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Home >> Signaling Pathways >> GPCR/G protein >> Glucocorticoid Receptor

Glucocorticoid Receptor

Glucocorticoid receptor is a neuroendocrine integration that functions as a major component of endocrine influence - specifically the stress response - upon the brain.

Products for  Glucocorticoid Receptor

  1. Cat.No. Product Name Information
  2. GC34965 (20S)-Protopanaxatriol

    20(S)-APPT, 20(S)-PPT

     An active ginsenoside metabolite (20S)-Protopanaxatriol Chemical Structure
  3. GC73737 (R)-GSK866 (R)-GSK866 is the (R)-enantiomer of GSK866. (R)-GSK866 Chemical Structure
  4. GC35002 (S)-Mapracorat

    (S)-ZK-245186; (S)-BOL-303242X

     (S)-Mapracorat is a selective and less active glucocorticoid receptor agonist. (S)-Mapracorat Chemical Structure
  5. GC60467 21-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione 21-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione is an intermediate of delta 9,11 steroids synthesis, for example, Vamorolone? 21-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione Chemical Structure
  6. GC63737 21-Desacetyldeflazacort-D5 21-Desacetyldeflazacort-D5 Chemical Structure
  7. GC42587 6α-Methylprednisolone 21-hemisuccinate

    Methylprednisolone 21-succinate, MPS

     6α-Methylprednisolone 21-hemisuccinate is a synthetic glucocorticoid and widely used as an anti-inflammatory agent. 6α-Methylprednisolone 21-hemisuccinate Chemical Structure
  8. GC32405 AL 082D06 (D06) AL 082D06 (D06) is a selective, nonsteroidal glucocorticoid receptor (GR) antagonist with Ki of 210 nM. AL 082D06 (D06) Chemical Structure
  9. GC42782 Amcinonide

    CL 34,699

     Amcinonide is a synthetic corticosteroid. Amcinonide Chemical Structure
  10. GC31929 Amebucort Amebucort is a synthetic glucocorticoid corticosteroid, may used for the research of inflammatory disorders. Amebucort Chemical Structure
  11. GC32585 AZD2906 AZD2906 is a selective glucocorticoid receptor (GR) agonist, increases micronucleated immature erythrocytes in the bone marrow of rats. AZD2906 Chemical Structure
  12. GC64949 AZD5423 AZD5423 is an inhaled, potent, selective, and non-steroidal glucocorticoid receptor (GR) modulator (SGRM). AZD5423 Chemical Structure
  13. GC19051 AZD7594

    AZD7594; AZ13189620

     AZD7594 is a potent selective nonsteroidal glucocorticoid receptor modulator, with an IC50 of 0.9 nM. AZD7594 Chemical Structure
  14. GC31894 AZD9567

    AZD9567

     AZD9567 (compound 15) is a potent, oral active, non-steroidal and selective glucocorticoid receptor modulator (SGRM), with an IC50 of 3.8 nM. AZD9567 Chemical Structure
  15. GC33856 Beclometasone (Beclomethasone)

    Beclometasone

     Beclometasone (Beclomethasone) (Beclomethasone) is a prototype glucocorticoid receptor agonist. Beclometasone (Beclomethasone) Chemical Structure
  16. GC35485 Beclometasone dipropionate Beclometasone dipropionate Chemical Structure
  17. GC70744 Beclometasone dipropionate-d10 Beclometasone dipropionate-d10 is the deuterium labeled Beclometasone dipropionate. Beclometasone dipropionate-d10 Chemical Structure
  18. GC61536 Beclomethasone 17-propionate Beclomethasone 17-propionate (Beclomethasone-17-monopropionate), an active metabolite of Beclomethasone dipropionate, is a glucocorticoid receptor (GR) agonist. Beclomethasone 17-propionate Chemical Structure
  19. GC17465 Beclomethasone dipropionate Corticosteroid used for asthma and rhinitis Beclomethasone dipropionate Chemical Structure
  20. GC10936 Betamethasone

