BAY-6035 |
| رقم الكتالوجGC45389 |
يعتبر BAY-6035 مثبطًا قويًا وانتقائيًا وتنافسيًا للركيزة لـ SMYD3BAY-6035 يمنع مثيلة ببتيد MEKK2 مع IC50 من 88 نانومتر
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Cas No.: 2247890-13-5
Sample solution is provided at 25 µL, 10mM.
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BAY-6035 is an inhibitor of SET and MYND domain-containing protein 3 (SMYD3). It is 100-fold selective for SMYD3 over other histone methyltransferases. BAY-6035 inhibits methylation of MEKK2 peptide in a cell-free assay and in cells (IC50s = 88 and 70 nM, respectively). See the Structural Genomic Consortium (SGC) website for more information.
References
Average Rating: 5 (Based on Reviews and 21 reference(s) in Google Scholar.)
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