GPCR/G protein

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Products Related to GPCR/G protein(3538)

GC79253 (Rac)-Ulotaront hydrochloride
CAS: 1310422-02-6
Purity: >98.00%
(Rac)-Ulotaront hydrochloride ((Rac)-SEP-363856 hydrochloride) is the racemate of Ulotaront hydrochloride.
GC79254 TGF-8027
Purity: >98%
TGF-8027 is a selective 5-HT 2A agonist that can cross the blood-brain barrier.
GC79255 EGIS-7625 free base
CAS: 751462-86-9
Purity: >99.50%
EGIS-7625 free base is an orally active and selective competitive antagonist of 5-HT2B receptor, with a human K i value of 1 nM.
GC79256 GR119566X
CAS: 237752-42-0
Purity: >98%
GR119566X is a 5-HT 3 receptor ligand with a pK i value of 8.80 against prufied 5-HT 3 receptor.
GC79257 PF-04781340 TFA
Purity: >99.50%
PF-04781340 TFA is a potent and selective 5-HT 2 C receptor agonist, with an EC 50 of 9 nM and a K i of 3 nM, respectively.
GC79258 GR119566X dihydrochloride
Purity: >98.00%
GR119566X dihydrochloride is a 5-HT 3 receptor ligand with a pK i value of 8.80 against prufied 5-HT 3 receptor.
GC79259 TMU4142
Purity: >98.50%
TMU4142 is a selective 5-HT 1a agonist with high GoA activity.
GC79260 Methyl-2-bromo-LSD
CAS: 50484-98-5
Purity: >98%
Methyl-2-bromo-LSD is a brain-penetrant 5-HT 2 receptor ligand.
GC79261 LY334370 fumarate
CAS: 182563-09-3
Purity: >99.50%
LY334370 fumarate is the fumarate of LY334370.
GC79262 SB-216641
CAS: 170230-39-4
Purity: >98%
SB-216641 is a selective 5-HT1b antagonist.
GC79263 (R)-Octopamine
CAS: 876-04-0
Purity: >95.00%
(R)-Octopamine is a Gs-coupled receptor agonist.
GC79264 Tuaminoheptane sulfate
CAS: 6411-75-2
Purity: >98%
Tuaminoheptane sulfate is an alpha- adrenergic receptor agonist.
GC79265 Toliprolol
CAS: 2933-94-0
Purity: >99.50%
Toliprolol is a β 1 /β 2 -selective β- adrenergic Receptor antagonist.
GC79266 α2AR agonist 2
CAS: 719277-27-7
Purity: >99.00%
α2AR agonist 2 is a selective α2B adrenergic receptor antagonist ( IC 50 = 1.2 µM).
GC79267 Brefonalol hydrochloride
CAS: 3026677-28-8
Purity: >98.00%
Brefonalol (Brefanolol) hydrochloride is an orally active, non-selective β-adrenergic receptor blocker with vasodilatory properties.
GC79268 α1A/1D-Adrenoceptor antagonist-1
CAS: 1049442-53-6
Purity: >99.50%
α1A/1D-Adrenoceptor antagonist-1 (Compound 15) is a selective α1A/1D-adrenoceptor dual antagonist with IC 50 values of 20.26 and 164.9 nM.
GC79269 KMCA-0011
Purity: >99.50%
KMCA-0011 is an orally active ɑ 2C adrenoceptor antagonist ( K i = 56.7 nM).
GC79270 PF-610355 hydrochloride
Purity: >98.00%
PF-610355 hydrochloride is a β2 - adrenergic receptor ( β2-AR ) full agonist with selectivity for β1-adrenergic receptors.
GC79271 RESA peptide
CAS: 133699-13-5
Purity: >99.50%
RESA peptide is a substrate peptide of β-adrenergic receptor kinase (βARK).
GC79272 Napamezole hydrochloride
CAS: 87495-33-8
Purity: >98.50%
Napamezole hydrochloride is an orally active α-2 adrenergic receptor antagonist and serotonin ( 5-HT Receptor ) reuptake inhibitor, with K i values of 28 nM and 93 nM for rat α-2 and α-1 adrenergic receptors, respectively.
GC79273 β2AR-IN-15
CAS: 2088234-50-6
Purity: >98.50%
β2AR-IN-15 is a selective β2-adrenergic receptor ( β2AR ) antagonist with a K d of 1.7 μM.
GC79274 CTR/AMYR modulator-2
CAS: 3108095-52-6
Purity: >98.00%
CTR/AMYR modulator-2 is a dual agonist of human amylin receptor 3 ( AMY3R ) and calcitonin receptor ( CTR ).
GC79275 KBP-089
CAS: 1776112-67-4
Purity: >99.00%
KBP-089 is a dual Amylin and Calcitonin Receptor agonist.
GC79276 Gramine-d 2
CAS: 95415-84-2
Purity: >98%
Gramine-d 2 is the deuterium labeled Gramine [1] . Gramine (Donaxine) is a natural alkaloid isolated from giant reed [2] , acts as an active adiponectin receptor (AdipoR) agonist, with IC 50 s of 3.2 and 4.2 μM for AdipoR2 and AdipoR1, respectively [2] . Gramine is also a human and mouse β2-Adrenergic receptor (β2-AR) agonist [3] . Gramine (Donaxine) has anti-tumor, anti-viral and anti-inflammatory properties [2] .

