DNA Damage/DNA Repair
Research Areas
- MTH1(4)
- PARP(103)
- ATM/ATR(31)
- DNA Alkylating(23)
- DNA Ligases(3)
- DNA Methyltransferase(27)
- DNA-PK(28)
- HDAC(143)
- Nucleoside Antimetabolite/Analogue(194)
- Telomerase(15)
- Topoisomerase(193)
- tankyrase(5)
- Antifolate(33)
- CDK(299)
- Checkpoint Kinase (Chk)(36)
- CRISPR/Cas9(9)
- Deubiquitinase(84)
- DNA Alkylator/Crosslinker(87)
- DNA/RNA Synthesis(575)
- Eukaryotic Initiation Factor (eIF)(33)
- IRE1(25)
- LIM Kinase (LIMK)(12)
- TOPK(6)
- Casein Kinase(59)
- DNA Intercalating Agents(8)
- DNA/RNA Oxidative Damage(13)
- Poly(ADP-ribose) Glycohydrolase (PARG)(5)
- Early 2 Factor (E2F)(2)
- Zinc Finger Protein(1)
Products Related to DNA Damage/DNA Repair(1968)
- GC74226Biotin-PEG3-benzophenoneCAS: 756525-96-9Purity: >99.00%
Biotin-PEG3-benzophenone는 바이오틴으로 표기된 벤조페논이다.
- GC74250Thymidine-13C10,15N2CAS: 1821188-00-4Purity: >99.00%
Thymidine-13C10,15N2는 13C와 15N이 Tmidine으로 표기되어 있습니다.
- GC74261(R)-(+)-O-DemethylbuchenavianineCAS: 1364123-68-1Purity: >98.00%
(R)-(+)-O-Demethylbuchenavianine 는 세포 주기 단백질 의존성 효소 CDK의 억제제입니다.
- GC74262(S)-(-)-O-DemethylbuchenavianineCAS: 91147-18-1
(S)-(-)-O-Demethylbuchenavianine (화합물 (S) - (‐) - 1) 은 플라보노이드의 일종이다.
- GC74316ATR kinase substrate peptidePurity: >99.00%
ATR kinase substrate peptide (화합물 45)는 ATR (Ataxia Telangiectasia and Rad3 related) protein kinase (Ki=6 nM)의 강력하고 선택적인 억제제이다.
- GC74652Exatecan Intermediate 2 hydrochlorideCAS: 2437603-23-9Purity: >99.00%
Exatecan Intermediate 2 hydrochloride (화합물 B) 는 Exatecan (DX-8951) 의 중간체입니다.
- GC74653Exatecan Intermediate 4CAS: 2436720-50-0
Exatecan Intermediate 4 (화합물 B)는 엑사테탄 (DX-8951,)의 중간체이다.
- GC74654Exatecan Intermediate 4 dihydrochloridePurity: >99.00%
Exatecan Intermediate 4 dihydrochloride은 Exatecan(DX-8951)의 중간체입니다.
- GC74656Topoisomerase IIα-IN-8CAS: 1251578-67-2
Topoisomerase IIα-IN-8 (15) 화합물은 약 한 인간의 DNA topoisomerase 설계 (htIIa) 억제, 462 ±의 IC50 38.0 μ M.
- GC74684Topoisomerase II inhibitor 14CAS: 305343-00-4Purity: >99.00%
Topoisomerase II inhibitor 14 (화합물 2f) 는 토폴로지아제 II의 강력한 억제제로서 항암 활성을 가지고 있다.
- GC74712N-6-Methyl-2-deoxyadenosine-d3CAS: 1354782-02-7Purity: >99.00%
N-6-Methyl-2-deoxyadenosine-d3 는 에테르 표기 N-6 - Metl-2 - 디옥시 아데노신이다.
- GC74733Methoxyamine-d3 HydrochlorideCAS: 110220-55-8Purity: >99.00%
Methoxyamine-d3 Hydrochloride (O-Metldroxylamine-d3)는 Methoxyamine drochloride로 표기된 중수소이다.
- GC78756Mocertatug rezetecan (DAR4)CAS: 3042848-25-6Purity: >98.00%
Mocertatug rezetecan (DAR4) (HS-20089 (DAR4); GSK5733584 (DAR4)) is an antibody-drug conjugate ( ADC ) targeting B7-H4, composed of Mocertatug and MC-Gly-Gly-Phe-Gly-(R)-Cyclopropane-Exatecan.
