DREADD
Products for DREADD
- Cat.No. Nom du produit Informations
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GC43284
Clozapine N-oxide (hydrochloride)
CNO
Clozapine N-oxide is a major metabolite of clozapine and an activator of designer receptors exclusively activated by designer drugs (DREADDs) derived from human muscarinic acetylcholine receptors (EC50s = 16.7, 323, 17.4, 18.3, and 18.7 nM for PASMCs expressing hM1-5D receptors, respectively).