EPZ-719 |
رقم الكتالوجGC64343 |
EPZ-719 هو مثبط جديد وقوي لـ SETD2 (IC = 0.005 ميكرومتر) مع انتقائية عالية على غيرها من هيستون ميثيل ترانسفيرازات
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2697176-16-0
Sample solution is provided at 25 µL, 10mM.
EPZ-719 is a novel and potent SETD2 inhibitor ( IC50 = 0.005 μM) with a high selectivity over other histone methyltransferases.
[1]. Lampe JW, et al. Discovery of a First-in-Class Inhibitor of the Histone Methyltransferase SETD2 Suitable for Preclinical Studies. ACS Med Chem Lett. 2021 Aug 24;12(10):1539-1545.
Average Rating: 5
(Based on Reviews and 39 reference(s) in Google Scholar.)GLPBIO products are for RESEARCH USE ONLY. Please make sure your review or question is research based.
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