- Cat.No. Nombre del producto Información
- GC42788 Aminopeptidase N Inhibitor Aminopeptidase N (AP-N) inhibitor is a reversible inhibitor of AP-N/CD13 (IC50 = 25 μM).
- GC40624 MMP-3 Inhibitor VIII Matrix metalloproteinases (MMPs) belong to a family of proteases that play a crucial role in tissue remodeling and repair by degrading extracellular matrix proteins to enable cell migration.
- GC49702 Papain Inhibitor (trifluoroacetate salt) A peptide inhibitor of papain
- GC44235 MMP Inhibitor I (trifluoroacetate salt) MMP inhibitor I is a peptide inhibitor of matrix metalloproteinase-1 (MMP-1), MMP-2, and MMP-3 (IC50s = 1.3, 30, and 150 μM, respectively).
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GC18218
MMP-3 Inhibitor
MMP-3 inhibitor is a peptide inhibitor of matrix metalloproteinase-3 (MMP-3) with a Ki value of 95 nM.
- GC18616 MMP-8 Inhibitor I MMP-8 Inhibitor I is a selective inhibitor of the neutrophil collagenase matrix metalloproteinase-8 (MMP-8) with an IC50 value of 4 nM.
- GC18315 Calpain Inhibitor VI Calpain inhibitor VI is an inhibitor of the calcium-dependent cysteine proteases u-calpain (calpain-1; IC50 = 7.5 nM) and m-calpain (calpain-2; IC50 = 78 nM).
- GC49915 Hexa-D-Arginine (trifluoroacetate salt) A furin inhibitor
- GC49704 Ac-FLTD-CMK (trifluoroacetate salt) An inhibitor of caspase-1, -4, -5, and -11
- GC49685 Trifluoroacetyl Tripeptide-2 (acetate) A peptide inhibitor of pancreatic and neutrophil elastases
- GC49605 H-Gly-Pro-Hyp-OH (acetate) A peptide DPP-4 inhibitor
- GC49322 GGACK (hydrochloride) A uPA and factor Xa inhibitor
- GC48470 Ac-DEVD-CHO (trifluoroacetate salt) A dual caspase3/caspase7 inhibitor
- GC48101 SSAA09E1 A SARS-CoV entry inhibitor
- GC46895 Aurintricarboxylic Acid (ammonium salt) A protein synthesis inhibitor with diverse biological activities
- GC45515 MX1013 MX1013 es un inhibidor dipéptido caspasa potente e irreversible con actividad antiapoptÓtica. MX1013 inhibe la caspasa 3 humana recombinante con una IC50de 30 nM.
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GC45177
Z-AEVD-FMK
Z-AEVD-FMK is an irreversible inhibitor of caspase-10 and related caspases.
- GC45066 Tosyl Phenylalanyl Chloromethyl Ketone Tosyl Phenylalanyl Chloromethyl Ketone (L-1-Tosilamido-2-feniletil clorometil cetona; L-Tosyl Phenylalanyl Chloromethyl Ketone) es un potente inhibidor de serina proteasa que reacciona con el nÚcleo de uniÓn a la proteÍna de retinoblastoma (RB) de la proteÍna E7 del VPH-18 y elimina su capacidad de uniÓn a RB.
- GC44313 Naphthofluorescein La naftofluoresceÍna inhibe la interacciÓn entre HIF-1 y Mint3. La naftofluoresceÍna suprime la actividad de HIF-1 dependiente de Mint3 y la glucÓlisis en células cancerosas y macrÓfagos sin citotoxicidad in vitro ni efectos adversos in vivo. La naftofluoresceÍna también es una sonda fluorescente sensible al pH que se puede utilizar para obtener imÁgenes funcionales de Cerenkov.
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GC43371
Dabigatran Acyl-β-D-Glucuronide
Dabigatran acyl-β-D-glucuronide is a major active metabolite of the thrombin inhibitor dabigatran.
- GC43150 CAY10406 CAY10406 is a trifluoromethyl analog of an isatin sulfonamide compound that selectively inhibits caspases 3 and 7.
- GC42721 Ac-YVAD-CMK Ac-YVAD-CMK es una inhibición caspase-1 (Ki=0.8nM) que sin reversibilidad selectivacaspase-1 (Ki=0.8nM), se puede impedir la actividad de citoquinas proinflamatorias IL-1β. Ac-YVAD-CMK puede reducir la información e induce efectos neuroprotectores duraderos.
- GC42665 AAF-CMK (trifluoroacetate salt) Tripeptidyl peptidase II (TPPII) is a serine peptidase of the subtilisin-type which removes tripeptides from the free NH2 terminus of oligopeptides.
- GC40622 Penicillide La penicillida (Vermixocin A), aislada de Talaromyces derxii cultivada en arroz, muestra actividad inhibitoria contra acil-CoA: colesterol aciltransferasa (ACAT) .
- GC40256 p-APMSF (hydrochloride) p-APMSF is an irreversible inhibitor of serine proteases with Ki values of 1.02, 1.18, 1.5, and 1.54 μM for bovine trypsin, human thrombin, bovine plasmin, and bovine Factor Xa, respectively.
- GC18699 JCP174 JCP174 es un inhibidor de la palmitoil proteÍna tioesterasa-1 (TgPPT1), una depalmitoilasa del parÁsito T.
- GC18021 Ac-YVAD-CHO Ac-YVAD-CHO (L-709049) es un inhibidor de la enzima convertidora de interleucina-1β (ICE) tetrapeptÍdico, reversible, potente y especÍfico con valores Ki humanos y de ratÓn de 3,0 y 0,76 nM.