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CarbinoxaMine Maleate (Synonyms: NSC 62362)

Catalog No.GC13757 Copy One-Click Copy Product Info

CarbinoxaMine Maleate es un antagonista del receptor de histamina H1.

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CarbinoxaMine Maleate Chemical Structure

Cas No.: 3505-38-2

Tamaño Precio Disponibilidad Cantidad
100mg
46,00 $
Disponible
500mg
140,00 $
Disponible

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Based on customer reviews.

Sample solution is provided at 25 µL, 10mM.



Description of CarbinoxaMine Maleate

Carbinoxamine maleate salt is a histamine H1 receptor antagonist.

References:
[1]. Harikrishnan A, et al. The cooperative effect of Lewis pairs in the Friedel-Crafts hydroxyalkylation reaction: a simple and effective route for the synthesis of (±)-carbinoxamine. Org Biomol Chem. 2015 Mar 28;13(12):3633-47.

Chemical Properties of CarbinoxaMine Maleate

Cas No. 3505-38-2 SDF
Sinónimos NSC 62362
Chemical Name 2-((4-chlorophenyl)(pyridin-2-yl)methoxy)-N,N-dimethylethanamine maleate
Canonical SMILES CN(CCOC(C1=NC=CC=C1)C2=CC=C(Cl)C=C2)C.OC(/C=C\C(O)=O)=O
Formula C16H19ClN2O.C4H4O4 M.Wt 406.86
Solubility DMSO : 100 mg/mL (245.78 mM; Need ultrasonic); H2O : 50 mg/mL (122.89 mM; Need ultrasonic) Storage Store at -20°C
General tips Please select the appropriate solvent to prepare the stock solution according to the solubility of the product in different solvents; once the solution is prepared, please store it in separate packages to avoid product failure caused by repeated freezing and thawing.Storage method and period of the stock solution: When stored at -80°C, please use it within 6 months; when stored at -20°C, please use it within 1 month.
To increase solubility, heat the tube to 37°C and then oscillate in an ultrasonic bath for some time.
Shipping Condition Evaluation sample solution: shipped with blue ice. All other sizes available: with RT, or with Blue Ice upon request.

Complete Stock Solution Preparation Table of CarbinoxaMine Maleate

Prepare stock solution
1 mg 5 mg 10 mg
1 mM 2.4578 mL 12.2892 mL 24.5785 mL
5 mM 491.6 μL 2.4578 mL 4.9157 mL
10 mM 245.8 μL 1.2289 mL 2.4578 mL
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In vivo Formulation Calculator (Clear solution) of CarbinoxaMine Maleate

Step 1: Enter information below (Recommended: An additional animal making an allowance for loss during the experiment)

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Step 2: Enter the in vivo formulation (This is only the calculator, not formulation. Please contact us first if there is no in vivo formulation at the solubility Section.)

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Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO ( Master liquid concentration mg/mL, Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug. )

Method for preparing in vivo formulation: Take μL DMSO master liquid, next addμL PEG300, mix and clarify, next addμL Tween 80, mix and clarify, next add μL saline, mix and clarify.

Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

Note: 1. Please make sure the liquid is clear before adding the next solvent.
2. Be sure to add the solvent(s) in order. You must ensure that the solution obtained, in the previous addition, is a clear solution before proceeding to add the next solvent. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.
3. All of the above co-solvents are available for purchase on the GlpBio website.

Product Documents

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Review for CarbinoxaMine Maleate

Average Rating: 5 ★★★★★ (Based on Reviews and 3 reference(s) in Google Scholar.)

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