- GC78757Mocertatug rezetecan (DAR6)CAS: 3042848-25-6Purity: >98.00%
Mocertatug rezetecan (DAR6) (HS-20089 (DAR6); GSK5733584 (DAR6)) is an antibody-drug conjugate ( ADC ) targeting B7-H4, composed of Mocertatug and MC-Gly-Gly-Phe-Gly-(R)-Cyclopropane-Exatecan.
- GC787592-MSP-5-HA-VA-PAB-ExatecanCAS: 2878440-72-1Purity: >97.50%
2-MSP-5-HA-Val-Cit-PAB-Exatecan (A-24) is a drug-linker conjugate for ADC.
- GC787602-MSP(4-OMe)-5-HA-PEG8-VA-ExatecanCAS: 3115661-30-5Purity: >97.50%
2-MSP(4-OMe)-5-HA-PEG8-VA-Exatecan is a Drug-linker conjugates for ADC consisting of the ADC Cytotoxin Exatecan and a linker.
- GC78766N-(Mal)-N-(PEG8-Val-Cit-PAB-MMAE)-N-(PEG8-Val-Cit-PAB-Exatecan)Purity: >98.00%
N-(Mal)-N-(PEG8-Val-Cit-PAB-MMAE)-N-(PEG8-Val-Cit-PAB-Exatecan) is a drug-linker conjugate for ADC (Drug-Linker Conjugate for ADC), consisting of a tubulin polymerization inhibitor MMAE and a DNA topoisomerase I inhibitor Exatecan, and an ADC linker composition.
- GC78767N-(DBCO-PEG4)-N-(PEG4-Val-Cit-PAB-MMAE)-N-(PEG4-Val-Cit-PAB-Exatecan)Purity: >98.00%
N-(DBCO-PEG4)-N-(PEG4-Val-Cit-PAB-MMAE)-N-(PEG4-Val-Cit-PAB-Exatecan) is a drug-linker conjugate for ADC (Drug-Linker Conjugate for ADC), consisting of a tubulin polymerization inhibitor MMAE and a DNA topoisomerase I inhibitor Exatecan, and an ADC linker composition.
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC74226 | Biotin-PEG3-benzophenone | 756525-96-9 | >99.00% | |
Biotin-PEG3-benzophenone는 바이오틴으로 표기된 벤조페논이다. | ||||
| GC74250 | Thymidine-13C10,15N2 | 1821188-00-4 | >99.00% | |
Thymidine-13C10,15N2는 13C와 15N이 Tmidine으로 표기되어 있습니다. | ||||
| GC74261 | (R)-(+)-O-Demethylbuchenavianine | 1364123-68-1 | >98.00% | |
(R)-(+)-O-Demethylbuchenavianine 는 세포 주기 단백질 의존성 효소 CDK의 억제제입니다. | ||||
| GC74262 | (S)-(-)-O-Demethylbuchenavianine | 91147-18-1 | - | |
(S)-(-)-O-Demethylbuchenavianine (화합물 (S) - (‐) - 1) 은 플라보노이드의 일종이다. | ||||
| GC74316 | ATR kinase substrate peptide | - | >99.00% | |
ATR kinase substrate peptide (화합물 45)는 ATR (Ataxia Telangiectasia and Rad3 related) protein kinase (Ki=6 nM)의 강력하고 선택적인 억제제이다. | ||||
| GC74324 | Cdk5i peptide | 2298317-00-5 | >99.00% | |
Cdk5i peptide는 Cdk5에서 유래한 12개 아미노산 펩타이드 조각이다. | ||||
| GC74652 | Exatecan Intermediate 2 hydrochloride | 2437603-23-9 | >99.00% | |
Exatecan Intermediate 2 hydrochloride (화합물 B) 는 Exatecan (DX-8951) 의 중간체입니다. | ||||
| GC74653 | Exatecan Intermediate 4 | 2436720-50-0 | - | |
Exatecan Intermediate 4 (화합물 B)는 엑사테탄 (DX-8951,)의 중간체이다. | ||||
| GC74654 | Exatecan Intermediate 4 dihydrochloride | - | >99.00% | |
Exatecan Intermediate 4 dihydrochloride은 Exatecan(DX-8951)의 중간체입니다. | ||||
| GC74656 | Topoisomerase IIα-IN-8 | 1251578-67-2 | - | |
Topoisomerase IIα-IN-8 (15) 화합물은 약 한 인간의 DNA topoisomerase 설계 (htIIa) 억제, 462 ±의 IC50 38.0 μ M. | ||||
