GPCR/G protein
Research Areas
- Neuropeptide FF/AF Receptors(54)
- Neuropeptide S Receptor(3)
- GPBA Receptor(5)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(431)
- Acetylcholine(28)
- Adenosine Deaminase(10)
- Adenosine Receptor(143)
- Adenosine Kinase(5)
- Adiponectin Receptor(3)
- Adrenergic Receptor(449)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(118)
- Bombesin Receptors(26)
- Bradykinin Receptors(30)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(121)
- Calcimimetic Agent(2)
- CaSR(27)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(98)
- Chemokine Receptors(23)
- CRF1 Receptors(10)
- CRF2 Receptors(3)
- CXCR(106)
- CysLT1 receptor(1)
- Endothelin Receptor(54)
- EP1 Receptor(2)
- EP4 Receptor(2)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(16)
- Galanin Receptors(11)
- Ghrelin Receptors(11)
- GHSR(20)
- GIP Receptor(5)
- Glucagon Receptor(54)
- Glucocorticoid Receptor(102)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(11)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(57)
- LPA Receptor(12)
- LPL Receptor(64)
- LTD4 Receptor(1)
- mGluR (126)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(62)
- Melatonin Receptors(23)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(26)
- NK2 Receptors(7)
- NK3 Receptor(5)
- NOP Receptor(20)
- NPY Receptors(26)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(58)
- Oxytocin Receptors(22)
- P2Y Receptor(66)
- PACAP Receptors(7)
- PAF Receptors(7)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(179)
- Prostanoid Receptors(25)
- Protease-Activated Receptors(9)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(47)
- Sigma Receptor(62)
- Vasopressin Receptor(34)
- 17,20-lyase(4)
- Ras(180)
- Urotensin-II Receptor(10)
- VIP Receptors(6)
- EBI2/GPR183(7)
- TSH Receptor(12)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(11)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(8)
- CRFR(27)
- RGS Protein(5)
- Urotensin Receptor(7)
- Cholecystokinin Receptor(29)
- GPR139(4)
- mAChR(200)
- MCHR1 (GPR24)(17)
- Neurokinin Receptor(78)
- cGMP(27)
- GRK(5)
- GPR88(3)
- Amylin Receptor(9)
- Arrestin(10)
- Mas-related G-protein-coupled Receptor (MRGPR)(10)
- GCGR(12)
- GLP Receptor(27)
- Succinate Receptor 1(1)
- PTHR(3)
- Protease Activated Receptor (PAR)(6)
- Free Fatty Acid Receptor(5)
- Formyl Peptide Receptor (FPR)(7)
- Hydroxycarboxylic Acid Receptor (HCAR)(2)
- RXFP Receptor(3)
- Adhesion G Protein-coupled Receptors (AGPCRs)(1)
- Taste Receptor(1)
- GPR52(1)
Products Related to GPCR/G protein(3726)
- GC79316L-797591 hydrochlorideCAS: 3026641-74-4Purity: >99.50%
L-797591 hydrochloride is a selective sst 1 agonist.
- GC79317SSTR3 Agonist-1CAS: 3086695-73-7Purity: >98.00%
SSTR3 Agonist-1 (Compound EX 38) is an orally active SSTR3 agonist, with an EC 50 of 0.14 nM.
- GC79319R06039-641CAS: 2138444-75-2Purity: >98.50%
R06039-641 is a neuropeptide S receptor ( NPSR ) agonist with an EC 50 of 169 nM.
- GC79320R06039-691CAS: 2138445-51-7Purity: >99.50%
R06039-691 is a neuropeptide S receptor ( NPSR ) agonist with an EC 50 of 93 nM.
- GC79321MRS 2179 ammoniumPurity: >99.00%
MRS 2179 ammonium is a selective and competitive antagonist for P2Y1 receptor, with K B of 0.177 μM [1] .
