L-838,417 |
Catalog No.GC11597 |
L-838,417 est un agoniste partiel sélectif au niveau des sous-types α2, α3 et α5 du récepteur GABAA et un antagoniste au niveau α1, avec des valeurs de Ki de liaison de 0,79 nM, 0,67 nM, 1,67 nM, 267 nM, 2,25 nM et 2183 nM pour α1β3γ2, α2β3γ2, α3β3γ2, α4β3γ2, α5β3γ2 et α6β3γ2.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 286456-42-6
Sample solution is provided at 25 µL, 10mM.
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