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Citrullination

Products for  Citrullination

  1. Cat.No. Nombre del producto Información
  2. GC48495 BMS-P5 BMS-P5 es un inhibidor de la peptidilarginina deiminasa 4 (PAD4) especÍfico y activo por vÍa oral. BMS-P5 bloquea la formaciÓn de NET inducida por MM y retrasa la progresiÓn de MM en un modelo de ratÓn singénico. BMS-P5  Chemical Structure
  3. GC43202 CAY10723

    CAY10723 es un potente inhibidor de la proteína arginina deiminasa 2 (PAD2) y tiene una excelente selectividad hacia PAD2.

    CAY10723  Chemical Structure
  4. GC47050 CAY10727 A PAD3 inhibitor CAY10727  Chemical Structure
  5. GC52351 Citrullinated α-Enolase (R8 + R14) (1-19)-biotin Peptide A biotinylated and citrullinated α-enolase peptide Citrullinated α-Enolase (R8 + R14) (1-19)-biotin Peptide  Chemical Structure
  6. GC52363 Citrullinated Histone H3 (R2 + R8 + R17) (2-22)-biotin Peptide

    A biotinylated and citrullinated histone H3 peptide

    Citrullinated Histone H3 (R2 + R8 + R17) (2-22)-biotin Peptide  Chemical Structure
  7. GC52367 Citrullinated Vimentin (G146R) (R144 + R146) (139-159)-biotin Peptide A biotinylated and citrullinated mutant vimentin peptide Citrullinated Vimentin (G146R) (R144 + R146) (139-159)-biotin Peptide  Chemical Structure
  8. GC52370 Citrullinated Vimentin (R144) (139-159)-biotin Peptide A biotinylated and citrullinated vimentin peptide Citrullinated Vimentin (R144) (139-159)-biotin Peptide  Chemical Structure
  9. GC43275 Citrulline-specific Probe-Rhodamine Protein arginine deiminases (PADs) catalyze the posttranslational modification of arginine residues on proteins to form citrulline, which plays a large role in regulating gene expression. Citrulline-specific Probe-Rhodamine  Chemical Structure
  10. GC43651 F-Amidine (trifluoroacetate salt) F-amidine is an inhibitor of protein arginine deiminases (PADs) that is selective for PAD1 and PAD4 (IC50s = 29.5, 350, and 21.6 μM for PAD1, PAD3, and PAD4 in vitro, respectively). F-Amidine (trifluoroacetate salt)  Chemical Structure
  11. GC43787 GSK106 (hydrochloride) GSK106 (clorhidrato) es un control inactivo para los inhibidores selectivos de PAD4, GSK484 y GSK199. GSK106 (hydrochloride)  Chemical Structure
  12. GC43788 GSK121 (trifluoroacetate salt) GSK-121 Trifluoroacetatos un inhibidor selectivo de PAD4. GSK121 (trifluoroacetate salt)  Chemical Structure
  13. GC43789 GSK199 (hydrochloride) GSK199 (clorhidrato) es un inhibidor reversible y selectivo de PAD4 con una IC50 de 200 nM en ausencia de calcio. GSK199 (hydrochloride)  Chemical Structure
  14. GC45548 Photoswitchable PAD Inhibitor (technical grade)   Photoswitchable PAD Inhibitor (technical grade)  Chemical Structure
  15. GC52364 Vimentin (139-159)-biotin Peptide A biotinylated vimentin peptide Vimentin (139-159)-biotin Peptide  Chemical Structure
  16. GC52371 Vimentin (G146R) (139-159)-biotin Peptide A biotinylated mutant vimentin peptide Vimentin (G146R) (139-159)-biotin Peptide  Chemical Structure

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