RORγt Inverse agonist 3 |
| رقم الكتالوجGC37557 |
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2364429-77-4
Sample solution is provided at 25 µL, 10mM.
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RORγt Inverse agonist 3 is a potent, selective and orally active RORγ inverse agonist, with EC50s of 0.22 μM and 0.15 μM for hRORγ and RORγt (human IL-17 cells), respectively[1]. EC50: 0.22 μM (hRORγ), 0.15 μM (RORγt, human IL-17 cells)[1]
[1]. Amaudrut J, et al. Discovery of novel quinoline sulphonamide derivatives as potent, selective and orally active RORγ inverse agonists. Bioorg Med Chem Lett. 2019 Jul 15;29(14):1799-1806.
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