- GC79322TP receptor antagonist-3CAS: 165537-72-4Purity: >99.50%
TP receptor antagonist-3 (compound 51280) is a potent thromboxane A2 prostanoid ( TP ) receptor with an IC 50 of 15.7 nM against Human TP.
- GC79323Terutroban sodiumCAS: 609340-89-8Purity: >98.00%
Terutroban (S-18886) sodium is a selective and orally active thromboxane-prostaglandin (TP) receptor antagonist with an IC 50 of 16.4 nM.
- GC79324HTL0039732CAS: 2639366-75-7Purity: >99.00%
HTL0039732 is an orally active antagonist of the prostaglandin EP4 receptor (Prostaglandin E2 Receptor EP4).
- GC79325ML161 analog 1CAS: 423740-83-4Purity: >99.50%
ML161 analog 1 (compound 38) is an analog of ML161.
- GC79326Tirzepatide sodiumPurity: >98.00%
Tirzepatide sodium (LY3298176 sodium) is a dual glucose-dependent insulinotropic polypeptide ( GIP ) and glucagon-like peptide-1 ( GLP-1 ) receptor agonist.
- GC79327BMS-986331CAS: 2375684-52-7Purity: >99.50%
BMS-986331 is an orally active selective N-Formyl Peptide Receptor 2 (FPR2) agonist with an EC 50 of 0.5 nM in humans and 1 nM in rats.
- GC79372Rosnilimab (Mouse IgG2a)Purity: >98.00%
Rosnilimab (Mouse IgG2a ) is a mouse-derived IgG2a antibody, Rosnilimab.
- GC79374PD-1/PD-L1-IN-63CAS: 2691796-92-4Purity: >98.00%
PD-1/PD-L1-IN-63 is an orally active PD-1/PD-L1 inhibitor with an IC 50 of 9.1 nM.
- GC79405TSLP modulator-1Purity: >99.50%
TSLP modulator-1 (Compound 14O) is a potent TSLP signaling modulator.
- GC79450Hydrocortisone-OVAPurity: >98.00%
Hydrocortisone -OVA is a conjugate of Hydrocortisone and OVA peptide.
- GC79504(R)-VerapamilCAS: 38321-02-7Purity: >98.50%
(R)-Verapamil (Dexverapamil) is an optically enantiomer of the oral-active Verapamil.
- GC79505RPI-GLYT2-82Purity: >99.00%
RPI-GLYT2-82 is a reversible, blood-brain barrier-permeable allosteric inhibitor of GlyT2 with an IC 50 value of 554 nM.
- GC79667AGFAGDDAPRCAS: 330204-04-1Purity: >98.00%
AGFAGDDAPR is a bioactive peptide that is a competitive and orally effective inhibitor of dipeptidyl peptidase-IV ( DPP-IV ).
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC79316 | L-797591 hydrochloride | 3026641-74-4 | >99.50% | |
L-797591 hydrochloride is a selective sst 1 agonist. | ||||
| GC79317 | SSTR3 Agonist-1 | 3086695-73-7 | >98.00% | |
SSTR3 Agonist-1 (Compound EX 38) is an orally active SSTR3 agonist, with an EC 50 of 0.14 nM. | ||||
| GC79318 | NOTA-TATE | 709043-21-0 | >98.50% | |
NOTA-TATE is a somatostatin receptor 2 ( SSTR2 ) binder. | ||||
| GC79319 | R06039-641 | 2138444-75-2 | >98.50% | |
R06039-641 is a neuropeptide S receptor ( NPSR ) agonist with an EC 50 of 169 nM. | ||||
| GC79320 | R06039-691 | 2138445-51-7 | >99.50% | |
R06039-691 is a neuropeptide S receptor ( NPSR ) agonist with an EC 50 of 93 nM. | ||||
| GC79321 | MRS 2179 ammonium | - | >99.00% | |
MRS 2179 ammonium is a selective and competitive antagonist for P2Y1 receptor, with K B of 0.177 μM [1] . | ||||
