Endomorphin 2 TFA |
Catalog No.GC35986 |
μ-opioid 수용체의 고친화성, 고선택성 작용제인 Endomorphin 2 TFA는 kappa3 결합 부위에 대해 합리적인 친화성을 나타내며 Ki 값은 20~30nM입니다.
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Cas No.: 1276124-00-5
Sample solution is provided at 25 µL, 10mM.
Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM[1]. Ki: 20-30 nM (kappa3 opioid receptor)[1]
[1]. Goldberg IE, et al. Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse brain. J Pharmacol Exp Ther. 1998 Aug;286(2):1007-13.
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