hGPR91 antagonist 1 |
| Catalog No.GC36225 |
L'antagoniste 1 de HGPR91 est un antagoniste puissant et sélectif de hGPR91 À petite molécule avec une IC50 de 7 μM.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1314796-00-3
Sample solution is provided at 25 µL, 10mM.
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HGPR91 antagonist 1 is a potent and selective small molecule hGPR91 antagonist with an IC50 of 7 μM[1]. IC50: 7 μM (HGPR91)[1]
HGPR91 antagonist 1 leads to 59, 76% inhibition of δMAP at 2, 4 hours and has shown rat plasma protein binding 99%. HGPR91 antagonist 1 has engaged the target under the in vivo condition. HGPR91 antagonist 1 has clearance (CL) of 0.2 nmol/min/mg of RLM[1]. Animal Model: Wistar rats[1]
[1]. Bhuniya D, et al. Discovery of a potent and selective small molecule hGPR91 antagonist. Bioorg Med Chem Lett. 2011 Jun 15;21(12):3596-602.
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