Endomorphin 2 TFA |
رقم الكتالوجGC35986 |
يُظهر Endomorphin 2 TFA ، وهو ناهض انتقائي للغاية لمستقبلات μ-opioid ، تقاربات معقولة لمواقع ربط kappa3 ، مع قيمة Ki بين 20 و 30 نانومتر
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Cas No.: 1276124-00-5
Sample solution is provided at 25 µL, 10mM.
Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM[1]. Ki: 20-30 nM (kappa3 opioid receptor)[1]
[1]. Goldberg IE, et al. Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse brain. J Pharmacol Exp Ther. 1998 Aug;286(2):1007-13.
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