GSK2018682 |
| Catalog No.GC31863 |
GSK2018682 es un agonista de los receptores S1P1 y S1P5 con pEC50 de 7,7 y 7,2, respectivamente, y no tiene actividad agonista frente a S1P2, S1P3 o S1P4 humanos.
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Cas No.: 1034688-30-6
Sample solution is provided at 25 µL, 10mM.
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GSK2018682 is an agonist for S1P1 and S1P5 receptor with pEC50s of 7.7 and 7.2, respectively, and has no agonist activity towards human S1P2, S1P3, or S1P4. GSK2018682 is used in the research of multiple sclerosis.
GSK2018682 is an agonist for S1P1 and S1P5 receptor with pEC50s of 7.7 and 7.2, respectively, and has no agonist activity towards human S1P2, S1P3, or S1P4[1].
[1]. Xu J, et al. Safety, pharmacokinetics, pharmacodynamics, and bioavailability of GSK2018682, a sphingosine-1-phosphate receptor modulator, in healthy volunteers. Clin Pharmacol Drug Dev. 2014 May;3(3):170-8.
Average Rating: 5 (Based on Reviews and 25 reference(s) in Google Scholar.)
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