Citrullination
Products for Citrullination
- Cat.No. Nombre del producto Información
- GC48495 BMS-P5 BMS-P5 es un inhibidor de la peptidilarginina deiminasa 4 (PAD4) especÍfico y activo por vÍa oral. BMS-P5 bloquea la formaciÓn de NET inducida por MM y retrasa la progresiÓn de MM en un modelo de ratÓn singénico.
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GC43202
CAY10723
CAY10723 es un potente inhibidor de la proteína arginina deiminasa 2 (PAD2) y tiene una excelente selectividad hacia PAD2.
- GC47050 CAY10727 A PAD3 inhibitor
- GC52351 Citrullinated α-Enolase (R8 + R14) (1-19)-biotin Peptide A biotinylated and citrullinated α-enolase peptide
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GC52363
Citrullinated Histone H3 (R2 + R8 + R17) (2-22)-biotin Peptide
A biotinylated and citrullinated histone H3 peptide
- GC52367 Citrullinated Vimentin (G146R) (R144 + R146) (139-159)-biotin Peptide A biotinylated and citrullinated mutant vimentin peptide
- GC52370 Citrullinated Vimentin (R144) (139-159)-biotin Peptide A biotinylated and citrullinated vimentin peptide
- GC43275 Citrulline-specific Probe-Rhodamine Protein arginine deiminases (PADs) catalyze the posttranslational modification of arginine residues on proteins to form citrulline, which plays a large role in regulating gene expression.
- GC43651 F-Amidine (trifluoroacetate salt) F-amidine is an inhibitor of protein arginine deiminases (PADs) that is selective for PAD1 and PAD4 (IC50s = 29.5, 350, and 21.6 μM for PAD1, PAD3, and PAD4 in vitro, respectively).
- GC43787 GSK106 (hydrochloride) GSK106 (clorhidrato) es un control inactivo para los inhibidores selectivos de PAD4, GSK484 y GSK199.
- GC43788 GSK121 (trifluoroacetate salt) GSK-121 Trifluoroacetatos un inhibidor selectivo de PAD4.
- GC43789 GSK199 (hydrochloride) GSK199 (clorhidrato) es un inhibidor reversible y selectivo de PAD4 con una IC50 de 200 nM en ausencia de calcio.
- GC45548 Photoswitchable PAD Inhibitor (technical grade)
- GC52364 Vimentin (139-159)-biotin Peptide A biotinylated vimentin peptide
- GC52371 Vimentin (G146R) (139-159)-biotin Peptide A biotinylated mutant vimentin peptide