Category Product List
Catalog No.	Product Name	CAS No.	Purity
GC79253	(Rac)-Ulotaront hydrochloride	1310422-02-6	>98.00%
GC79253	(Rac)-Ulotaront hydrochloride ((Rac)-SEP-363856 hydrochloride) is the racemate of Ulotaront hydrochloride.
GC79254	TGF-8027	-	>98%
GC79254	TGF-8027 is a selective 5-HT 2A agonist that can cross the blood-brain barrier.
GC79255	EGIS-7625 free base	751462-86-9	>99.50%
GC79255	EGIS-7625 free base is an orally active and selective competitive antagonist of 5-HT2B receptor, with a human K i value of 1 nM.
GC79256	GR119566X	237752-42-0	>98%
GC79256	GR119566X is a 5-HT 3 receptor ligand with a pK i value of 8.80 against prufied 5-HT 3 receptor.
GC79257	PF-04781340 TFA	-	>99.50%
GC79257	PF-04781340 TFA is a potent and selective 5-HT 2 C receptor agonist, with an EC 50 of 9 nM and a K i of 3 nM, respectively.
GC79258	GR119566X dihydrochloride	-	>98.00%
GC79258	GR119566X dihydrochloride is a 5-HT 3 receptor ligand with a pK i value of 8.80 against prufied 5-HT 3 receptor.
GC79259	TMU4142	-	>98.50%
GC79259	TMU4142 is a selective 5-HT 1a agonist with high GoA activity.
GC79260	Methyl-2-bromo-LSD	50484-98-5	>98%
GC79260	Methyl-2-bromo-LSD is a brain-penetrant 5-HT 2 receptor ligand.
GC79261	LY334370 fumarate	182563-09-3	>99.50%
GC79261	LY334370 fumarate is the fumarate of LY334370.
GC79262	SB-216641	170230-39-4	>98%
GC79262	SB-216641 is a selective 5-HT1b antagonist.
GC79263	(R)-Octopamine	876-04-0	>95.00%
GC79263	(R)-Octopamine is a Gs-coupled receptor agonist.
GC79264	Tuaminoheptane sulfate	6411-75-2	>98%
GC79264	Tuaminoheptane sulfate is an alpha- adrenergic receptor agonist.
GC79265	Toliprolol	2933-94-0	>99.50%
GC79265	Toliprolol is a β 1 /β 2 -selective β- adrenergic Receptor antagonist.
GC79266	α2AR agonist 2	719277-27-7	>99.00%
GC79266	α2AR agonist 2 is a selective α2B adrenergic receptor antagonist ( IC 50 = 1.2 µM).
GC79267	Brefonalol hydrochloride	3026677-28-8	>98.00%
GC79267	Brefonalol (Brefanolol) hydrochloride is an orally active, non-selective β-adrenergic receptor blocker with vasodilatory properties.
GC79268	α1A/1D-Adrenoceptor antagonist-1	1049442-53-6	>99.50%
GC79268	α1A/1D-Adrenoceptor antagonist-1 (Compound 15) is a selective α1A/1D-adrenoceptor dual antagonist with IC 50 values of 20.26 and 164.9 nM.
GC79269	KMCA-0011	-	>99.50%
GC79269	KMCA-0011 is an orally active ɑ 2C adrenoceptor antagonist ( K i = 56.7 nM).
GC79270	PF-610355 hydrochloride	-	>98.00%
GC79270	PF-610355 hydrochloride is a β2 - adrenergic receptor ( β2-AR ) full agonist with selectivity for β1-adrenergic receptors.
GC79271	RESA peptide	133699-13-5	>99.50%
GC79271	RESA peptide is a substrate peptide of β-adrenergic receptor kinase (βARK).
GC79272	Napamezole hydrochloride	87495-33-8	>98.50%
GC79272	Napamezole hydrochloride is an orally active α-2 adrenergic receptor antagonist and serotonin ( 5-HT Receptor ) reuptake inhibitor, with K i values of 28 nM and 93 nM for rat α-2 and α-1 adrenergic receptors, respectively.
GC79273	β2AR-IN-15	2088234-50-6	>98.50%
GC79273	β2AR-IN-15 is a selective β2-adrenergic receptor ( β2AR ) antagonist with a K d of 1.7 μM.
GC79274	CTR/AMYR modulator-2	3108095-52-6	>98.00%
GC79274	CTR/AMYR modulator-2 is a dual agonist of human amylin receptor 3 ( AMY3R ) and calcitonin receptor ( CTR ).
GC79275	KBP-089	1776112-67-4	>99.00%
GC79275	KBP-089 is a dual Amylin and Calcitonin Receptor agonist.
GC79276	Gramine-d 2	95415-84-2	>98%
GC79276	Gramine-d 2 is the deuterium labeled Gramine [1] . Gramine (Donaxine) is a natural alkaloid isolated from giant reed [2] , acts as an active adiponectin receptor (AdipoR) agonist, with IC 50 s of 3.2 and 4.2 μM for AdipoR2 and AdipoR1, respectively [2] . Gramine is also a human and mouse β2-Adrenergic receptor (β2-AR) agonist [3] . Gramine (Donaxine) has anti-tumor, anti-viral and anti-inflammatory properties [2] .