Membrane Transporter/Ion Channel
Research Areas
- AMPAR(55)
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- ATPase(79)
- Calcium Channel(363)
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- Glycine Receptors(2)
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- GTPase(31)
- ICB(1)
- MCT2(2)
- Monoamine transporter(18)
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- NKCC(10)
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- Nucleoside Transporters(6)
- Pannexin-1(2)
- P2X purinergic receptor(71)
- P-gp(10)
- Proton Pump(60)
- Potassium Channel(340)
- Sodium Channel(235)
- TRP Channel(194)
- TRPV1(10)
- URAT1(14)
- Other Channel Modulators(10)
- MCT(3)
- Kainate Receptors(11)
- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(34)
- CRAC Channel(14)
- EAAT2(6)
- HCN Channel(11)
- Na+/HCO3- Cotransporter(1)
- Na+/K+ ATPase(31)
- P-glycoprotein(61)
- iGluR(190)
- nAChR(131)
- VDAC(4)
- GlyR(1)
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- Urea Transporter(1)
- Na+/H+ Exchanger (NHE)(3)
- NTPDase(5)
- EAAT(7)
- ASCT(6)
- Apical Sodium-Dependent Bile Acid Transporter(1)
- Sec61(2)
- ATP-binding cassette (ABC) transporters(5)
- SLC39 (Zinc Transporter)(2)
- Sodium Phosphate Cotransporter(1)
Products Related to Membrane Transporter/Ion Channel(2501)
- GC45180Ziconotide (trifluoroacetate salt)CAS: 1660960-77-9Purity: >95.00%
Ziconotide is a synthetic version of ω-conopeptide MVIIA, a peptide toxin originally found in the venom of the fish-eating marine snail C.
- GC45196α-Bungarotoxin (trifluoroacetate salt)Purity: >98.00%
α-Bungarotoxin is a snake venom-derived toxin that irreversibly binds nicotinic acetylcholine receptors (Ki = ~2.5 μM in rat) present in skeletal muscle, blocking action of acetylcholine at the postsynaptic membrane and leading to paralysis.
- GC45240ω-Agatoxin IVA (trifluoroacetate salt)Purity: >98.00%
ω-Agatoxin IVA is a natural peptide first isolated from the venom of funnel spiders.
- GC45241ω-Conotoxin GVIA (trifluoroacetate salt)Purity: >98.00%
ω-Conotoxin GVIA is a peptide originally isolated from the marine mollusk C.
- GC45242ω-Conotoxin MVIIC (trifluoroacetate salt)Purity: >98.00%
ω-Conotoxin MVIIC is a peptide originally isolated from the marine mollusk C.
- GC45380Aminooxyacetic AcidCAS: 645-88-5Purity: >98.00%
يعد Aminooxyacetic Acid مثبطا لإنزيم ناقلة أمين حمض جاما أمينوبوتيريك.
- GC45387AspergillimideCAS: 195966-93-9Purity: >98.00%
Aspergillimide ((rel)-Aspergillimide) ، مستقلب طارد للديدان ، معزول من البوكارا التي تم تخميرها باستخدام Aspergillus japonicas JV-23.
- GC45487IsofluraneCAS: 26675-46-7Purity: >98.00%
Isoflurane is a widely used inhalational anesthetic with a potent anesthetic effect, rapid onset, and quick elimination.
- GC45494Lavendustin BCAS: 125697-91-8Purity: >98.00%
Lavendustin B هو مثبط لتفاعل HIV-1 Integrase مع LEDGF / p75 مع IC50 من 94.07 ميكرومترLavendustin B هو مثبط GLUT1 تنافسي لـ ATP مع Ki من 15 ميكرومتريعتبر Lavendustin B أيضًا مثبطًا ضعيفًا لكينازات التيروزين
- GC45532Nε-(1-Carboxyethyl)-L-lysineCAS: 5746-03-2Purity: >95.00%
Nε-(1-Carboxyethyl)-L-lysine is an advanced glycation end product (AGE) formed by the reaction of methylglyoxal with lysine residues in proteins.
- GC45564Sematilide (hydrochloride)CAS: 101526-62-9Purity: >98.00%
Sematilide (هيدروكلوريد) (CK-1752 هيدروكلوريد) هو مانع انتقائي لقناة IKr.