    β-Methasone, NSC 39470, SCH 4831

     Glucocorticoid receptor agonist Betamethasone Chemical Structure
  21. GC35502 Betamethasone acibutate Betamethasone acibutate, derives from Betamethasone, is an acetate ester. Betamethasone acibutate Chemical Structure
  22. GC12122 Betamethasone Dipropionate Glucocorticoid receptor agonist Betamethasone Dipropionate Chemical Structure
  23. GC35503 Betamethasone hydrochloride Betamethasone hydrochloride is a synthetic glucocorticoid with anti-inflammatory and immunosuppressive activities. Betamethasone hydrochloride Chemical Structure
  24. GC13638 Betamethasone Valerate anti-inflammatory corticosteroid Betamethasone Valerate Chemical Structure
  25. GC65345 BI 653048 BI 653048 is a selective and orally active nonsteroidal?glucocorticoid (GC)?agonist with an IC50 value of 55 nM. BI 653048 Chemical Structure
  26. GC11897 Budesonide Anti-inflammatory corticosteroid Budesonide Chemical Structure
  27. GC68814 Budesonide impurity C

    Budesonide impurity C is an impurity of Budesonide. Budesonide is an inhaled corticosteroid and a glucocorticoid receptor agonist with oral activity.

     Budesonide impurity C Chemical Structure
  28. GC70575 C108297 C108297 is a selective glucocorticoid receptor (GR) modulator (GR binding Ki 0.7 nM; GR reporter gene functional Ki 0.6 nM). C108297 Chemical Structure
  29. GC17571 Ciclesonide

    CIC, RPR 251526

     glucocorticoid Ciclesonide Chemical Structure
  30. GC11976 Clobetasol propionate

    CCl-4725, CGP 9555, Clobetasol 17-Propionate

     Glucocorticoid receptor agonist Clobetasol propionate Chemical Structure
  31. GC39362 Clobetasone butyrate Clobetasone butyrate is a synthetic glucocorticoid and has topical anti-inflammatory activity especially in skin. Clobetasone butyrate Chemical Structure
  32. GC12327 Corticosterone

    17deoxy Cortisol, 11β,21DHP, NSC 9705, 11β,21dihydroxy Progesterone

     Corticosterone (17 deoxycortisol) is a glucocorticoid with oral activity and produced by adrenal cortex, which plays an important role in regulating the neuronal function of limbic system (including hippocampus, prefrontal cortex and amygdala). Corticosterone Chemical Structure
  33. GC33839 Cortisone (17-Hydroxy-11-dehydrocorticosterone) Cortisone (17-Hydroxy-11-dehydrocorticosterone) Chemical Structure
  34. GC16772 Cortisone acetate

    Cortisone 21-acetate, NSC 49420

     Glucocorticoid receptor agonist Cortisone acetate Chemical Structure
  35. GC39363 Cortodoxone Cortodoxone is a glucocorticoid steroid hormone that can be oxygenated to cortisol (Hydrocortisone). Cortodoxone Chemical Structure
  36. GC31844 Dagrocorat (PF-00251802)

    PF-00251802

     Dagrocorat (PF-00251802) (PF-00251802) is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor. Dagrocorat (PF-00251802) Chemical Structure
  37. GC63872 Dagrocorat hydrochloride

    PF-00251802 hydrochloride

     Dagrocorat (PF-00251802) hydrochloride is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor. Dagrocorat hydrochloride Chemical Structure
  38. GC64330 Dazucorilant

    CORT113176

     Dazucorilant (CORT113176) is a selective and high affinity non-steroidal glucocorticoid receptor (GR) modulator with a Ki value ＜1 nM in vitro. Dazucorilant Chemical Structure
  39. GC12931 Deflazacort

