Phosphodiesterase

Cat.No. Nombre del producto Información

GC46030 3,3'-((2-Chlorophenyl)methylene)bis(4-hydroxy-2H-chromen-2-one) An ENPP1 inhibitor

3,3'-((2-Chlorophenyl)methylene)bis(4-hydroxy-2H-chromen-2-one) Chemical Structure

GC40692 3-Propylxanthine La 3-propilxantina actÚa como antagonista selectivo y competitivo de los receptores A2B con Ki de 7 μM. 3-Propylxanthine Chemical Structure

GC46867 Apremilast-d5 Apremilast D5 (CC-10004 D5) es un apremilast etiquetado con deuterio. Apremilast-d5 Chemical Structure

GC42951 BMP-22 BMP-22 is an inhibitor of autotaxin (IC50 = 170 nM). BMP-22 Chemical Structure

GC49079 C82 An Mtb CdnP inhibitor C82 Chemical Structure

GC41449 Carbazeran Carbazeran, un potente inhibidor de la fosfodiesterasa, es sustrato de la aldehÍdo oxidasa. Carbazeran Chemical Structure

GC46114 CAY10761 An ENPP1 inhibitor CAY10761 Chemical Structure

GC47088 Cilostazol-d4 An internal standard for the quantification of cilostazol Cilostazol-d4 Chemical Structure

GC43574 Drotaverine (hydrochloride) Drotaverine is an alkaloid that has been described as an inhibitor of phosphodiesterase 4 and negative allosteric modulator of L-type Ca2+ channels. Drotaverine (hydrochloride) Chemical Structure

Drotaverine (hydrochloride) Chemical Structure

GC46138 ENPP1 Inhibitor C El inhibidor C de ENPP1 (Compuesto C) es un potente inhibidor de ENPP1 (ectonucleÓtido pirofosfatasa/fosfodiesterasa 1) con valores IC50 de 0,26, 0,48 y 2,0 μ M evaluado mediante ensayos de TG-mAMP, pNP-TMP y ATP, respectivamente. TG (Tokyo Green)-mAMP: una sonda de fluorescencia ENPP1 sensible recién sintetizada. ENPP1 Inhibitor C Chemical Structure

GC48856 Fenspiride-d5 An internal standard for the quantification of fenspiride Fenspiride-d5 Chemical Structure

GC60886 GSK356278 GSK356278 es un inhibidor de la fosfodiesterasa 4 (PDE4) potente, selectivo, biodisponible por vÍa oral y que penetra en el cerebro, con pIC50 de 8,6, 8,8 y 8,7 para las PDE4A, PDE4B y PDE4D humanas, respectivamente. GSK356278 Chemical Structure

GC48469 Moexipril-d5 An internal standard for the quantification of moexipril Moexipril-d5 Chemical Structure

GC49683 N-desethyl-N-methyl Vardenafil A potential impurity found in commercial preparations of vardenafil

N-desethyl-N-methyl Vardenafil Chemical Structure

GC49186 O-Demethyl Apremilast An active metabolite of apremilast O-Demethyl Apremilast Chemical Structure

GC49349 O-Desethyl Sildenafil A metabolite of sildenafil O-Desethyl Sildenafil Chemical Structure

GC47931 PDE4B Inhibitor A PDE4B inhibitor PDE4B Inhibitor Chemical Structure

GC41635 Phosphodiesterase 4 Inhibitor Phosphodiesterase 4 (PDE4) inhibitor is an inhibitor of PDE4 with an IC50 value of 0.10 μM for the human recombinant enzyme.

Phosphodiesterase 4 Inhibitor Chemical Structure

GC44673 PQ-10 PQ-10 es un potente inhibidor de la fosfodiesterasa 10A (PDE10A) con IC50 y ED50 de 4,6 nM y 13 mg/kg, respectivamente. PQ-10 Chemical Structure

GC46208 Propentofylline La propentofilina es un derivado de la xantina que inhibe la captaciÓn de adenosina y bloquea la actividad de la fosfodiesterasa. Propentofylline Chemical Structure

GC45903 Quazinone A PDE3 inhibitor Quazinone Chemical Structure

GC48057 Roflumilast-d4 An internal standard for the quantification of roflumilast Roflumilast-d4 Chemical Structure

GC10005 SEP-0372814 A PDE10A inhibitor SEP-0372814 Chemical Structure

GC48078 Sildenafil-d3 Sildenafil-d3 es Sildenafil-d3 etiquetado con deuterio. Sildenafil-d3 Chemical Structure

GC48121 Tadalafil-d3 An internal standard for the quantification of tadalafil Tadalafil-d3 Chemical Structure

GC48163 Theophylline-d6 La teofilina-d6 (1,3-dimetilxantina-d6) es la teofilina marcada con deuterio. La teofilina es un inhibidor no selectivo de la fosfodiesterasa (PDE), un bloqueador del receptor de adenosina y un activador de la histona desacetilasa (HDAC). Theophylline-d6 Chemical Structure

GC48243 Vardenafil-d5 An internal standard for the quantification of vardenafil Vardenafil-d5 Chemical Structure

Products for Phosphodiesterase