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(rel)-Tranylcypromine D5 hydrochloride

Catalog No.GC60004

Le chlorhydrate de tranylcypromine-d5 (SKF 385-d5) est un chlorhydrate de (rel)-tranylcypromine marqué au deutérium.

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(rel)-Tranylcypromine D5 hydrochloride Chemical Structure

Cas No.: 107077-98-5

Taille Prix Stock Qté
5mg
1 298,00 $US
En stock

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Sample solution is provided at 25 µL, 10mM.

Product Documents

Quality Control & SDS

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Background

(rel)-Tranylcypromine D5 hydrochloride (2-Phenylcyclopropylamine D5 hydrochloride) is a deuterium labeled (rel)-Tranylcypromine hydrochloride. (rel)-Tranylcypromine hydrochloride is an irreversible, nonselective monoamine oxidase (MAO) inhibitor used in the treatment of depression. (rel)-Tranylcypromine hydrochloride is also a lysine-specific demethylase 1 (LSD1) inhibitor, suppresses lesion growth and improves generalized hyperalgesia in mouse with induced endometriosis[1][2].

[1]. Caraci F, et al. Neuroprotective effects of the monoamine oxidase inhibitor tranylcypromine and its amide derivatives against Aβ(1-42)-induced toxicity. Eur J Pharmacol. 2015 Oct 5;764:256-263. [2]. Sun Q, et al. Tranylcypromine, a lysine-specific demethylase 1 (LSD1) inhibitor, suppresses lesion growth and improves generalized hyperalgesia in mouse with induced endometriosis. Reprod Biol Endocrinol. 2016 Apr 9;14:17.

Chemical Properties

Cas No. 107077-98-5 SDF
Canonical SMILES N[C@H]1[C@H](C2=C([2H])C([2H])=C([2H])C([2H])=C2[2H])C1.[H]Cl.[Relative stereochemistry]
Formula C9H7D5ClN M.Wt 174.68
Solubility Storage
General tips Please select the appropriate solvent to prepare the stock solution according to the solubility of the product in different solvents; once the solution is prepared, please store it in separate packages to avoid product failure caused by repeated freezing and thawing.Storage method and period of the stock solution: When stored at -80°C, please use it within 6 months; when stored at -20°C, please use it within 1 month.
To increase solubility, heat the tube to 37°C and then oscillate in an ultrasonic bath for some time.
Shipping Condition Evaluation sample solution: shipped with blue ice. All other sizes available: with RT, or with Blue Ice upon request.

Complete Stock Solution Preparation Table

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1 mg 5 mg 10 mg
1 mM 5.7248 mL 28.6238 mL 57.2475 mL
5 mM 1.145 mL 5.7248 mL 11.4495 mL
10 mM 0.5725 mL 2.8624 mL 5.7248 mL
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Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

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Review for (rel)-Tranylcypromine D5 hydrochloride

Average Rating: 5 ★★★★★ (Based on Reviews and 13 reference(s) in Google Scholar.)

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