L 888607 Racemate |
| رقم الكتالوجGC31975 |
L 888607 Racemate هو مضاد انتقائي لمستقبل البروستاغلاندين D2 من النوع الفرعي 1 (DP1) ، مع Kis من 132 نانومتر و 17 نانومتر لمستقبل DP1 ومستقبل الثرموبوكسان A2 (TP) ، على التوالي
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Cas No.: 1030017-51-6
Sample solution is provided at 25 µL, 10mM.
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L 888607 Racemate is a selective prostaglandin D2 receptor subtype 1 (DP1) antagonist, with Kis of 132 nM and 17 nM for DP1 and thromboxane A2 receptor (TP), respectively.
L 888607 Racemate (compound 3) maintains a modest binding affinity for the DP1 receptor (Ki = 132 nM) and is actually 8-fold more potent on the TP receptor (Ki = 17 nM)[1].
[1]. Beaulieu C, et al. Identification of prostaglandin D2 receptor antagonists based on a tetrahydropyridoindole scaffold. Bioorg Med Chem Lett. 2008 Apr 15;18(8):2696-700.
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