Abiraterone metabolite 1 (Synonyms: 3β-OH-5α-Abi) |
رقم الكتالوجGC35219 |
مستقلب Abiraterone 1 هو مستقلب 5β مخفض من AbirateroneAbiraterone ، دواء الستيرويد ، يثبط CYP17A1 ، ويمنع تخليق الأندروجين ويطيل بقاء سرطان البروستاتا
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Cas No.: 1940176-03-3
Sample solution is provided at 25 µL, 10mM.
Abiraterone metabolite 1 is a 5β-reduced metabolite of abiraterone. Abiraterone, a steroidal drug, inhibits CYP17A1, blocks androgen synthesis and prolongs survival in prostate cancer.
[1]. Li Z, et al. Redirecting abiraterone metabolism to fine-tune prostate cancer anti-androgen therapy. Nature. 2016 May 26;533(7604):547-51.
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