GPCR/G protein
Research Areas
- Neuropeptide FF/AF Receptors(52)
- Neuropeptide S Receptor(3)
- GPBA Receptor(5)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(429)
- Acetylcholine(28)
- Adenosine Deaminase(10)
- Adenosine Receptor(141)
- Adenosine Kinase(5)
- Adiponectin Receptor(3)
- Adrenergic Receptor(444)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(118)
- Bombesin Receptors(26)
- Bradykinin Receptors(30)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(121)
- Calcimimetic Agent(2)
- CaSR(27)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(97)
- Chemokine Receptors(23)
- CRF1 Receptors(10)
- CRF2 Receptors(3)
- CXCR(103)
- CysLT1 receptor(1)
- Endothelin Receptor(54)
- EP1 Receptor(2)
- EP4 Receptor(2)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(16)
- Galanin Receptors(11)
- Ghrelin Receptors(11)
- GHSR(20)
- GIP Receptor(5)
- Glucagon Receptor(54)
- Glucocorticoid Receptor(101)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(11)
- GPR120(9)
- GPR35(10)
- GPR44(1)
- GPR55(11)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(57)
- LPA Receptor(12)
- LPL Receptor(63)
- LTD4 Receptor(1)
- mGluR (125)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(60)
- Melatonin Receptors(23)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(26)
- NK2 Receptors(7)
- NK3 Receptor(5)
- NOP Receptor(20)
- NPY Receptors(26)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(57)
- Oxytocin Receptors(22)
- P2Y Receptor(66)
- PACAP Receptors(7)
- PAF Receptors(7)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(179)
- Prostanoid Receptors(25)
- Protease-Activated Receptors(9)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(47)
- Sigma Receptor(60)
- Vasopressin Receptor(34)
- 17,20-lyase(4)
- Ras(178)
- Urotensin-II Receptor(10)
- VIP Receptors(6)
- EBI2/GPR183(7)
- TSH Receptor(11)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(10)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(8)
- CRFR(27)
- RGS Protein(5)
- Urotensin Receptor(7)
- Cholecystokinin Receptor(28)
- GPR139(4)
- mAChR(196)
- MCHR1 (GPR24)(17)
- Neurokinin Receptor(78)
- cGMP(27)
- GRK(5)
- GPR88(2)
- Amylin Receptor(9)
- Arrestin(10)
- Mas-related G-protein-coupled Receptor (MRGPR)(9)
- GCGR(12)
- GLP Receptor(26)
- Succinate Receptor 1(1)
- PTHR(3)
- Protease Activated Receptor (PAR)(6)
- Free Fatty Acid Receptor(5)
- Formyl Peptide Receptor (FPR)(7)
- Hydroxycarboxylic Acid Receptor (HCAR)(2)
- RXFP Receptor(3)
- Adhesion G Protein-coupled Receptors (AGPCRs)(1)
- Taste Receptor(1)
- GPR52(1)
Products Related to GPCR/G protein(3690)
- GC81563GUB10194 acetatePurity: >98.50%
GUB10194 acetate is a fully potent and selective GPR10 agonist with an EC 50 of 15 nM.
- GC81565palm11-PrRP31 TFAPurity: >99.00%
palm11-PrRP31 TFA is a lipidized endogenous appetite inhibitory neuropeptide (PrRP) analogue.
- GC81566Ro 25-1553 TFAPurity: >99.00%
Ro 25-1553 TFA is a 31 amino acid vasoactive intestinal peptide (VIP) analog, that acts as an agonist for VIP2 receptor ( VPAC2 receptor ).
- GC81567Ro 25-1553 acetatePurity: >98.00%
Ro 25-1553 acetate is a selective VIP 2 receptor ( VPAC 2 receptor ) agonist.
- GC81677APJ receptor agonist 10 free baseCAS: 2415197-87-2Purity: >99.00%
APJ receptor agonist 10 free base is an agonist of the APJ Receptor.
- GC81693GPR52 agonist-4CAS: 1313195-88-8Purity: >98.00%
GPR52 agonist-4 (Compound 65) is a highly selective G-protein-coupled receptor GPR52 modulator.
- GC81704Ractopamine-d 6CAS: 1185177-97-2Purity: >98.00%
Ractopamine -d 6 is the deuterium labeled Ractopamine.
- GC81729Neuropeptide W-30 (rat) acetatePurity: >98.00%
Neuropeptide W-30 (rat) is an important stress mediator in the central nervous system that modulates the hypothalamus-pituitary-adrenal (HPA) axis and sympathetic outflow.
- GC817573-Ethoxy-5,6-dibromosalicylaldehydeCAS: 20041-64-9Purity: >99.50%
3-Ethoxy-5,6-dibromosalicylaldehyde is an IRE1/ERN1 inhibitor, with an IC 50 of 0.12 μM, a K i of 71-88 nM, and a K d of 100 nM against the ribonuclease activity of hIRE1α, as well as an IC 50 of 4.8 μM against yeast Ire1.
- GC81851Pancreatic Polypeptide, rat TFAPurity: >98.00%
Pancreatic Polypeptide, rat TFA (Rat pancreatic polypeptide TFA) is a rat-derived Pancreatic Polypeptide.
- GC81855(R)-RXFP2 agonist 2CAS: 3123585-08-7Purity: >98.00%
(R)-RXFP2 agonist 2 is the R-type isomer of RXFP2 agonist 2.
- GC81859TH-Z827 diTFAPurity: >98.00%
TH-Z827 diTFA is a selective KRAS G12D inhibitor that exhibits activity against GDP-bound and GMPPNP-bound KRAS G12D, but shows no activity against KRAS (WT) and KRAS G12C.
