Drug Metabolite
Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.
Products Related to Drug Metabolite(546)
- GC49399N-Desbutyl Dronedarone (hydrochloride)CAS: 197431-02-0Purity: >95.00%
Debutyldronedarone (SR35021) hydrochloride, the main metabolite of Dronedarone, is a selective thyroid hormone receptor α1 (TRα1) inhibitor.
- GC49421Atorvastatin lactone-d5CAS: 125995-03-1Purity: >99.00%
An internal standard for the quantification of atorvastatin lactone
- GC49428O-Des[2-aminoethyl]-O-carboxymethyl dehydroamlodipineCAS: 113994-45-9Purity: >95.00%
A major metabolite of amlodipine
- GC49480Salicylic Acid-d4CAS: 78646-17-0Purity: >98.00%
Salicylic Acid-d4 is the deuterium labeled 2-Carboxyphenol.
- GC494886-Methylmercaptopurine-d3CAS: 33312-93-5Purity: >99.00%
An internal standard for the quantification of 6-MMP
- GC49559Hydroxymethyl Tolperisone (hydrochloride)CAS: 352233-14-8Purity: >95.00%
A metabolite of tolperisone
- GC49565RoxatidineCAS: 78273-80-0Purity: >95.00%
Roxatidine is an active metabolite of Roxatidine acetate hydrochloride, is a histamine H2-receptor antagonist.
- GC49583N-desmethyl Sertraline (hydrochloride)CAS: 675126-09-7Purity: >95.00%
A metabolite of sertraline
- GC49637O-desethyl DapagliflozinCAS: 864070-37-1Purity: >98.00%
An SGLT2 inhibitor and active metabolite of dapagliflozin
- GC49677Olmesartan-d6CAS: 1185144-74-4Purity: >99.00%
An internal standard for the quantification of olmesartan
- GC49686N-desmethyl Regorafenib N-oxideCAS: 835621-12-0Purity: >90.00%
An active metabolite of regorafenib
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC49399 | N-Desbutyl Dronedarone (hydrochloride) | 197431-02-0 | >95.00% | |
Debutyldronedarone (SR35021) hydrochloride, the main metabolite of Dronedarone, is a selective thyroid hormone receptor α1 (TRα1) inhibitor. | ||||
| GC49403 | Benzarone | 1477-19-6 | >98.00% | |
An active metabolite of benzbromarone | ||||
| GC49406 | ACT-373898 | 1433875-14-9 | >90.00% | |
A metabolite of macitentan | ||||
| GC49409 | Desmethyl Ranolazine | 172430-45-4 | >95.00% | |
A metabolite of ranolazine | ||||
| GC49410 | CVT-2738 | 5294-61-1 | >98.00% | |
An active metabolite of ranolazine | ||||
| GC49421 | Atorvastatin lactone-d5 | 125995-03-1 | >99.00% | |
An internal standard for the quantification of atorvastatin lactone | ||||
| GC49428 | O-Des[2-aminoethyl]-O-carboxymethyl dehydroamlodipine | 113994-45-9 | >95.00% | |
A major metabolite of amlodipine | ||||
| GC49480 | Salicylic Acid-d4 | 78646-17-0 | >98.00% | |
Salicylic Acid-d4 is the deuterium labeled 2-Carboxyphenol. | ||||
| GC49488 | 6-Methylmercaptopurine-d3 | 33312-93-5 | >99.00% | |
An internal standard for the quantification of 6-MMP | ||||
| GC49501 | Nirvanol | 631-07-2 | >98.00% | |
An active metabolite of mephenytoin | ||||
| GC49511 | Nicorandil N-oxide | 107833-98-7 | >98.00% | |
A metabolite of nicorandil | ||||
| GC49538 | Lamotrigine N2-oxide | 136565-76-9 | >95.00% | |
A metabolite of lamotrigine | ||||
| GC49544 | 8-hydroxy Mirtazapine | 102335-57-9 | >95.00% | |
A metabolite of mirtazapine | ||||
| GC49559 | Hydroxymethyl Tolperisone (hydrochloride) | 352233-14-8 | >95.00% | |
A metabolite of tolperisone | ||||
| GC49565 | Roxatidine | 78273-80-0 | >95.00% | |
Roxatidine is an active metabolite of Roxatidine acetate hydrochloride, is a histamine H2-receptor antagonist. | ||||
| GC49575 | 4-hydroxy Omeprazole sulfide | 103876-98-8 | >98.00% | |
A metabolite of omeprazole | ||||
| GC49583 | N-desmethyl Sertraline (hydrochloride) | 675126-09-7 | >95.00% | |
A metabolite of sertraline | ||||
| GC49627 | Rabeprazole sulfone | 117976-47-3 | >95.00% | |
A metabolite of rabeprazole | ||||
| GC49629 | 6β-hydroxy Prednisolone | 16355-29-6 | >95.00% | |
A metabolite of prednisolone | ||||
| GC49637 | O-desethyl Dapagliflozin | 864070-37-1 | >98.00% | |
An SGLT2 inhibitor and active metabolite of dapagliflozin | ||||
| GC49655 | 5-hydroxy Buspirone | 105496-33-1 | >95.00% | |
A metabolite of buspirone | ||||
| GC49676 | 6β-hydroxy Budesonide | - | >95.00% | |
A metabolite of budesonide | ||||
| GC49677 | Olmesartan-d6 | 1185144-74-4 | >99.00% | |
An internal standard for the quantification of olmesartan | ||||
| GC49686 | N-desmethyl Regorafenib N-oxide | 835621-12-0 | >90.00% | |
An active metabolite of regorafenib | ||||