Pipamperone |
رقم الكتالوجGC36924 |
Pipamperone (Floropipamide ؛ McN-JR 3345 ؛ R 3345) هو مضاد شديد التقارب لمستقبل 5-HT2A (pKi = 8.2) ومستقبل D4 (pKi = 8.0) ومضاد منخفض التقارب لمستقبل D2 (pKi = 6.7)
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Cas No.: 1893-33-0
Sample solution is provided at 25 µL, 10mM.
Pipamperone (Floropipamide; McN-JR 3345; R 3345) is a high-affinity antagonist of 5-HT2A receptor (pKi=8.2) and D4 receptor (pKi=8.0) and a low-affinity antagonist of D2 receptor (pKi=6.7)[1]. 5-HT2A Receptor|8.2 (pKi)|5-HT2C Receptor|6.9 (pKi)|5-HT1 Receptor|5.7 (pKi)|D4 receptor|8.0 (pKi)|D2 receptor|6.7 (pKi)|α1 receptor|7.2 (pKi)
[1]. Erik Buntinx, MD, et al. Selective Serotonergic Properties of Low-Dose Pipamperone May Enhance Antidepressant Effect: Preclinical Evidence.
Average Rating: 5
(Based on Reviews and 13 reference(s) in Google Scholar.)GLPBIO products are for RESEARCH USE ONLY. Please make sure your review or question is research based.
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