CYN 154806 |
| Catalog No.GC14747 |
CYN 154806, un octapéptido cÍclico, es un potente y selectivo antagonista del receptor de somatostatina sst2, con valores de pIC50 de 8,58, 5,41, 6,07, 5,76 y 6,48 para los receptores recombinantes humanos sst2, sst1, sst3, sst4 y sst5 respectivamente .
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 183658-72-2
Sample solution is provided at 25 µL, 10mM.
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CYN 154806, a cyclic octapeptide, is a potent and selective somatostatin sst2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively[1][2].
References:
[1]. Bass RT, et al. Identification and characterization of novel somatostatin antagonists. Mol Pharmacol. 1996 Oct;50(4):709-15.
[2]. Feniuk W, et al. Selective somatostatin sst(2) receptor blockade with the novel cyclic octapeptide, CYN-154806. Neuropharmacology. 2000 Jun 8;39(8):1443-50.
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