| GC74684 | Topoisomerase II inhibitor 14 | 305343-00-4 | >99.00% | |
Topoisomerase II inhibitor 14 (화합물 2f) 는 토폴로지아제 II의 강력한 억제제로서 항암 활성을 가지고 있다. | ||||
| GC74712 | N-6-Methyl-2-deoxyadenosine-d3 | 1354782-02-7 | >99.00% | |
N-6-Methyl-2-deoxyadenosine-d3 는 에테르 표기 N-6 - Metl-2 - 디옥시 아데노신이다. | ||||
| GC74727 | JSH-009 | 2247481-08-7 | - | |
JSH-009은 새롭고, 매우 선택적인 CDK9억제제로 전사 연장 조절에 중요하다. | ||||
| GC74733 | Methoxyamine-d3 Hydrochloride | 110220-55-8 | >99.00% | |
Methoxyamine-d3 Hydrochloride (O-Metldroxylamine-d3)는 Methoxyamine drochloride로 표기된 중수소이다. | ||||
| GC75685 | PolQi1 | 2607139-80-8 | >98.00% | |
PolQi1 is a selective inhibitor targeting the structure domain of DNA polymerase Polθ. | ||||
| GC75826 | YL-5092 | 3056857-07-6 | >98.00% | |
YL-5092 is a novel, highly selective inhibitor of YTHDC1 (IC 50 =7.4nM; K D =29.6nM). | ||||
| GC78755 | ZW-251 | - | >98% | |
ZW-251 is a glypican-3 ( GPC3 )-targeted antibody-drug conjugate ( ADC ) with topoisomerase-I inhibitory activity. | ||||
| GC78756 | Mocertatug rezetecan (DAR4) | 3042848-25-6 | >98.00% | |
Mocertatug rezetecan (DAR4) (HS-20089 (DAR4); GSK5733584 (DAR4)) is an antibody-drug conjugate ( ADC ) targeting B7-H4, composed of Mocertatug and MC-Gly-Gly-Phe-Gly-(R)-Cyclopropane-Exatecan. | ||||
| GC78757 | Mocertatug rezetecan (DAR6) | 3042848-25-6 | >98.00% | |
Mocertatug rezetecan (DAR6) (HS-20089 (DAR6); GSK5733584 (DAR6)) is an antibody-drug conjugate ( ADC ) targeting B7-H4, composed of Mocertatug and MC-Gly-Gly-Phe-Gly-(R)-Cyclopropane-Exatecan. | ||||
| GC78759 | 2-MSP-5-HA-VA-PAB-Exatecan | 2878440-72-1 | >97.50% | |
2-MSP-5-HA-Val-Cit-PAB-Exatecan (A-24) is a drug-linker conjugate for ADC. | ||||
| GC78760 | 2-MSP(4-OMe)-5-HA-PEG8-VA-Exatecan | 3115661-30-5 | >97.50% | |
2-MSP(4-OMe)-5-HA-PEG8-VA-Exatecan is a Drug-linker conjugates for ADC consisting of the ADC Cytotoxin Exatecan and a linker. | ||||
| GC78761 | BLD1102 | 3025473-38-2 | >99.50% | |
BLD1102 is a linker-load conjugate ( Drug-Linker Conjugates for ADC ) consisting of a DNA topoisomerase I inhibitor BCPT02 and a protease-cleavable linker. | ||||
| GC78766 | N-(Mal)-N-(PEG8-Val-Cit-PAB-MMAE)-N-(PEG8-Val-Cit-PAB-Exatecan) | - | >98.00% | |
N-(Mal)-N-(PEG8-Val-Cit-PAB-MMAE)-N-(PEG8-Val-Cit-PAB-Exatecan) is a drug-linker conjugate for ADC (Drug-Linker Conjugate for ADC), consisting of a tubulin polymerization inhibitor MMAE and a DNA topoisomerase I inhibitor Exatecan, and an ADC linker composition. | ||||
| GC78767 | N-(DBCO-PEG4)-N-(PEG4-Val-Cit-PAB-MMAE)-N-(PEG4-Val-Cit-PAB-Exatecan) | - | >98.00% | |
N-(DBCO-PEG4)-N-(PEG4-Val-Cit-PAB-MMAE)-N-(PEG4-Val-Cit-PAB-Exatecan) is a drug-linker conjugate for ADC (Drug-Linker Conjugate for ADC), consisting of a tubulin polymerization inhibitor MMAE and a DNA topoisomerase I inhibitor Exatecan, and an ADC linker composition. | ||||
