DRAK2-IN-1 |
Catalog No.GC65140 |
DRAK2-IN-1, compuesto 16, es un inhibidor de DRAK2 potente, selectivo y competitivo con ATP con valores IC50 y Ki de 3 nM y 0,26 nM, respectivamente.
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Cas No.: 871837-60-4
Sample solution is provided at 25 µL, 10mM.
DRAK2-IN-1, compound 16, is a potent, selective and ATP-competitive DRAK2 inhibitor with IC50and Kivalues of 3 nM and 0.26 nM, respectively.DRAK2-IN-1 also has inbitory effect on DRAK1 (IC50=51 nM)[1].
[1]. Jung ME, et al.Discovery of indirubin derivatives as new class of DRAK2 inhibitors from high throughput screening.Bioorg Med Chem Lett. 2016 Jun 1;26(11):2719-23
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(Based on Reviews and 30 reference(s) in Google Scholar.)GLPBIO products are for RESEARCH USE ONLY. Please make sure your review or question is research based.
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