CB2R-IN-1 |
Catalog No.GC33756 |
CB2R-IN-1 es un potente agonista inverso del receptor cannabinoide CB2 con una Ki de 0,9 nM.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1257555-79-5
Sample solution is provided at 25 µL, 10mM.
CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM.
CB2R-IN-1 (Compound 37) is a potent cannabinoid CB2 receptor ligand (Ki=0.9 nM) with excellent selectivity over the CB1 receptor (Ki=8259.3 nM)[1].
[1]. Tong L, et al. Expansion of SAR studies on triaryl bis sulfone cannabinoid CB2 receptor ligands. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6785-9.
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