >99.00% | |
AZD9567 (compound 15) is a potent, oral active, non-steroidal and selective glucocorticoid receptor modulator (SGRM), with an IC50 of 3.8 nM. | ||||
| GC31929 | Amebucort | 83625-35-8 | >99.00% | |
Amebucort is a synthetic glucocorticoid corticosteroid, may used for the research of inflammatory disorders. | ||||
| GC31936 | GW-870086 | 827319-43-7 | >98.00% | |
GW-870086 is a potent anti-inflammatory agent, acting as a glucocorticoid receptor agonist, with a pIC50 of 10.1 in A549 cells expressing NF-κB. | ||||
| GC32405 | AL 082D06 (D06) | 256925-03-8 | >99.00% | |
AL 082D06 (D06) is a selective, nonsteroidal glucocorticoid receptor (GR) antagonist with Ki of 210 nM. | ||||
| GC32585 | AZD2906 | 1034148-15-6 | >99.50% | |
AZD2906 is a selective glucocorticoid receptor (GR) agonist, increases micronucleated immature erythrocytes in the bone marrow of rats. | ||||
| GC33839 | Cortisone (17-Hydroxy-11-dehydrocorticosterone) | 53-06-5 | >97.00% | |
Cortisone (17-Hydroxy-11-dehydrocorticosterone) is an oxidized metabolite of Cortisol with anti-inflammatory properties. | ||||
| GC33856 | Beclometasone (Beclomethasone) | 4419-39-0 | >98% | |
Beclometasone (Beclomethasone) (Beclomethasone) is a prototype glucocorticoid receptor agonist. | ||||
| GC33868 | Triamcinolone Benetonide | 31002-79-6 | >98% | |
Triamcinolone benetonide is a synthetic glucocorticoid corticosteroid with anti-inflammatory activity. | ||||
| GC34965 | (20S)-Protopanaxatriol | 34080-08-5 | >98.00% | |
(20S)-Protopanaxatriol is a metabolite derived from ginsenosides, possessing diverse biological activities and pharmacological effects. | ||||
| GC35002 | (S)-Mapracorat | 887375-15-7 | >99.00% | |
(S)-Mapracorat is a selective and less active glucocorticoid receptor agonist. | ||||
| GC35485 | Beclometasone dipropionate | 5534-09-8 | >98% | |
| GC35502 | Betamethasone acibutate | 5534-05-4 | >98% | |
Betamethasone acibutate, derives from Betamethasone, is an acetate ester. | ||||
| GC35503 | Betamethasone hydrochloride | 956901-32-9 | >98% | |
Betamethasone hydrochloride is a synthetic glucocorticoid with anti-inflammatory and immunosuppressive activities. | ||||
| GC35843 | Desisobutyryl-ciclesonide | 161115-59-9 | >95.00% | |
Desisobutyryl-ciclesonide is the active metabolite of Ciclesonide. | ||||
| GC36268 | Hydrocortisone cypionate | 508-99-6 | >99.00% | |
Hydrocortisone cypionate is a synthetic glucocorticoid corticosteroid and a corticosteroid ester. | ||||
