A2B receptor antagonist 2 |
Catalog No.GC62820 |
L'antagoniste 2 des récepteurs A2B (composé 18) est un antagoniste des récepteurs A2B de l'adénosine, avec des valeurs de Ki de 2,30 μM, 6,8 μM et 3,44 μM pour rA1, rA2A et hA2B, respectivement .
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Cas No.: 784-90-7
Sample solution is provided at 25 µL, 10mM.
A2B receptor antagonist 2 (compound 18) is an adenosine receptor A2B antagonist, with Ki values of 2.30 μM, 6.8 μM and 3.44 μM for rA1, rA2A and hA2B, respectively[1].
[1]. Thomas R Webb, et al. Quinazolines as adenosine receptor antagonists: SAR and selectivity for A2B receptors. Bioorg Med Chem. 2003 Jan 2;11(1):77-85.
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