DRAK2-IN-1 |
| Katalog-Nr.GC65140 |
DRAK2-IN-1, Verbindung 16, ist ein potenter, selektiver und ATP-kompetitiver DRAK2-Inhibitor mit IC50- und Ki-Werten von 3 nM bzw. 0,26 nM.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 871837-60-4
Sample solution is provided at 25 µL, 10mM.
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DRAK2-IN-1, compound 16, is a potent, selective and ATP-competitive DRAK2 inhibitor with IC50and Kivalues of 3 nM and 0.26 nM, respectively.DRAK2-IN-1 also has inbitory effect on DRAK1 (IC50=51 nM)[1].
[1]. Jung ME, et al.Discovery of indirubin derivatives as new class of DRAK2 inhibitors from high throughput screening.Bioorg Med Chem Lett. 2016 Jun 1;26(11):2719-23
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