- GC45879Palonosetron-d3 (hydrochloride)Purity: >99.00%
A neuropeptide with diverse biological activities
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC45150 | Voacamine | 3371-85-5 | >98.00% | |
يُظهر Voacamine ، وهو قلويد إندولي ، نشاطًا مضادًا لمستقبلات CB1 القنب القوية | ||||
| GC45159 | WOBE437 | 2108100-73-6 | >97.00% | |
WOBE437 is a potent endocannabinoid uptake inhibitor with IC50 values of 10 and 283 nM for arachidonoyl ethanolamide and 2-arachidonoyl glycerol uptake, respectively, in U937 cells. | ||||
| GC45180 | Ziconotide (trifluoroacetate salt) | 1660960-77-9 | >95.00% | |
Ziconotide is a synthetic version of ω-conopeptide MVIIA, a peptide toxin originally found in the venom of the fish-eating marine snail C. | ||||
| GC45196 | α-Bungarotoxin (trifluoroacetate salt) | - | >98.00% | |
α-Bungarotoxin is a snake venom-derived toxin that irreversibly binds nicotinic acetylcholine receptors (Ki = ~2.5 μM in rat) present in skeletal muscle, blocking action of acetylcholine at the postsynaptic membrane and leading to paralysis. | ||||
| GC45240 | ω-Agatoxin IVA (trifluoroacetate salt) | - | >98.00% | |
ω-Agatoxin IVA is a natural peptide first isolated from the venom of funnel spiders. | ||||
| GC45241 | ω-Conotoxin GVIA (trifluoroacetate salt) | - | >98.00% | |
ω-Conotoxin GVIA is a peptide originally isolated from the marine mollusk C. | ||||
| GC45242 | ω-Conotoxin MVIIC (trifluoroacetate salt) | - | >98.00% | |
ω-Conotoxin MVIIC is a peptide originally isolated from the marine mollusk C. | ||||
| GC45378 | Alaproclate (hydrochloride) | 60719-83-7 | >95.00% | |
| ||||
| GC45380 | Aminooxyacetic Acid | 645-88-5 | >98.00% | |
يعد Aminooxyacetic Acid مثبطا لإنزيم ناقلة أمين حمض جاما أمينوبوتيريك. | ||||
| GC45387 | Aspergillimide | 195966-93-9 | >98.00% | |
Aspergillimide ((rel)-Aspergillimide) ، مستقلب طارد للديدان ، معزول من البوكارا التي تم تخميرها باستخدام Aspergillus japonicas JV-23. | ||||
| GC45454 | Flumazenil-d5 | 2700278-14-2 | >99.00% | |
| ||||
| GC45487 | Isoflurane | 26675-46-7 | >98.00% | |
Isoflurane is a widely used inhalational anesthetic with a potent anesthetic effect, rapid onset, and quick elimination. | ||||
| GC45494 | Lavendustin B | 125697-91-8 | >98.00% | |
Lavendustin B هو مثبط لتفاعل HIV-1 Integrase مع LEDGF / p75 مع IC50 من 94.07 ميكرومترLavendustin B هو مثبط GLUT1 تنافسي لـ ATP مع Ki من 15 ميكرومتريعتبر Lavendustin B أيضًا مثبطًا ضعيفًا لكينازات التيروزين | ||||
| GC45532 | Nε-(1-Carboxyethyl)-L-lysine | 5746-03-2 | >95.00% | |
Nε-(1-Carboxyethyl)-L-lysine is an advanced glycation end product (AGE) formed by the reaction of methylglyoxal with lysine residues in proteins. | ||||
| GC45536 | Oleic Acid-13C | 82005-44-5 | >98.00% | |
| ||||
| GC45539 | Pantoprazole-d6 | 922727-65-9 | >99.00% | |
| ||||
| GC45557 | Safinamide-d4 | 2748522-33-8 | >99.00% | |
| ||||
| GC45564 | Sematilide (hydrochloride) | 101526-62-9 | >98.00% | |
Sematilide (هيدروكلوريد) (CK-1752 هيدروكلوريد) هو مانع انتقائي لقناة IKr. | ||||
| GC45573 | Talatisamine | 20501-56-8 | >98.00% | |
Talatisamine ، قلويد البيش ، هو مانع قناة K + محدد | ||||
| GC45675 | ML335 | 825658-06-8 | >99.50% | |
ML335 هو منشط انتقائي لكل من TREK-1 و TREK-2 | ||||
| GC45776 | LY404187 | 211311-95-4 | >98.00% | |
LY404187 عبارة عن مُعدِّل خيفي إيجابي قوي وانتقائي ونشط مركزيًا لمستقبلات AMPA ، مع EC50s من 5.65 و 0.15 و 1.44 و 1.66 و 0.21 ميكرومتر لـ GluR1i و GluR2i و GluR2o و GluR3i و GluR4i ، على التوالي. | ||||
| GC45787 | Moxidectin-d3 | - | >99.00% | |
A neuropeptide with diverse biological activities | ||||
| GC45820 | Balsalazide-d4 | - | >99.00% | |
Balsalazide-d4 هو الديوتيريوم المسمى بالسالازيد | ||||
| GC45879 | Palonosetron-d3 (hydrochloride) | - | >99.00% | |
A neuropeptide with diverse biological activities | ||||