MRS 1706 |
| Catalog No.GC10320 |
MRS 1706 es un agonista inverso potente y selectivo del receptor de adenosina A2B.
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Cas No.: 264622-53-9
Sample solution is provided at 25 µL, 10mM.
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MRS-1706 is a potent and selective adenosine A2B receptor inverse agonist. MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1 and A3 receptors respectively[1][2].
References:
[1]. Li Q, et al. ZM241385, DPCPX, MRS1706 are inverse agonists with different relative intrinsic efficacies on constitutively active mutants of the human adenosine A2B receptor. J Pharmacol Exp Ther. 2007 Feb;320(2):637-45.
[2]. Desai A, et al. Adenosine A2A receptor stimulation increases angiogenesis by down-regulating production of the antiangiogenic matrix protein thrombospondin 1. Mol Pharmacol. 2005 May;67(5):1406-13.
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