IEM 1754 dihydrobroMide |
Catalog No.GC12198 |
El dihidrobromuro IEM 1754, un derivado de adamantano dicatiÓnico, es un potente bloqueador de los canales abiertos de los receptores de glutamato ionotrÓpicos nativos, incluidos los receptores sensibles al quiscualato en los mÚsculos de los insectos, NMDAR en neuronas corticales de rata cultivadas y AMPAR en células de hipocampo recién aisladas.
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Cas No.: 162831-31-4
Sample solution is provided at 25 µL, 10mM.
IEM 1754 dihydrobroMide is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM.
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