| GC79322 | TP receptor antagonist-3 | 165537-72-4 | >99.50% | |
TP receptor antagonist-3 (compound 51280) is a potent thromboxane A2 prostanoid ( TP ) receptor with an IC 50 of 15.7 nM against Human TP. | ||||
| GC79323 | Terutroban sodium | 609340-89-8 | >98.00% | |
Terutroban (S-18886) sodium is a selective and orally active thromboxane-prostaglandin (TP) receptor antagonist with an IC 50 of 16.4 nM. | ||||
| GC79324 | HTL0039732 | 2639366-75-7 | >99.00% | |
HTL0039732 is an orally active antagonist of the prostaglandin EP4 receptor (Prostaglandin E2 Receptor EP4). | ||||
| GC79325 | ML161 analog 1 | 423740-83-4 | >99.50% | |
ML161 analog 1 (compound 38) is an analog of ML161. | ||||
| GC79326 | Tirzepatide sodium | - | >98.00% | |
Tirzepatide sodium (LY3298176 sodium) is a dual glucose-dependent insulinotropic polypeptide ( GIP ) and glucagon-like peptide-1 ( GLP-1 ) receptor agonist. | ||||
| GC79327 | BMS-986331 | 2375684-52-7 | >99.50% | |
BMS-986331 is an orally active selective N-Formyl Peptide Receptor 2 (FPR2) agonist with an EC 50 of 0.5 nM in humans and 1 nM in rats. | ||||
| GC79328 | HDB-1 | 3021527-82-9 | >98.00% | |
HDB-1 is a selective inhibitor of the P2Y14 receptor ( P2Y14R ) with an IC 50 of 26 pM. | ||||
| GC79372 | Rosnilimab (Mouse IgG2a) | - | >98.00% | |
Rosnilimab (Mouse IgG2a ) is a mouse-derived IgG2a antibody, Rosnilimab. | ||||
| GC79373 | FK3453 | 560111-91-3 | >99.50% | |
FK3453 is a dual adenosine A1/A2 inhibitor and a TSLP inhibitor. | ||||
| GC79374 | PD-1/PD-L1-IN-63 | 2691796-92-4 | >98.00% | |
PD-1/PD-L1-IN-63 is an orally active PD-1/PD-L1 inhibitor with an IC 50 of 9.1 nM. | ||||
| GC79405 | TSLP modulator-1 | - | >99.50% | |
TSLP modulator-1 (Compound 14O) is a potent TSLP signaling modulator. | ||||
| GC79450 | Hydrocortisone-OVA | - | >98.00% | |
Hydrocortisone -OVA is a conjugate of Hydrocortisone and OVA peptide. | ||||
| GC79504 | (R)-Verapamil | 38321-02-7 | >98.50% | |
(R)-Verapamil (Dexverapamil) is an optically enantiomer of the oral-active Verapamil. | ||||
| GC79505 | RPI-GLYT2-82 | - | >99.00% | |
RPI-GLYT2-82 is a reversible, blood-brain barrier-permeable allosteric inhibitor of GlyT2 with an IC 50 value of 554 nM. | ||||
| GC79507 | PSB-12054 | 1407632-07-8 | >98.50% | |
PSB-12054 is a P2X4 receptor antagonist with IC 50 values of 0.19 μM, 2.10 μM and 1.77 μM against human, rat and mouse receptors, respectively, and exhibits selectivity over other human P2X receptor subtypes. | ||||
| GC79667 | AGFAGDDAPR | 330204-04-1 | >98.00% | |
AGFAGDDAPR is a bioactive peptide that is a competitive and orally effective inhibitor of dipeptidyl peptidase-IV ( DPP-IV ). | ||||
| GC79668 | RES-701-3 peptide TFA | - | >98.00% | |
RES-701-3 peptide TFA is a class II lasso peptide. | ||||
| GC79675 | FTO-IN-17 | 1434867-98-7 | >98.00% | |
FTO-IN-17 is an orally active and brain-penetrant FTO (m 6 A RNA demethylase) inhibitor with an IC 50 of 1.1 μM. | ||||