    DL-458IT, L-5,458, MDL 458

     anti-inflammatory and immunosuppressant Deflazacort Chemical Structure
  40. GC63739 Deflazacort-D5 Deflazacort-D5 Chemical Structure
  41. GC63738 Deflazacort-D7 Deflazacort-D7 Chemical Structure
  42. GC35843 Desisobutyryl-ciclesonide

    CIC-AP, des-CIC

     Desisobutyryl-ciclesonide is the active metabolite of Ciclesonide. Desisobutyryl-ciclesonide Chemical Structure
  43. GC15690 Desonide

    Budesonide acetonide

     nonfluorinated corticosteroid anti-inflammatory agent Desonide Chemical Structure
  44. GC40775 Dexamethasone

    MK-125, NSC 34521

    Dexamethasone, as one member of the glucocorticoid family, can protect against arthritis-related changes in cartilage structure and function, including matrix loss, inflammation and cartilage viability.

     Dexamethasone Chemical Structure
  45. GC11237 Dexamethasone acetate

    NSC 39471

    IL Receptor modulator

     Dexamethasone acetate Chemical Structure
  46. GC38573 Dexamethasone palmitate

    Dexamethasone 21-palmitate, DXP, Limethason

     Dexamethasone palmitate (DXP), a lipophilic prodrug of Dexamethasone (DXM), is a glucocorticoid receptor agonist with a 47-fold lower affinity for the glucocorticoid receptor than DXM. Dexamethasone palmitate Chemical Structure
  47. GC31658 Dexamethasone phosphate disodium (Dexamethasone 21-phosphate disodium salt)

    Dexamethasone 21-phosphate, Dexamethasone Sodium Phosphate

     Dexamethasone phosphate disodium (Dexamethasone 21-phosphate disodium salt) is a glucocorticoid receptor agonist. Dexamethasone phosphate disodium (Dexamethasone 21-phosphate disodium salt) Chemical Structure
  48. GC64466 Dexamethasone-d5 Dexamethasone-d5 Chemical Structure
  49. GC70442 Exicorilant Exicorilant (CORT 125281) is a selective and oral active glucocorticoid receptor (GR) antagonist, with a Ki value of 7 nM. Exicorilant Chemical Structure
  50. GC31747 Flunisolide

    RS 3999

     A fluorinated corticosteroid receptor agonist Flunisolide Chemical Structure
  51. GC11257 Fluocinolone Acetonide

    NSC 92339

     Glucocorticoid receptor agonist Fluocinolone Acetonide Chemical Structure
  52. GC10714 Fluocinonide

    NSC 101791

     Glucocorticoid receptor agonist Fluocinonide Chemical Structure
  53. GC40771 Fluorometholone

    NSC 33001, U-8614

     Fluorometholone is a synthetic glucocorticoid that binds to glucocorticoid receptors (IC50 = 1.5 nM; Kd = 2.8 nM in a radioligand binding assay). Fluorometholone Chemical Structure
  54. GC39222 Fluticasone furoate

    GSK685698, GW 685698X

     A synthetic glucocorticoid Fluticasone furoate Chemical Structure
  55. GC13371 Fluticasone propionate

    Fluticasone 17-Propionate

    High affinity, selective glucocorticoid receptor agonist

     Fluticasone propionate Chemical Structure
  56. GC31885 Fosdagrocorat (PF-04171327)

    PF-04171327

     Fosdagrocorat (PF-04171327) (PF-04171327) is a dissociated glucocorticoid receptor agonist. Fosdagrocorat (PF-04171327) Chemical Structure
  57. GC74031 GA32 GA32 (compound 58r) is potent androgen receptor (AR)/glucocorticoid receptor (GR) dual inhibitor with IC50 values of 0.13 μM and 0.83 μM for AR and GR, respectively. GA32 Chemical Structure
  58. GC11399 Glucocorticoid receptor agonist Glucocorticoid receptor agonist Chemical Structure
  59. GC62663 Glucocorticoid receptor agonist-1 Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM extracted from patent WO2017210471A1, compound 41. Glucocorticoid receptor agonist-1 Chemical Structure
  60. GC71233 Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Br Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Br is an Drug-linker conjugates for ADC that can be used as a reaction reagent for the synthesis of anti-CD40 antibody agent conjugates (ADCs). Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Br Chemical Structure
  61. GC69172 Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal

    Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal is a type of glucocorticoid receptor agonist. It can be used for anti-CD40 antibody-drug conjugate (ADC) therapy and in research related to inflammation and immune regulation.

     Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal Chemical Structure
  62. GC73858 Glucocorticoid receptor agonist-4 Glucocorticoid receptor agonist-4 (Compound Preparation 5) is a glucocorticoid receptor agonist that can be conjugated to TNF-α antibodies for the study of autoimmune and inflammatory diseases. Glucocorticoid receptor agonist-4 Chemical Structure
  63. GC71075 Glucocorticoid receptor modulator 2 Glucocorticoid receptor modulator 2 (Example 1) is a glucocorticoid receptor modulator, with an IC50 value less than 100 nM. Glucocorticoid receptor modulator 2 Chemical Structure
  64. GC13900 GSK 9027 glucocorticoid receptor agonist GSK 9027 Chemical Structure
  65. GC73736 GSK866 GSK866 is a selective glucocorticoid receptor agonist, with an IC50 of 4.6 nM. GSK866 Chemical Structure
  66. GC31936 GW-870086 GW-870086 is a potent anti-inflammatory agent, acting as a glucocorticoid receptor agonist, with a pIC50 of 10.1 in A549 cells expressing NF-κB. GW-870086 Chemical Structure
  67. GC70973 HP210 HP210 is a selective glucocorticoid receptor modulator (SGRM). HP210 Chemical Structure
  68. GC11551 Hydrocortisone

    Cortisol, Dihydrocostisone, NSC 10483

     Hydrocortisone, a natural glucocorticoid secreted by adrenal and extra-adrenal tissues Hydrocortisone Chemical Structure
  69. GC45994 Hydrocortisone Acetate

    Cortef Acetate, Hydrin 2, Hydrocortisone 21-Acetate, Hydroxycorticosterone Acetate, 17α-Hydroxycorticosterone Acetate, Isopto-Hydrocortisone

     A synthetic corticosteroid Hydrocortisone Acetate Chemical Structure
  70. GC36268 Hydrocortisone cypionate Hydrocortisone cypionate is a synthetic glucocorticoid corticosteroid and a corticosteroid ester. Hydrocortisone cypionate Chemical Structure
  71. GC60914 Hydrocortisone hemisuccinate Hydrocortisone hemisuccinate (Hydrocortisone 21-hemisuccinate), a physiological glucocorticoid, is an orally active steroidal anti-in?ammatory drug (SAID). Hydrocortisone hemisuccinate Chemical Structure
  72. GC36269 Hydrocortisone phosphate Hydrocortisone phosphate (Hydrocortisone 21-phosphate), a physiological glucocorticoid, and is an orally active steroidal anti-in?ammatory drug (SAID). Hydrocortisone phosphate Chemical Structure
  73. GC69274 INCB13739

    INCB13739 is an orally effective, selective, and tissue-specific inhibitor of 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1), with IC50 values of 3.2 nM (for the enzyme) and 1.1 nM (for PBMC). INCB13739 can be used for research on type 2 diabetes (T2DM) and obesity.

