BTR-1 |
Catalog No.GC34511 |
BTR-1 est un agent anticancéreux actif, provoque l'arrêt de la phase S et affecte la réplication de l'ADN dans les cellules leucémiques. BTR-1 active l'apoptose et induit la mort cellulaire.
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Cas No.: 18331-34-5
Sample solution is provided at 25 µL, 10mM.
BTR-1 is an active anti-cancer agent, causes S phase arrest, and affects DNA replication in leukemic cells. BTR-1 activates apoptosis and induces cell death[1]. Apoptosis[1]
BTR-1 (10, 50, 100, and 250 µM, 5 days) dose-dependently causes cytotoxicity in human leukemic cells, with IC50s of 8 and 6 µM at 48 and 72 h, respectively[1]. Cell Viability Assay[1] Cell Line: T-cell leukemic cell lines
[1]. Moorthy BT, et al. Novel rhodanine derivatives induce growth inhibition followed by apoptosis. Bioorg Med Chem Lett. 2010 Nov 1;20(21):6297-301.
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