AGX51 |
Catalog No.GC38590 |
AGX51 es un antagonista y degradador pan-Id (inhibidores de proteÍnas de uniÓn/diferenciaciÓn de ADN) de primera clase. AGX51 inhibe la interacciÓn Id1-E47, lo que conduce a la degradaciÓn de Ids mediada por ubiquitina, la detenciÓn del crecimiento celular y reduce la viabilidad. AGX51 inhibe las lÍneas celulares TNBC con IC50 de casi 25 μM. AGX51 se puede utilizar para la investigaciÓn del cÁncer.
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Cas No.: 330834-54-3
Sample solution is provided at 25 µL, 10mM.
AGX51 is a first-in-class pan-Id (inhibitors of DNA-binding/differentiation proteins) antagonist and degrader. AGX51 inhibits the Id1-E47 interaction, leading to ubiquitin-mediated degradation of Ids, cell growth arrest, and reduces viability. AGX51 inhibits pathologic ocular neovascularization[1].
[1]. Wojnarowicz PM, et al. A Small-Molecule Pan-Id Antagonist Inhibits Pathologic Ocular Neovascularization. Cell Rep. 2019 Oct 1;29(1):62-75.e7.
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