LPA2 antagonist 1 (Synonyms: LPA2-IN-1) |
| Catalog No.GC12655 |
L'antagoniste LPA2 1 est un antagoniste LPA2 avec une IC50 de 17 nM.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1017606-66-4
Sample solution is provided at 25 µL, 10mM.
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LPA2 antagonist 1 is a LPA2 antagonist with an IC50 of 17 nM.
LPA2 antagonist 1 inhibits the phosphorylation of Erk induced by LPA in a concentration dependent manner. LPA2 antagonist 1 inhibits HCT-116 colon cancer cell proliferation caused by LPA in a doses dependent manner[1].
References:
[1]. Beck HP, et al. Discovery of potent LPA2 (EDG4) antagonists as potential anticancer agents. Bioorg Med Chem Lett. 2008 Feb 1;18(3):1037-41.
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