     INCB13739 Chemical Structure
  74. GC14975 Loteprednol etabonate potent glucocorticoid receptor agonist Loteprednol etabonate Chemical Structure
  75. GC68316 Loteprednol Etabonate-d5 Loteprednol Etabonate-d5 Chemical Structure
  76. GC19239 Mapracorat

    ZK-245186; BOL-303242X

     Mapracorat is a novel non-steroidal selective glucocorticoid receptor agonist. Mapracorat Chemical Structure
  77. GC12974 Medroxyprogesterone acetate

    NSC 21171, NSC 26386, U-8839

     Medroxyprogesterone acetate (MPA) is a synthetic progestin. Medroxyprogesterone acetate Chemical Structure
  78. GC61850 Medroxyprogesterone acetate D3 Medroxyprogesterone acetate D3 Chemical Structure
  79. GC15668 Meprednisone

    Methylprednisone, NSC 527579, SCH 4358

     Glucocorticoid receptor (GR) agonist Meprednisone Chemical Structure
  80. GC15505 Methylprednisolone

    Medesone, Medrol, Noretona, NSC 19987, U-7532

     Methylprednisolone is a corticosteroid that interacts with the glucocorticoid receptor and inhibits cortisol secretion with an IC50 of 1.7ng/ml. Methylprednisolone Chemical Structure
  81. GC70229 Methylprednisolone aceponate Methylprednisolone aceponate (ZK 91588) is a glucocorticoid and anti-inflammatory agent with weak systemic effects. Methylprednisolone aceponate Chemical Structure
  82. GC11637 Mifepristone

    RU486; RU 38486

     Mifepristone (RU486) is an orally effective progesterone (PR) receptor and glucocorticoid receptor (GR) antagonist used as an abortion drug with in vitro IC50 values of 0.2nM and 2.6nM, respectively . Mifepristone Chemical Structure
  83. GC15746 Mometasone furoate

    SCH 32088

     glucocorticoid receptor agonist Mometasone furoate Chemical Structure
  84. GC73137 Nenocorilant Nenocorilantis a potent, orally activity glucocorticoid receptor (GR) antagonist with Ki value of 0.15 nM. Nenocorilant Chemical Structure
  85. GC36809 OP-3633 OP-3633 is a potent and selective steroidal glucocorticoid receptor (GR) antagonist with an IC50 of 29 nM, with inhibition of GR transcriptional activity. OP-3633 Chemical Structure
  86. GC65370 ORIC-101 ORIC-101 is a highly potent and selective glucocorticoid receptor antagonist, with an EC50 of 5.6 nM. ORIC-101 Chemical Structure
  87. GC15331 Prednisolone

    NSC 9120, NSC 9900

     synthetic glucocorticoid Prednisolone Chemical Structure
  88. GC44678 Prednisolone Phosphate (sodium salt)

    Disodium Prednisolone 21Phosphate, Prednisolone Sodium Phosphate

     Prednisolone Phosphate (sodium salt) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. Prednisolone Phosphate (sodium salt) Chemical Structure
  89. GC36961 Prednisolone Tebutate Prednisolone tebutate is a synthetic glucocorticoid used as an antiinflammatory and immunosuppressant. Prednisolone Tebutate Chemical Structure
  90. GC16450 Prednisone

    1,2-Dehydrocortisone, NSC 10023

     Glucocorticoid receptor agonist Prednisone Chemical Structure
  91. GC36962 Prednisone acetate Prednisone acetate (Prednisone 21-acetate), the acetate salt form of prednisolone, is a glucocorticoid receptor agonist with anti-inflammatory and immunomodulating properties. Prednisone acetate Chemical Structure
  92. GC10434 Triamcinolone

    NSC 13397

     synthetic glucocorticoid agonist Triamcinolone Chemical Structure
  93. GC12611 Triamcinolone Acetonide

    NSC 21916

     Antiinflammatory steroid Triamcinolone Acetonide Chemical Structure
  94. GC33868 Triamcinolone Benetonide Triamcinolone benetonide is a synthetic glucocorticoid corticosteroid with anti-inflammatory activity. Triamcinolone Benetonide Chemical Structure
  95. GC39564 Vamorolone Vamorolone (VBP15) is a first-in-class, orally active dissociative steroidal anti-inflammatory drug and membrane-stabilizer. Vamorolone Chemical Structure

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