- GC81870Bethanidine hydriodideCAS: 2863-34-5Purity: >98.00%
Bethanidine hydriodide is an orally active antihypertensive agent and adrenergic neuron blocker.
- GC909521-Aminoguanosine-3',5'-monophosphate (sodium salt)CAS: 1380911-23-8Purity: >95.00%
cGMP-의존성 단백질 키나아제의 기질
| Catalog No. | Product Name | CAS No. | Purity | Structure |
|---|---|---|---|---|
| GC81563 | GUB10194 acetate | - | >98.50% | |
GUB10194 acetate is a fully potent and selective GPR10 agonist with an EC 50 of 15 nM. | ||||
| GC81564 | Z52 | 3077480-59-9 | >98.50% | |
Z52 is a Ras protein inhibitor. | ||||
| GC81565 | palm11-PrRP31 TFA | - | >99.00% | |
palm11-PrRP31 TFA is a lipidized endogenous appetite inhibitory neuropeptide (PrRP) analogue. | ||||
| GC81566 | Ro 25-1553 TFA | - | >99.00% | |
Ro 25-1553 TFA is a 31 amino acid vasoactive intestinal peptide (VIP) analog, that acts as an agonist for VIP2 receptor ( VPAC2 receptor ). | ||||
| GC81567 | Ro 25-1553 acetate | - | >98.00% | |
Ro 25-1553 acetate is a selective VIP 2 receptor ( VPAC 2 receptor ) agonist. | ||||
| GC81662 | nor-MC3 | 2870681-06-2 | >98.00% | |
nor-MC3 is an MC3 -type ionizable lipid with C 17 unsaturated chains, formulated in lipid nanoparticles for nucleic acid ( mRNA and siRNA) delivery and supports in vitro and in vivo transfection [1] . | ||||
| GC81677 | APJ receptor agonist 10 free base | 2415197-87-2 | >99.00% | |
APJ receptor agonist 10 free base is an agonist of the APJ Receptor. | ||||
| GC81693 | GPR52 agonist-4 | 1313195-88-8 | >98.00% | |
GPR52 agonist-4 (Compound 65) is a highly selective G-protein-coupled receptor GPR52 modulator. | ||||
| GC81704 | Ractopamine-d 6 | 1185177-97-2 | >98.00% | |
Ractopamine -d 6 is the deuterium labeled Ractopamine. | ||||
| GC81727 | HOR1-C59 | 189574-20-7 | >99.50% | |
HOR1-C59 is a highly selective Or5v1/Olfr110 agonist with an EC 50 of 7.12 nM. | ||||
| GC81728 | TTFB | 352560-76-0 | >98.00% | |
TTFB (N-(4-tert-butyl-1,3-thiazol-2-yl)-3-fluorobenzamide) is a selective, non-competitive zinc-activated channel ( ZAC ) antagonist. | ||||
| GC81729 | Neuropeptide W-30 (rat) acetate | - | >98.00% | |
Neuropeptide W-30 (rat) is an important stress mediator in the central nervous system that modulates the hypothalamus-pituitary-adrenal (HPA) axis and sympathetic outflow. | ||||
| GC81739 | LY 78335 | 39226-94-3 | >99.00% | |
LY 78335 (DCMB) is a brain-penetrant phenylethanolamine-N-methyltransferase ( PNMT ) inhibitor with a K i of 0.09 μM. | ||||
| GC81757 | 3-Ethoxy-5,6-dibromosalicylaldehyde | 20041-64-9 | >99.50% | |
3-Ethoxy-5,6-dibromosalicylaldehyde is an IRE1/ERN1 inhibitor, with an IC 50 of 0.12 μM, a K i of 71-88 nM, and a K d of 100 nM against the ribonuclease activity of hIRE1α, as well as an IC 50 of 4.8 μM against yeast Ire1. | ||||
| GC81769 | LP-856866 | - | >99.50% | |
LP-856866 is an orally active ACSL5 inhibitor, with IC 50 values of 8 nM and 4 nM against mouse and human ACSL5, respectively, and IC 50 values of 6 nM and 17 nM against mouse and human ACSL1, respectively. | ||||
| GC81824 | (+)-Talinolol | 71369-60-3 | >99.00% | |
(+)-Talinolol is an isomer of Talinolol. | ||||
| GC81851 | Pancreatic Polypeptide, rat TFA | - | >98.00% | |
Pancreatic Polypeptide, rat TFA (Rat pancreatic polypeptide TFA) is a rat-derived Pancreatic Polypeptide. | ||||
| GC81855 | (R)-RXFP2 agonist 2 | 3123585-08-7 | >98.00% | |
(R)-RXFP2 agonist 2 is the R-type isomer of RXFP2 agonist 2. | ||||
| GC81859 | TH-Z827 diTFA | - | >98.00% | |
TH-Z827 diTFA is a selective KRAS G12D inhibitor that exhibits activity against GDP-bound and GMPPNP-bound KRAS G12D, but shows no activity against KRAS (WT) and KRAS G12C. | ||||
| GC81870 | Bethanidine hydriodide | 2863-34-5 | >98.00% | |
Bethanidine hydriodide is an orally active antihypertensive agent and adrenergic neuron blocker. | ||||
| GC90924 | TNP-GTP (sodium salt) | - | >95.00% | |
GTP의 형광 유도체 | ||||
| GC90952 | 1-Aminoguanosine-3',5'-monophosphate (sodium salt) | 1380911-23-8 | >95.00% | |
cGMP-의존성 단백질 키나아제의 기질 | ||||
| GC91090 | Oxamyl-d6 | 2470229-60-6 | >99.00% | |
옥살닐 양량 측정을 위한 내부 표준제 | ||||
| GC91093 | MR2938 | 1044870-65-6 | >95.00% | |
AChE 억제제 | ||||
